Recent Advances in Oral Prodrug Discovery

Annual Reports in Medicinal Chemistry

Volumn 41, Issue , 2006, Pages 395-407

  Cho, Aesop ^a  

^a GILEAD SCIENCES   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

EID: 33846399758     PISSN: 00657743     EISSN: None     Source Type: Book Series    
DOI: 10.1016/S0065-7743(06)41027-7     Document Type: Review

References (46)

1. Testa B., and Mayer J.M. Hydrolysis in Drug and Prodrug Metabolism (2003), VHCA, Switzerland p. 420
2. Gomez-Orellana I. Expert Opin. Drug Deliv. 2 (2005) 419
3. Beaumont K., Webster R., Gardner I., and Dack K. Curr. Drug Metab. 4 (2004) 416
4. Ettmayer P., Amidon G.L., Clement B., and Testa B. J. Med. Chem. 47 (2004) 1
5. Fleisher D., Bong R., and Stewart B.H. Adv. Drug Deliv. Rev. 19 (1996) 115
6. Taylor M.D. Adv. Drug Deliv. Rev. 19 (1996) 131
7. Majumdar S., Duvvuri S., and Mitra A.K. Adv. Drug Deliv. Rev. 56 (2004) 1437
8. Chan O.H., Schmid H.L., Stilgenbauer L.A., Howson W., Horwell D.C., and Stewart B.H. Pharmaceut. Res. 15 (1998) 1012
9. Furfine E.S., Baker C.T., Hale M.R., Reynolds D.J., Salisbury J.A., Searle A.D., Studenberg S.D., Todd D., Tung R.D., and Spaltenstein A. Antimicrob. Agents Chemother. 48 (2004) 791
10. Y. Ueda, T. P. Connolly, J. F. Kadow, N. A. Meanwell, T. Wang, C. H. Chen, K. Yeung, Z. Zhang, D. K. Leahy, S. K. Pack, N. Soundararajan, P. Sirard, K. Levesque and D. Thoraval, US Patent 2005/0209246 A1, 2005.
11. Ohwada J., Tsukazaki M., Hayase T., Oikawa N., Isshiki Y., Fukuda H., Mizuguchi E., Sakaitani M., Shiratori Y., Yamazaki T., Ichihara S., Umeda I., and Shimma N. Bioorg. Med. Chem. Lett. 13 (2003) 191
12. Schmitt-Hoffmann A., Roos B., Heep M., Schleimer M., Weidekamm E., Brown T., Roehrle M., and Beglinger C. Antimicrob. Agents Chemother. 50 (2006) 279
13. T. Hayase, S. Ichihara, Y. Isshiki, P. Liu, J. Ohwada, T. Sakai, N. Shimma, M. Tsukazaki, I. Umeda and T. Yamazaki, US Patent 6,300,353 B1, 2001.
14. Nielsen A.B., Buur A., and Larsen C. Eur. J. Pharm. Sci. 26 (2005) 421
15. L. Schaller, T. Burnette, J. Cowan, P. Feldman, G. Freeman, H. Marr, B. Owens, K. Romines, J. Shepard, L. Boone, J. Chan, Abstr. 43rd Intersci. Conf. Antimicrob. Agents Chemother., poster H-872, 2003.
16. Ferris R.G., Hazen R.J., Roberts G.B., Clair M.H., Chan J.H., Romines K.R., Freeman G.A., Tidwell J.H., Schaller L.T., Cowan J.R., Short S.A., Weaver K.L., Selleseth D.W., Moniri K.R., and Boone L.R. Antimicrob. Agents Chemother. 49 (2005) 4046
17. Gingrich D.E., Reddy D.R., Igbal M.A., Singh J., Aimone L.D., Angeles T.S., Albom M., Yang S., Ator M.A., Meyer S.L., Robinson C., Ruggeri B.A., Dionne C.A., Vaught J.L., Mallamo J.P., and Hudkins R.L. J. Med. Chem. 46 (2003) 5375
