Scintillation proximity assay for measuring uptake by the human drug transporters hOCT1, hOAT3, and hOATP1B1

Analytical Biochemistry

Volumn 366, Issue 2, 2007, Pages 117-125

  Lohmann, Christina ^a   Gelius, Birgitta ^b   Danielsson, Jeanette ^b   Skoging Nyberg, Ulrica ^b   Hollnack, Evelyn ^a   Dudley, Adam ^c   Wahlberg, Johanna ^b   Hoogstraate, Janet ^b   Gustavsson, Lena ^a  

^a ASTRAZENECA R AND D   (Sweden)

^b ASTRAZENECA R AND D   (Sweden)

^c ASTRAZENECA   (United Kingdom)

Author keywords

Drug; hOAT3; hOATP1B1; hOCT1; Scintillation proximity; Transporter

Indexed keywords

AMMONIUM COMPOUNDS; DRUG PRODUCTS; SUBSTRATES; SULFUR COMPOUNDS;

DRUG; HOAT3; HOATP1B1; HOCT1; TRANSPORTER;

SCINTILLATION;

ESTRONE SULFATE; FUROSEMIDE; IBUPROFEN; METHYLPHENYLPYRIDINIUM; ORGANIC ANION TRANSPORTER 1; ORGANIC CATION TRANSPORTER 1; ORGANIC CATION TRANSPORTER 3; PYRIDINIUM DERIVATIVE; RADIOISOTOPE; TETRYLAMMONIUM; UNCLASSIFIED DRUG;

ARTICLE; CELL STRAIN HEK293; CONCENTRATION RESPONSE; CONTROLLED STUDY; EMBRYO; GENETIC TRANSFECTION; HUMAN; HUMAN CELL; INFRARED RADIATION; PRIORITY JOURNAL; PROTEIN ANALYSIS; PROTEIN DETERMINATION; PROTEIN TRANSPORT; SCINTILLATION;

AVENA;

EID: 34250347331     PISSN: 00032697     EISSN: 10960309     Source Type: Journal    
DOI: 10.1016/j.ab.2007.04.038     Document Type: Article

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