Classification of anti-estrogens according to intramolecular FRET effects on phospho-mutants of estrogen receptor α

Molecular Cancer Therapeutics

Volumn 6, Issue 5, 2007, Pages 1526-1533

  Zwart, Wilbert ^a   Griekspoor, Alexander ^a   Rondaij, Mariska ^a   Verwoerd, Desiree ^a   Neefjes, Jacques ^a   Michalides, Rob ^a  

^a NETHERLANDS CANCER INSTITUTE   (Netherlands)

Author keywords

[No Author keywords available]

Indexed keywords

ACOLBIFENE; ANTIESTROGEN; CYCLIC AMP DEPENDENT PROTEIN KINASE; ESTROGEN RECEPTOR ALPHA; FULVESTRANT; MITOGEN ACTIVATED PROTEIN KINASE; N BUTYL 11 (3,17BETA DIHYDROXYESTRA 1,3,5(10) TRIEN 7ALPHA YL) N METHYLUNDECANAMIDE; TAMOXIFEN;

ARTICLE; BREAST CANCER; CONTROLLED STUDY; DRUG MECHANISM; ENZYME ACTIVITY; ENZYME ANALYSIS; ENZYME PHOSPHORYLATION; FLUORESCENCE RESONANCE ENERGY TRANSFER; HORMONAL THERAPY; HORMONE ACTION; HORMONE BINDING; HUMAN; HUMAN CELL; PRIORITY JOURNAL; PROTEIN CONFORMATION; PROTEIN MODIFICATION;

BACTERIAL PROTEINS; CELL LINE, TUMOR; ESTRADIOL; ESTROGEN ANTAGONISTS; ESTROGEN RECEPTOR ALPHA; ESTROGENS; FLUORESCENCE RESONANCE ENERGY TRANSFER; HUMANS; LUMINESCENT PROTEINS; MODELS, BIOLOGICAL; MODELS, CHEMICAL; MUTATION; PIPERIDINES; TAMOXIFEN; TRANS-ACTIVATION (GENETICS);

EID: 34250723932     PISSN: 15357163     EISSN: None     Source Type: Journal    
DOI: 10.1158/1535-7163.MCT-06-0750     Document Type: Article

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