메뉴 건너뛰기




Volumn 87, Issue 3, 2007, Pages 238-247

In vitro metabolism and interaction of profenofos by human, mouse and rat liver preparations

Author keywords

Human; In vitro; Insecticide; LC MS; Metabolism; Mouse; Profenofos; Rat; Toxicology

Indexed keywords

MAMMALIA; RATTUS;

EID: 33846597074     PISSN: 00483575     EISSN: 10959939     Source Type: Journal    
DOI: 10.1016/j.pestbp.2006.08.002     Document Type: Article
Times cited : (41)

References (40)
  • 1
    • 79955102195 scopus 로고    scopus 로고
    • Classification and uses of organophosphates and carbamates
    • Gupta R.C. (Ed), Academic Press
    • Gupta R.C. Classification and uses of organophosphates and carbamates. In: Gupta R.C. (Ed). Toxicology of Organophosphate and Carbamate Compounds (2006), Academic Press 5
    • (2006) Toxicology of Organophosphate and Carbamate Compounds , pp. 5
    • Gupta, R.C.1
  • 2
    • 33846598561 scopus 로고    scopus 로고
    • WHO, The WHO recommended classification of pesticides by hazard and guidelines to classification 1990-1991, WHO/PCS/90.1, World Health Organization, Geneva, Switzerland, 1990.
  • 4
    • 0025100471 scopus 로고
    • Mechanism of action of organophosphorus and carbamate insecticides
    • Fukuto T.R. Mechanism of action of organophosphorus and carbamate insecticides. Environ. Health Perspect. 87 (1990) 245-254
    • (1990) Environ. Health Perspect. , vol.87 , pp. 245-254
    • Fukuto, T.R.1
  • 5
    • 0035949809 scopus 로고    scopus 로고
    • Biotransformation of organophosphorus compounds
    • Jokanovic M. Biotransformation of organophosphorus compounds. Toxicology 166 (2001) 139-160
    • (2001) Toxicology , vol.166 , pp. 139-160
    • Jokanovic, M.1
  • 6
    • 0034674894 scopus 로고    scopus 로고
    • Evidence for the activation of organophosphate pesticides by cytochromes P450 3A4 and 2D6 in human liver microsomes
    • Sams C., Mason H.J., and Rawbone R. Evidence for the activation of organophosphate pesticides by cytochromes P450 3A4 and 2D6 in human liver microsomes. Toxicol. Lett. 116 (2000) 217-221
    • (2000) Toxicol. Lett. , vol.116 , pp. 217-221
    • Sams, C.1    Mason, H.J.2    Rawbone, R.3
  • 7
    • 0034861252 scopus 로고    scopus 로고
    • Metabolism of chlorpyrifos by human cytochrome P450 isoforms and human, mouse, and rat liver microsomes
    • Tang J., Cao Y., Rose R.L., Brimfield A.A., Dai D., Goldstein J.A., and Hodgson E. Metabolism of chlorpyrifos by human cytochrome P450 isoforms and human, mouse, and rat liver microsomes. Drug Metab. Dispos. 29 (2001) 1201-1204
    • (2001) Drug Metab. Dispos. , vol.29 , pp. 1201-1204
    • Tang, J.1    Cao, Y.2    Rose, R.L.3    Brimfield, A.A.4    Dai, D.5    Goldstein, J.A.6    Hodgson, E.7
  • 8
    • 0037291881 scopus 로고    scopus 로고
    • CYP-specific bioactivation of four organophosphorothioate pesticides by human liver microsomes
    • Buratti F.M., Volpe M.T., Meneguz A., Vittozzi L., and Testai E. CYP-specific bioactivation of four organophosphorothioate pesticides by human liver microsomes. Toxicol. Appl. Pharmacol. 186 (2003) 143-154
    • (2003) Toxicol. Appl. Pharmacol. , vol.186 , pp. 143-154
    • Buratti, F.M.1    Volpe, M.T.2    Meneguz, A.3    Vittozzi, L.4    Testai, E.5
  • 9
    • 0037387854 scopus 로고    scopus 로고
    • In vitro rat hepatic and intestinal metabolism of the organophosphate pesticides chlorpyrifos and diazinon
    • Poet T.S., Wu H., Kousba A.A., and Timchalk C. In vitro rat hepatic and intestinal metabolism of the organophosphate pesticides chlorpyrifos and diazinon. Toxicol. Sci. 72 (2003) 193-200
