메뉴 건너뛰기




Volumn 51, Issue 4, 2007, Pages 1473-1480

Interpretation of genotype and pharmacokinetics for resistance to fosamprenavir-ritonavir-based regimens in antiretroviral-experienced patients

Author keywords

[No Author keywords available]

Indexed keywords

ABACAVIR; ALANINE; AMPRENAVIR PHOSPHATE; ARGININE; ATAZANAVIR; CD4 ANTIGEN; CYSTEINE; EMTRICITABINE; ENFUVIRTIDE; GLUTAMIC ACID; ISOLEUCINE; LAMIVUDINE; LEUCINE; LOPINAVIR; LOPINAVIR PLUS RITONAVIR; LYSINE; METHIONINE; PHENYLALANINE; PROLINE; PROTEINASE; RITONAVIR; RNA DIRECTED DNA POLYMERASE; SAQUINAVIR; TENOFOVIR; TENOFOVIR DISOPROXIL; VALINE; VIRUS ENZYME; ZIDOVUDINE;

EID: 34247147510     PISSN: 00664804     EISSN: None     Source Type: Journal    
DOI: 10.1128/AAC.00481-06     Document Type: Article
Times cited : (22)

References (44)
  • 3
    • 34247155889 scopus 로고    scopus 로고
    • Breilh, D., I. Pellegrin, G. Coureau, J. B. Gordien, D. Lacoste, J. L. Pellegrin, D. Neau, M. Dupon, H. J. A. Fleury, M. C. Saux, and the GECSA. 2005. Switch to fosamprenavir/ritonavir (FPV/r) based HAART in experienced patients with virological failure on HAART (ZEPHIR study): impact of pharmacokinetics on response at M3. 45th Intersci. Conf. Antimicrob. Agents Chemother., abstr. H-1903.
    • Breilh, D., I. Pellegrin, G. Coureau, J. B. Gordien, D. Lacoste, J. L. Pellegrin, D. Neau, M. Dupon, H. J. A. Fleury, M. C. Saux, and the GECSA. 2005. Switch to fosamprenavir/ritonavir (FPV/r) based HAART in experienced patients with virological failure on HAART (ZEPHIR study): impact of pharmacokinetics on response at M3. 45th Intersci. Conf. Antimicrob. Agents Chemother., abstr. H-1903.
  • 6
  • 7
    • 34247093938 scopus 로고    scopus 로고
    • DeJesus, E., A. Lamarca, M. Sension, C. Beltran, and P. Yeni. 2003. The context study: efficacy and safety of GW433908/RTV in PI-experienced subjects with virological failure (24 week results) 10th Conf. Retrovir. Opportun. Infect., abstr. 178.
    • DeJesus, E., A. Lamarca, M. Sension, C. Beltran, and P. Yeni. 2003. The context study: efficacy and safety of GW433908/RTV in PI-experienced subjects with virological failure (24 week results) 10th Conf. Retrovir. Opportun. Infect., abstr. 178.
  • 8
    • 0003468344 scopus 로고    scopus 로고
    • Prise en charge thérapeutique des personnes infectées par le VIH, recommandations du groupe d'experts
    • Paris, France
    • Delfraissy, J. F. 2004. Prise en charge thérapeutique des personnes infectées par le VIH, recommandations du groupe d'experts. Editions Flammarion: Medecine-Sciences, Paris, France.
    • (2004) Editions Flammarion: Medecine-Sciences
    • Delfraissy, J.F.1
  • 10
    • 0036148608 scopus 로고    scopus 로고
    • Amprenavir inhibitory quotient and virological response in human immunodeficiency virus-infected patients on an amprenavir-containing salvage regimen without or with ritonavir
    • Duval, X., C. Lamotte, E. Race, D. Descamps, F. Damond, F. Clavel, C. Leport, G. Peytavin, and J. L. Vilde. 2002. Amprenavir inhibitory quotient and virological response in human immunodeficiency virus-infected patients on an amprenavir-containing salvage regimen without or with ritonavir. Antimicrob. Agents Chemother. 46:570-574.
    • (2002) Antimicrob. Agents Chemother , vol.46 , pp. 570-574
    • Duval, X.1    Lamotte, C.2    Race, E.3    Descamps, D.4    Damond, F.5    Clavel, F.6    Leport, C.7    Peytavin, G.8    Vilde, J.L.9
  • 12
    • 3843151487 scopus 로고    scopus 로고
    • SOLO: 48-week efficacy and safety comparison of once-daily fosamprenavir/ritonavir versus twice-daily nelfinavir in naive HIV-1-infected patients
