Synthesis and antibacterial activity of C11, C12-cyclic urea analogues of ketolides

Bioorganic and Medicinal Chemistry Letters

Volumn 17, Issue 18, 2007, Pages 5013-5018

  Kaneko, Takushi ^a   McMillen, William ^a   Lynch, Meghan Keaney ^a  

^a PFIZER INC   (United States)

Author keywords

Cyclic urea; Haemophillus influenzae; Ketene acetal; Ketolide; Macrolide; Streptococcus pneumoniae; Streptococcus pyogenes; Telithromycin

Indexed keywords

KETOLIDE; TELITHROMYCIN; UREA DERIVATIVE;

ANTIBACTERIAL ACTIVITY; ARTICLE; DRUG RESEARCH; DRUG STRUCTURE; DRUG SYNTHESIS; HAEMOPHILUS INFLUENZAE; IN VITRO STUDY; MINIMUM INHIBITORY CONCENTRATION; NONHUMAN; STAPHYLOCOCCUS AUREUS; STEREOSPECIFICITY; STREPTOCOCCUS PNEUMONIAE; STREPTOCOCCUS PYOGENES; STRUCTURE ACTIVITY RELATION;

ANTI-BACTERIAL AGENTS; KETOLIDES; MICROBIAL SENSITIVITY TESTS; STREPTOCOCCUS PYOGENES; UREA;

STREPTOCOCCUS PNEUMONIAE; STREPTOCOCCUS PYOGENES;

EID: 34547875726     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2007.07.041     Document Type: Article

References (9)

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