    • (2003) Toxicol. Sci. , vol.72 , pp. 193-200
    • Poet, T.S.1    Wu, H.2    Kousba, A.A.3    Timchalk, C.4
  • 11
    • 14044273640 scopus 로고    scopus 로고
    • Malathion bioactivation in the human liver: the contribution of different cytochrome P450 isoform
    • Buratti F.M., D'Aniello A., Volpe M.T., Meneguz A., and Testai E. Malathion bioactivation in the human liver: the contribution of different cytochrome P450 isoform. Drug Metab. Dispos. 33 (2005) 295-302
    • (2005) Drug Metab. Dispos. , vol.33 , pp. 295-302
    • Buratti, F.M.1    D'Aniello, A.2    Volpe, M.T.3    Meneguz, A.4    Testai, E.5
  • 12
    • 0020682177 scopus 로고
    • Oxidative bioactivation of S-alkyl phosphorothiolate pesticides: stereospecificity of profenofos insecticide activation
    • Wing K.D., Glickman A.H., and Casida J.E. Oxidative bioactivation of S-alkyl phosphorothiolate pesticides: stereospecificity of profenofos insecticide activation. Science 219 (1983) 63-65
    • (1983) Science , vol.219 , pp. 63-65
    • Wing, K.D.1    Glickman, A.H.2    Casida, J.E.3
  • 13
    • 0021267157 scopus 로고
    • Phosphorothiolate pesticides and related compounds: oxidative bioactivation and aging of the inhibited acetylcholinesterase
    • Wing K.D., Glickman A.H., and Casida J.E. Phosphorothiolate pesticides and related compounds: oxidative bioactivation and aging of the inhibited acetylcholinesterase. Pestic. Biochem. Physiol. 21 (1984) 22-30
    • (1984) Pestic. Biochem. Physiol. , vol.21 , pp. 22-30
    • Wing, K.D.1    Glickman, A.H.2    Casida, J.E.3
  • 15
    • 18944404910 scopus 로고    scopus 로고
    • Platelet-activating factor acetylhydrolase: selective inhibition by potent n-alkyl methylphosphonofluoridates
    • Quistad G.B., Fisher K.J., Owen S.C., Klintenberg R., and Casida J.E. Platelet-activating factor acetylhydrolase: selective inhibition by potent n-alkyl methylphosphonofluoridates. Toxicol. Appl. Pharmacol. 205 (2005) 149-156
    • (2005) Toxicol. Appl. Pharmacol. , vol.205 , pp. 149-156
    • Quistad, G.B.1    Fisher, K.J.2    Owen, S.C.3    Klintenberg, R.4    Casida, J.E.5
  • 16
    • 0016245360 scopus 로고
    • Cytochrome P 450-linked monooxygenase system and drug-induced spectral interactions in human liver microsomes
    • Pelkonen O., Kaltiala E.H., Larmi T.K.I., and Karki N.T. Cytochrome P 450-linked monooxygenase system and drug-induced spectral interactions in human liver microsomes. Chem. Biol. Interact. 9 (1974) 205-216
    • (1974) Chem. Biol. Interact. , vol.9 , pp. 205-216
    • Pelkonen, O.1    Kaltiala, E.H.2    Larmi, T.K.I.3    Karki, N.T.4
  • 17
    • 0017184389 scopus 로고
    • A rapid and sensitive method for the quantitation of microgram quantities of protein utilizing the principle of protein-dye binding
    • Bradford M.M. A rapid and sensitive method for the quantitation of microgram quantities of protein utilizing the principle of protein-dye binding. Anal. Biochem. 72 (1976) 248-254
    • (1976) Anal. Biochem. , vol.72 , pp. 248-254
    • Bradford, M.M.1
  • 18
    • 0017363296 scopus 로고
    • Characteristics of a microsomal cytochrome P-448-mediated reaction. Ethoxyresorufin O-de-ethylation
    • Burke M.D., Prough R.A., and Mayer R.T. Characteristics of a microsomal cytochrome P-448-mediated reaction. Ethoxyresorufin O-de-ethylation. Drug Metab. Dispos. 5 (1977) 1-8
    • (1977) Drug Metab. Dispos. , vol.5 , pp. 1-8