    • Gathe, J. C., P. Ive, R. Wood, D. Schurmannd, N. C. Bellos, E. DeJesus, A. Gladysz, C. Garris, and J. Yeo. 2004. SOLO: 48-week efficacy and safety comparison of once-daily fosamprenavir/ritonavir versus twice-daily nelfinavir in naive HIV-1-infected patients. AIDS 18:1529-1537.
    • (2004) AIDS , vol.18 , pp. 1529-1537
    • Gathe, J.C.1    Ive, P.2    Wood, R.3    Schurmannd, D.4    Bellos, N.C.5    DeJesus, E.6    Gladysz, A.7    Garris, C.8    Yeo, J.9
  • 16
    • 0034129696 scopus 로고    scopus 로고
    • Population pharmacokinetics/pharmacodynamics modeling: Parametric and nonparametric methods
    • Jelliffe, R., A. Schumitzky, and M. Van Guilder. 2000. Population pharmacokinetics/pharmacodynamics modeling: parametric and nonparametric methods. Ther. Drug Monit. 22:354-365.
    • (2000) Ther. Drug Monit , vol.22 , pp. 354-365
    • Jelliffe, R.1    Schumitzky, A.2    Van Guilder, M.3
  • 18
    • 33750570685 scopus 로고    scopus 로고
    • Pharmacokinetics and safety of tenofovir disoproxil fumarate on coadministration with lopinavir/ritonavir
    • Kearney, B. P., A. Mathias, A. Mittan, J. Sayre, R. Ebrahimi, and A. K. Cheng. 2006. Pharmacokinetics and safety of tenofovir disoproxil fumarate on coadministration with lopinavir/ritonavir. J. Acquir. Immune Defic. Syndr. 43:278-283.
    • (2006) J. Acquir. Immune Defic. Syndr , vol.43 , pp. 278-283
    • Kearney, B.P.1    Mathias, A.2    Mittan, A.3    Sayre, J.4    Ebrahimi, R.5    Cheng, A.K.6
  • 19
    • 9644272512 scopus 로고    scopus 로고
    • Clinically relevant interpretation of genotype and relationship to plasma drug concentrations for resistance to saquinavir-ritonavir in human immunodeficiency virus type 1 protease inhibitor-experienced patients
    • Marcelin, A. G., C. Dalban, G. Peytavin, C. Lamotte, R. Agher, C. Delaugerre, M. Wirden, F. Conan, S. Dantin, C. Katlama, D. Costagliola, and V. Calvez. 2004. Clinically relevant interpretation of genotype and relationship to plasma drug concentrations for resistance to saquinavir-ritonavir in human immunodeficiency virus type 1 protease inhibitor-experienced patients. Antimicrob. Agents Chemother. 48:4687-4692.
    • (2004) Antimicrob. Agents Chemother , vol.48 , pp. 4687-4692
    • Marcelin, A.G.1    Dalban, C.2    Peytavin, G.3    Lamotte, C.4    Agher, R.5    Delaugerre, C.6    Wirden, M.7    Conan, F.8    Dantin, S.9    Katlama, C.10    Costagliola, D.11    Calvez, V.12
  • 20
    • 0037308542 scopus 로고    scopus 로고
    • Marcelin, A. G., C. Lamotte, C. Delaugerre, N. Ktorza, H. Ait Mohand, R. Cacace, M. Bonmarchand, M. Wirden, A. Simon, P. Bossi, F. Bricaire, D. Costagliola, C. Katlama, G. Peytavin, V. Calvez, and the Genophar Study Group. 2003. Genotypic inhibitory quotient as predictor of virological re-sponse to ritonavir-amprenavir in human immunodeficiency virus type 1 protease inhibitor-experienced patients. Antimicrob. Agents Chemother. 47:594-600.
    • Marcelin, A. G., C. Lamotte, C. Delaugerre, N. Ktorza, H. Ait Mohand, R. Cacace, M. Bonmarchand, M. Wirden, A. Simon, P. Bossi, F. Bricaire, D. Costagliola, C. Katlama, G. Peytavin, V. Calvez, and the Genophar Study Group. 2003. Genotypic inhibitory quotient as predictor of virological re-sponse to ritonavir-amprenavir in human immunodeficiency virus type 1 protease inhibitor-experienced patients. Antimicrob. Agents Chemother. 47:594-600.
  • 22
    • 0037470276 scopus 로고    scopus 로고
    • Methods for categorizing a prognostic variable in a multivariable setting
    • Mazumdar, M., A. Smith, and J. Bacik. 2003. Methods for categorizing a prognostic variable in a multivariable setting. Stat. Med. 22:559-571.
