Assay optimization and kinetic profile of the human and the rabbit isoforms of 11β-HSD1

Biochemical and Biophysical Research Communications

Volumn 357, Issue 2, 2007, Pages 561-566

  Castro, Arturo ^a   Zhu, Jeff X ^a   Alton, Gordon R ^a   Rejto, Paul ^a   Ermolieff, Jacques ^a  

^a PFIZER INC   (United States)

Author keywords

11 Hydroxysteroid dehydrogenase type 1; Carbenoxolone; Cortisol; Cortisone; Ordered sequential mechanism

Indexed keywords

11BETA HYDROXYSTEROID DEHYDROGENASE; CORTISONE; ISOENZYME; REDUCED NICOTINAMIDE ADENINE DINUCLEOTIDE PHOSPHATE;

ARTICLE; CONTROLLED STUDY; DISSOCIATION CONSTANT; ENZYME ACTIVE SITE; ENZYME ASSAY; EQUILIBRIUM CONSTANT; HUMAN; KINETICS; MICHAELIS CONSTANT; NONHUMAN; PRIORITY JOURNAL; RABBIT;

11-BETA-HYDROXYSTEROID DEHYDROGENASE TYPE 1; ANIMALS; ENZYME ACTIVATION; ENZYME STABILITY; HUMANS; ISOENZYMES; KINETICS; RABBITS; SPECIES SPECIFICITY;

ORYCTOLAGUS CUNICULUS;

EID: 34247132757     PISSN: 0006291X     EISSN: 10902104     Source Type: Journal    
DOI: 10.1016/j.bbrc.2007.04.005     Document Type: Article

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