    • Burke, M.D.1    Prough, R.A.2    Mayer, R.T.3
  • 19
    • 0017847465 scopus 로고
    • An improved assay of 7-ethoxycoumarin O-deethylase activity: induction of hepatic enzyme activity in C57BL/6J and DBA/2J mice by phenobarbital, 3-methylcholanthrene and 2,3,7,8-tetrachlorodibenzo-p-dioxin
    • Greenlee W., and Poland A. An improved assay of 7-ethoxycoumarin O-deethylase activity: induction of hepatic enzyme activity in C57BL/6J and DBA/2J mice by phenobarbital, 3-methylcholanthrene and 2,3,7,8-tetrachlorodibenzo-p-dioxin. J. Pharmacol. Exp. Ther. 205 (1978) 596-605
    • (1978) J. Pharmacol. Exp. Ther. , vol.205 , pp. 596-605
    • Greenlee, W.1    Poland, A.2
  • 20
    • 0018170362 scopus 로고
    • A simple and sensitive assay of 7-ethoxycoumarin deethylation
    • Aitio A. A simple and sensitive assay of 7-ethoxycoumarin deethylation. Anal. Biochem. 85 (1978) 488-491
    • (1978) Anal. Biochem. , vol.85 , pp. 488-491
    • Aitio, A.1
  • 23
    • 0023355128 scopus 로고
    • Hepatic metabolism of tolbutamide: characterization of the form of cytochrome P-450 involved in methyl hydroxylation and relationship to in vivo disposition
    • Knodell R.G., Hall S.D., Wilkinson G.R., and Guengerich F.P. Hepatic metabolism of tolbutamide: characterization of the form of cytochrome P-450 involved in methyl hydroxylation and relationship to in vivo disposition. J. Pharmacol. Exp. Ther. 241 (1987) 1112-1119
    • (1987) J. Pharmacol. Exp. Ther. , vol.241 , pp. 1112-1119
    • Knodell, R.G.1    Hall, S.D.2    Wilkinson, G.R.3    Guengerich, F.P.4
  • 25
    • 0021336171 scopus 로고
    • Quantitative determination of dextromethorphan and three metabolites in urine by reverse-phase high-performance liquid chromatography
    • Park Y.H., Kullberg M.P., and Hinsvark O.N. Quantitative determination of dextromethorphan and three metabolites in urine by reverse-phase high-performance liquid chromatography. J. Pharm. Sci. 73 (1984) 24-29
    • (1984) J. Pharm. Sci. , vol.73 , pp. 24-29
    • Park, Y.H.1    Kullberg, M.P.2    Hinsvark, O.N.3
  • 26
    • 0023258883 scopus 로고
    • High-performance liquid chromatographic assays for bufuralol 1′-hydroxylase, debrisoquine 4-hydroxylase, and dextromethorphan O-demethylase in microsomes and purified cytochrome P-450 isozymes of human liver
    • Kronbach T., Mathys D., Gut J., Catin T., and Meyer U.A. High-performance liquid chromatographic assays for bufuralol 1′-hydroxylase, debrisoquine 4-hydroxylase, and dextromethorphan O-demethylase in microsomes and purified cytochrome P-450 isozymes of human liver. Anal. Biochem. 162 (1987) 24-32
    • (1987) Anal. Biochem. , vol.162 , pp. 24-32
    • Kronbach, T.1    Mathys, D.2    Gut, J.3    Catin, T.4    Meyer, U.A.5
  • 28
    • 0024373348 scopus 로고
    • Oxidation of midazolam and triazolam by human liver cytochrome P450IIIA4
    • Kronbach T., Mathys D., Umeno M., Gonzalez F.J., and Meyer U.A. Oxidation of midazolam and triazolam by human liver cytochrome P450IIIA4. Mol. Pharmacol. 36 (1989) 89-96
    • (1989) Mol. Pharmacol. , vol.36 , pp. 89-96
    • Kronbach, T.1    Mathys, D.2    Umeno, M.3    Gonzalez, F.J.4    Meyer, U.A.5
  • 31
    • 33845191144 scopus 로고    scopus 로고
    • In vitro metabolism and interactions of the fungicide metalaxyl in human liver preparations
    • Abass K., Reponen P., Jalonen J., and Pelkonen O. In vitro metabolism and interactions of the fungicide metalaxyl in human liver preparations. Environ. Toxicol. Pharmacol. 23 (2007) 39-47