    • (2003) Stat. Med , vol.22 , pp. 559-571
    • Mazumdar, M.1    Smith, A.2    Bacik, J.3
  • 23
    • 34247162386 scopus 로고    scopus 로고
    • Parikh, U., C. Calef, B. A. Larder, R. Schinazi, and J. W. Mellors. 2002. Mutations in retroviral genes associated with drug resistance, p. 95-183. In C. Kuiken, B. Foley, E. Freed, B. Hahn, B. Korber, P. Marx, F. McCutchan, and J. W. Mellors (ed.), HIV sequence compendium 2002. Theoretical Biology and Biophysics Group, Los Alamos National Laboratory, Los Alamos, NM.
    • Parikh, U., C. Calef, B. A. Larder, R. Schinazi, and J. W. Mellors. 2002. Mutations in retroviral genes associated with drug resistance, p. 95-183. In C. Kuiken, B. Foley, E. Freed, B. Hahn, B. Korber, P. Marx, F. McCutchan, and J. W. Mellors (ed.), HIV sequence compendium 2002. Theoretical Biology and Biophysics Group, Los Alamos National Laboratory, Los Alamos, NM.
  • 24
    • 0038555736 scopus 로고    scopus 로고
    • Improving lopinavir genotype algorithm through phenotype correlations: "novel" mutation patterns and amprenavir cross-resistance
    • Parkin, N. T., C. Chappey, and C. J. Petropoulos. 2003. Improving lopinavir genotype algorithm through phenotype correlations: "novel" mutation patterns and amprenavir cross-resistance. AIDS 17:955-961.
    • (2003) AIDS , vol.17 , pp. 955-961
    • Parkin, N.T.1    Chappey, C.2    Petropoulos, C.J.3
  • 25
    • 34247141593 scopus 로고    scopus 로고
    • Parks, D. A., H. C. Jennings, C. W. Taylor, and E. D. Acosta. 2005. Pharmacokinetics of fosamprenavir, ritonavir, tenofovir and emtricitabine administered once daily in treament naive HIV-infected subjects. 3rd Int. AIDS Soc. Conf., abstr. TuPeLB3.1B.01.23001.
    • Parks, D. A., H. C. Jennings, C. W. Taylor, and E. D. Acosta. 2005. Pharmacokinetics of fosamprenavir, ritonavir, tenofovir and emtricitabine administered once daily in treament naive HIV-infected subjects. 3rd Int. AIDS Soc. Conf., abstr. TuPeLB3.1B.01.23001.
  • 26
    • 0034838469 scopus 로고    scopus 로고
    • Comparison of capillary electrophoresis sequencing with the new CEQ32000 System (Beckman Coulter Inc.) to conventional gel based systems for HIV-1 drug resistance analysis
    • Pellegrin, I., P. Merel, I. Garrigue, A. Caumont, M. H. Schrive, V. Birac, P. Bonot, and H. J. A. Fleury. 2001. Comparison of capillary electrophoresis sequencing with the new CEQ32000 System (Beckman Coulter Inc.) to conventional gel based systems for HIV-1 drug resistance analysis. J. Virol. Methods 98:9-16.
    • (2001) J. Virol. Methods , vol.98 , pp. 9-16
    • Pellegrin, I.1    Merel, P.2    Garrigue, I.3    Caumont, A.4    Schrive, M.H.5    Birac, V.6    Bonot, P.7    Fleury, H.J.A.8
  • 27
    • 34247117921 scopus 로고    scopus 로고
    • Pellegrin, I., G. Coureau, D. Neau, D. Lacoste, E. Lazaro, H. J. A. Fleury, D. Breilh, and the GECSA. 2005. Impact of protease drug mutations and pharmacokinetics on virological response to fosamprenavir/r-based HAART in antiretroviral-experienced patients (Zephir study). 45th Intersci. Conf. Antimicrob. Agents Chemother., abstr. H-1059.
    • Pellegrin, I., G. Coureau, D. Neau, D. Lacoste, E. Lazaro, H. J. A. Fleury, D. Breilh, and the GECSA. 2005. Impact of protease drug mutations and pharmacokinetics on virological response to fosamprenavir/r-based HAART in antiretroviral-experienced patients (Zephir study). 45th Intersci. Conf. Antimicrob. Agents Chemother., abstr. H-1059.
  • 31
    • 34247117920 scopus 로고    scopus 로고
