Synthesis and bactericidal activities of novel pyrazole-1-carbothioamide derivatives

Frontiers of Chemistry in China

Volumn 2, Issue 3, 2007, Pages 311-314

  Liu, Xinhua ^a   Wang, Shifan ^b   Song, Baoan ^c  

^a ANHUI UNIVERSITY OF TECHNOLOGY   (China)

^b NANJING UNIVERSITY   (China)

^c BEIJING UNIVERSITY OF POSTS AND TELECOMMUNICATIONS   (China)

Author keywords

Bioactivity; Carbothioamide; Pyrazole

Indexed keywords

EID: 34547221914     PISSN: 16733495     EISSN: 16733614     Source Type: Journal    
DOI: 10.1007/s11458-007-0057-x     Document Type: Article

References (21)

1. Jennifer A T, Golebiowski A, Michael P. The development of new bicyclic pyrazole-based cytokine synthesis inhibitors. Bioorg Med Chem Lett, 2004, 14(19): 4945-4948
2. Sharp S, Boxall K, Matthews T. 347 Biological evaluation of a novel, synthetic pyrazole class of Hsp90 inhibitors. Eur J Cancer Suppl, 2004, 2(8): 105-108
3. Bekhit A A, Tarek A A. Design, synthesis and biological evaluation of some pyrazole derivatives as anti-inflammatoryantimicrobial agents. Bioorg Med Chem, 2004, 12(8): 1935-1945
4. Baraldi P G, Beria I, Cozzi P. Cinnamoyl nitrogen mustard derivatives of pyrazole analogues of tallimustine modified at the amidino moiety: Design, synthesis, molecular modeling and antitumor activity studies. Bioor Med Chem, 2004, 12(8): 3911-3921
5. John L K Jr., Bradford H. Ureas of 5-aminopyrazole and 2-aminothiazole inhibit growth of gram-positive bacteria. Bioorg Med Chem Lett, 2003, 13(24): 4463-4466
6. Kordik C P, Luo C, Brian C. Aminopyrazoles with high affinity for the human neuropeptide Y5 receptor. Bioorg Med Chem Lett, 2001, 11(17): 2283-2286
7. Michon V, Hervé du Penhoat C, Tombret F. Preparation, structural analysis and anticonvulsant activity of 3- and 5-aminopyrazole N-benzoyl derivatives. Eur J Med Chem, 1995, 30(2): 147-155
8. Liu Y, Ren J, Chen W Q, Jin G Y. Synthesis of N-(substituted) pyrazolylmethene imino-N'- (substituted) phenyl (thio) Ur. Chin J Appl Chem, 2001, 18(7): 513 (in Chinese)
9. Fan Z J, Zhong B, Wang S H, Li Z M. Synthesis and fungicidal activity of derivatives of 1, 3-dimethyl-5-methylthio-4-phenylhydrazonocarboxyl pyrazole. Chin J Appl Chem, 2003, 20(4): 365 (in Chinese)
10. Sova V K, Svoboda M, Waisser K. Synthesis of 2-benzylthi opyridine-4-carbothioamide derivatives and their antimycobacterial, antifungal and photosynthesis-inhibiting activity. Eur J Med Chem, 1999, 34(5): 433-440
11. Liu X H, Bau L S, Wang S F. Synthesis and antibacterial activity of 5-(2-hydroxyphenyl)-3-methyl aminopyrazole. Chin J Synth Chem, 2006, 14(2): 147-149 (in Chinese)
12. Liu X H, Bau L S, Wang S F. Synthesis of 5-(2-hydroxy-6-methoxylphenyl)- 3-methyl-4, 5-dihydropyrazole-1-carbothioamide derivatives. Chin J Synth Chem, 2006, 14(3): 272-274 (in Chinese)
13. Liu X H. Synthesis and fungicide activity of novel arylpyrazole derivatives. Chin J Synth Chem, 2007, 15(2): in press (in Chinese)
14. Liu X H, Song B A. Synthesis and fungicide activity of novel 3,5-diarylpyrazole derivatives. Chin J Appl Chem, 2007, 24(7): in press (in Chinese)
15. Liu X H, Zhu J, Pan C X, Song B A. Synthesis and fungicide activity of novel J-arylpyrazole derivatives. Chin J Appl Chem, 2007, 24(8): in press (in Chinese)
16. Liu X H. Synthesis and characterize of 5-(2-hydroxy-6-methoxylphenyl)-3- methyl aminopyrazole. J Anhui Univ Technol, 2006, 23(3): 275-277 (in Chinese)
17. Svetlic J, Hanus V, Bella J. Extend oxygen-bridged pyridines and pyrimi-dines. J Chem Res (s), 1991, : 4-5
18. Svetlic J, Liptaj T. Novel heterocycle containing the pyrazole unit. J Chem Soc Perkin Transi, 2002, : 1260-1265
19. Finkelstein B L, Benner E A, Hendrixson M C, Kranis K T, Rauh J J, Sethuraman M R, McCann S F. Tricyclic cyanoguanidines: Synthesis, site of action and insecticidal activity of a novel class of reversible acetylcholinesterase inhibitors. Bioorg Med Chem, 2002, 10: 599-613
20. Zhang Z Y, Zhang Y, Hui X P, Xu P F, Shen D P. Achievements on the application of hydrazine and related compounds for the synthesis of five membered azole heterocycles. Chin J Org Chem, 2004, 24(11): 1348-1365 (in Chinese)
21. Song B A, Liu X H, Yang S, Hu D Y, Jin L H, Zhang H. Synthesis and anticancer activity of 2,3,4-trimethoxyacetophenoxime ester containing benzothiazole moiety. Chin J Chem, 2005, 23(9): 1236-1240 (in Chinese)