    • (2007) Environ. Toxicol. Pharmacol. , vol.23 , pp. 39-47
    • Abass, K.1    Reponen, P.2    Jalonen, J.3    Pelkonen, O.4
  • 33
    • 0012304444 scopus 로고    scopus 로고
    • Interindividual variation of P450 enzymes in vitro and its causes
    • Pacifici G.M., and Pelkonen O. (Eds), Taylor & Francis
    • Pelkonen O., Boobis A.R., Kremers P., Ingelman-Sundberg M., and Rane A. Interindividual variation of P450 enzymes in vitro and its causes. In: Pacifici G.M., and Pelkonen O. (Eds). Variation of Drug Metabolism in Humans (2001), Taylor & Francis 269-332
    • (2001) Variation of Drug Metabolism in Humans , pp. 269-332
    • Pelkonen, O.1    Boobis, A.R.2    Kremers, P.3    Ingelman-Sundberg, M.4    Rane, A.5
  • 34
    • 0021033669 scopus 로고
    • Activation of an O-ethyl S-n-propyl phosphorothiolate, TIA-230, in the central nerve of Spodoptera larvae
    • Kono Y., Sato Y., and Okada Y. Activation of an O-ethyl S-n-propyl phosphorothiolate, TIA-230, in the central nerve of Spodoptera larvae. Pestic. Biochem. Physiol. 20 (1983) 225-231
    • (1983) Pestic. Biochem. Physiol. , vol.20 , pp. 225-231
    • Kono, Y.1    Sato, Y.2    Okada, Y.3
  • 35
    • 33646480180 scopus 로고    scopus 로고
    • Metabolic resistance mechanisms of the housefly (Musca domestica) resistant to pyraclofos
    • Lee S., Ohta K., Tashiro S., and Shono T. Metabolic resistance mechanisms of the housefly (Musca domestica) resistant to pyraclofos. Pestic. Biochem. Physiol. 85 (2006) 76-83
    • (2006) Pestic. Biochem. Physiol. , vol.85 , pp. 76-83
    • Lee, S.1    Ohta, K.2    Tashiro, S.3    Shono, T.4
  • 37
    • 0344933196 scopus 로고    scopus 로고
    • Cytochrome P450 isoenzymes involved in parathion metabolism in the rat
    • Mutch E., Blain P.G., and Williams F.M. Cytochrome P450 isoenzymes involved in parathion metabolism in the rat. Hum. Exp. Toxicol. 15 (1996) 689
    • (1996) Hum. Exp. Toxicol. , vol.15 , pp. 689
    • Mutch, E.1    Blain, P.G.2    Williams, F.M.3
  • 38
    • 26944449329 scopus 로고    scopus 로고
    • The refinement of uncertainty/safety factors in risk assessment by the incorporation of data on toxicokinetic variability in humans
    • Dorne J.L.C.M., and Renwick A.G. The refinement of uncertainty/safety factors in risk assessment by the incorporation of data on toxicokinetic variability in humans. Toxicol. Sci. 86 (2005) 20-26
    • (2005) Toxicol. Sci. , vol.86 , pp. 20-26
    • Dorne, J.L.C.M.1    Renwick, A.G.2
  • 39
    • 0031809917 scopus 로고    scopus 로고
    • Human variability and noncancer risk assessment-an analysis of the default uncertainty factor
    • Renwick A.G., and Lazarus N.R. Human variability and noncancer risk assessment-an analysis of the default uncertainty factor. Regul. Toxicol. Pharmacol. 27 (1998) 3-20
    • (1998) Regul. Toxicol. Pharmacol. , vol.27 , pp. 3-20
    • Renwick, A.G.1    Lazarus, N.R.2
  • 40
    • 0023229967 scopus 로고
    • The interaction between phosphorothionate insecticides, pneumotoxic trialkyl phosphorothiolates and effects on lung 7-ethoxycoumarin O-deethylase activity
    • Verschoyle R.D., and Aldridge W.N. The interaction between phosphorothionate insecticides, pneumotoxic trialkyl phosphorothiolates and effects on lung 7-ethoxycoumarin O-deethylase activity. Arch. Toxicol. 60 (1987) 311-318
    • (1987) Arch. Toxicol. , vol.60 , pp. 311-318
    • Verschoyle, R.D.1    Aldridge, W.N.2


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.