    • Peytavin, G., A. G. Marcelin, A. Rouault, R. Agher, D. Descamps, V. Calvez, and C. Katlama. 2005. Plasma concentrations of amprenavir, ritonavir and tenofovir in HIV-infected patients treated with fosamprenavir/ritonavir (700/ 100 mg BID) and tenofovir (300 mg QD) containing regimen. 6th Int. Workshop Clin. Pharmacology HIV Ther., abstr. 2.25.
    • Peytavin, G., A. G. Marcelin, A. Rouault, R. Agher, D. Descamps, V. Calvez, and C. Katlama. 2005. Plasma concentrations of amprenavir, ritonavir and tenofovir in HIV-infected patients treated with fosamprenavir/ritonavir (700/ 100 mg BID) and tenofovir (300 mg QD) containing regimen. 6th Int. Workshop Clin. Pharmacology HIV Ther., abstr. 2.25.
  • 32
    • 0347990584 scopus 로고    scopus 로고
    • The NEAT study: A 48-week open label study to compare the antiviral efficacy and safety of GW433908 versus nelfinavir in antiretroviral therapy-naive HIV-1 infected patients
    • Rodriguez-French, A., J. Boghossian, G. E. Gray, J. P. Nadler, A. R. Quinones, G. E. Sepulveda, J. M. Millard, and P. G. Wannamaker. 2004. The NEAT study: a 48-week open label study to compare the antiviral efficacy and safety of GW433908 versus nelfinavir in antiretroviral therapy-naive HIV-1 infected patients. J. Acquir. Immune Defic. Syndr. 35:22-32.
    • (2004) J. Acquir. Immune Defic. Syndr , vol.35 , pp. 22-32
    • Rodriguez-French, A.1    Boghossian, J.2    Gray, G.E.3    Nadler, J.P.4    Quinones, A.R.5    Sepulveda, G.E.6    Millard, J.M.7    Wannamaker, P.G.8
  • 33
    • 0006179308 scopus 로고    scopus 로고
    • Pharmacokinetics and safety of amprenavir and ritonavir following multiple-dose, co-administration to healthy volunteers
    • Sadler, B. M., P. J. Piliero, S. L. Preston, P. P. Lloyd, Y. Lou, and D. S. Stein. 2001. Pharmacokinetics and safety of amprenavir and ritonavir following multiple-dose, co-administration to healthy volunteers. AIDS 15:1009-1018.
    • (2001) AIDS , vol.15 , pp. 1009-1018
    • Sadler, B.M.1    Piliero, P.J.2    Preston, S.L.3    Lloyd, P.P.4    Lou, Y.5    Stein, D.S.6
  • 34
    • 0036173443 scopus 로고    scopus 로고
    • Pharmacokinetic modeling and simulations of interaction of amprenavir and ritonavir
    • Sale, M., B. M. Sadler, and D. S. Stein. 2002. Pharmacokinetic modeling and simulations of interaction of amprenavir and ritonavir. Antimicrob. Agents Chemother. 46:746-754.
    • (2002) Antimicrob. Agents Chemother , vol.46 , pp. 746-754
    • Sale, M.1    Sadler, B.M.2    Stein, D.S.3
  • 35
    • 29144434086 scopus 로고    scopus 로고
    • Evolution of resistance during first-line treatment with boosted fosamprenavir is associated with baseline mutations
    • Shurmann, D., R. Elston, F. Xu, N. Kleinkauf, T. Wunsche, and N. Suttorp. 2006. Evolution of resistance during first-line treatment with boosted fosamprenavir is associated with baseline mutations. AIDS 2:138-140.
    • (2006) AIDS , vol.2 , pp. 138-140
    • Shurmann, D.1    Elston, R.2    Xu, F.3    Kleinkauf, N.4    Wunsche, T.5    Suttorp, N.6
  • 37
    • 2542502584 scopus 로고    scopus 로고
    • Taburet, A. M., C. Piketty, C. Chazallon, I. Vincent, L. Gérard, V. Calvez, F. Clavel, J. P. Aboulker, P. M. Girard, and the ANRS Protocol 107 Puzzle 2 Investigators. 2004. Interactions between atazanavir-ritonavir and tenofovir in heavily pretreated human immunodeficiency virus-infected patients. Antimicrob. Agents Chemother. 48:2091-2096.
    • Taburet, A. M., C. Piketty, C. Chazallon, I. Vincent, L. Gérard, V. Calvez, F. Clavel, J. P. Aboulker, P. M. Girard, and the ANRS Protocol 107 Puzzle 2 Investigators. 2004. Interactions between atazanavir-ritonavir and tenofovir in heavily pretreated human immunodeficiency virus-infected patients. Antimicrob. Agents Chemother. 48:2091-2096.
  • 38
    • 0034119111 scopus 로고    scopus 로고
    • Clinical progression of HIV-1 infection according to the viral response during the first year of antiretroviral treatment
    • Thiébaut, R., P. Morlat, H. Jacqmin-Gadda, D. Neau, P. Mercié, F. Dabis, and G. Chene. 2000. Clinical progression of HIV-1 infection according to the viral response during the first year of antiretroviral treatment. AIDS 14:971-978.
    • (2000) AIDS , vol.14 , pp. 971-978
    • Thiébaut, R.1    Morlat, P.2    Jacqmin-Gadda, H.3    Neau, D.4    Mercié, P.5    Dabis, F.6    Chene, G.7
  • 39
    • 27744600007 scopus 로고    scopus 로고
    • Predictive value of drug levels, HIV genotyping, and the genotypic inhibitory quotient (GIQ) on response to saquinavir/ritonavir in antiretroviral-experienced HIV-infected patients
    • Valer, L., C. De Mendoza, and V. Soriano. 2005. Predictive value of drug levels, HIV genotyping, and the genotypic inhibitory quotient (GIQ) on response to saquinavir/ritonavir in antiretroviral-experienced HIV-infected patients. J. Med. Virol. 77:460-464.
    • (2005) J. Med. Virol , vol.77 , pp. 460-464
    • Valer, L.1    De Mendoza, C.2    Soriano, V.3
  • 40
    • 29144526047 scopus 로고    scopus 로고
    • Vora, S., A. G. Marcelin H. Günthard, P. Flandre, H. H. Hirsch, B. Masquelier, A. Zinkernagel, G. Peytavin, V. Calvez, L. Perrin, and S. Yerly; Swiss HIV Cohort Study. 2006. Clinical validation of atazanavir/ritonavir genotypic resistance score in protease inhibitor-experienced patients. AIDS 20:35-40.
    • Vora, S., A. G. Marcelin H. Günthard, P. Flandre, H. H. Hirsch, B. Masquelier, A. Zinkernagel, G. Peytavin, V. Calvez, L. Perrin, and S. Yerly; Swiss HIV Cohort Study. 2006. Clinical validation of atazanavir/ritonavir genotypic resistance score in protease inhibitor-experienced patients. AIDS 20:35-40.
  • 41
    • 33645789309 scopus 로고    scopus 로고
    • Ritonavir increases plasma amprenavir (APV) exposure to a similar extent when coadministered with either fosamprenavir or APV
    • Wire, M. B., K. L. Baker, L. S. Jones, M. J. Shelton, Y. Lou, G. J. Thomas, and M. M. Berrey. 2006. Ritonavir increases plasma amprenavir (APV) exposure to a similar extent when coadministered with either fosamprenavir or APV. Antimicrob. Agents Chemother. 50:1578-1580.
    • (2006) Antimicrob. Agents Chemother , vol.50 , pp. 1578-1580
    • Wire, M.B.1    Baker, K.L.2    Jones, L.S.3    Shelton, M.J.4    Lou, Y.5    Thomas, G.J.6    Berrey, M.M.7
  • 42
    • 33344460707 scopus 로고    scopus 로고
    • Fosamprenavir: Clinical pharmacokinetics and drug interactions of the amprenavir prodrug
    • Wire, M. B., M. J. Shelton, and S. Studenberg. 2006. Fosamprenavir: clinical pharmacokinetics and drug interactions of the amprenavir prodrug. Clin. Pharmacokinet. 45:137-168.
    • (2006) Clin. Pharmacokinet , vol.45 , pp. 137-168
    • Wire, M.B.1    Shelton, M.J.2    Studenberg, S.3
  • 44
    • 20244387096 scopus 로고    scopus 로고
    • Mutation patterns and structural correlates in human immunodeficiency virus type 1 protease following different protease inhibitor treatments
    • Wu, T. D., C. A. Schiffer, M. J. Gonzales, J. Taylor, R. Kantor, S. Chou, D. Israelski, A. R. Zolopa, W. J. Fessel, and R. W. Shafer. 2003. Mutation patterns and structural correlates in human immunodeficiency virus type 1 protease following different protease inhibitor treatments. J. Virol. 77:4836-4847.
    • (2003) J. Virol , vol.77 , pp. 4836-4847
    • Wu, T.D.1    Schiffer, C.A.2    Gonzales, M.J.3    Taylor, J.4    Kantor, R.5    Chou, S.6    Israelski, D.7    Zolopa, A.R.8    Fessel, W.J.9    Shafer, R.W.10


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.