18. Bouerat L., Fensholdt J., Liang X., Havez S., Nielsen S.F., Hansen J.R., Bolvig S., and Andersson C. J. Med. Chem. 48 (2005) 5412
19. V. Josyula, R. Gadwood, L. Thomasco, J. Kim and A. Choy, WO Patent 2005/028473 A1, 2005.
20. A. Marfat, D. G. McLeod and J. P. O'Donnell, US Patent 2005/0004093 A1, 2005.
21. Filla S.A., Winter M.A., Johnson K.W., Bleakman D., Bell M.G., Bleisch T.J., Castano A.M., Clemens-Smith A., del Prado M., Dieckman D.K., Dominguez E., Escribano A., Ho K.H., Hudziak K.J., Katofiasc M.A., Martinez-Perez J.A., Mateo A., Mathes B.M., Mattiuz E.L., Ogden A.M.L., Phebus L.A., Stack D.R., Stratford R.E., and Ornstein P.L. J. Med. Chem. 45 (2002) 4383
22. Kondo C., Onuki R., Kusuhara H., Suzuki H., Suzuki M., Okudaira N., Kojima M., Ishiwata K., Jonker J.W., and Sugiyama Y. Pharmaceut. Res. 22 (2005) 613
23. Dantzig A.H., Hillgren K.M., and de Alwis D.P. Annu. Rep. Med. Chem. 39 (2004) 279
24. Chanteux H., Bambeke F.V., Mingeot-Leclercq M.-P., and Tulkens P.M. Antimicrob. Agents Chemother 49 (2005) 1279
25. R. Daifuku, A. Gall, D. Sergueev, D. Sologub, K. Harris, US Patent 2005/0014752 A1, 2005.
26. Beutner K.R. Antivir. Res. 28 (1995) 281
27. Thomsen A.E., Christensen M.S., Bagger M.A., and Steffansen B. Eur. J. Pharm. Sci. 23 (2004) 319
28. Bueno A.B., Collado I., de Dios A., Dominguez C., Martin J.A., Martin L.M., Martinez-Grau M.A., Montero C., Pedregal C., Catlow J., Coffey D.S., Clay M.P., Dantzig A.H., Lindstrom T., Monn J.A., Jiang H., Schoepp D.D., Stratford R.E., Tobas L.B., Tizzano J.P., Wright R.A., and Herin M.F. J. Med. Chem. 48 (2005) 5305
29. Rorick-Kehn L.M., Perkins E.J., Knitowski K.M., Hart J.C., Johnson B.G., Schoepp D.D., and McKinzie D.L. J. Pharmacol. Exp. Ther. 316 (2006) 905
30. Cundy K.C., Branch R., Chernov-Rogan T., Dias T., Estrada T., Hold K., Koller K., Liu X., Mann A., Panuwat M., Raillard S.P., Upadhyay S., Wu Q.Q., Xiang J., Yan H., Zerangue N., Zhou C.X., Barrett R.W., and Gallop M.A. J. Pharmacol. Exp. Ther. 311 (2004) 315
31. Cundy K.C., Annamalai T., Bu L., De Vera J., Estrela J., Luo W., Shirsat P., Torneros A., Yao F., Zou J., Barrett R.W., and Gallop M.A. J. Pharmacol. Exp. Ther. 311 (2004) 324
32. Miwa M., Ura M., Nishida M., Sawada N., Ishikawa T., Mori K., Shimma N., Umeda I., and Ishitsuka H. Eur. J. Cancer 34 (1998) 1274
33. Desmoulin F., Gilard V., Malet-Martino M., and Martino R. Drug Metab. Dispos. 30 (2002) 1221
34. Hattori K., Kohchi Y., Oikawa N., Suda H., Ura M., Ishikawa T., Miwa M., Endoh M., Eda H., Tanimura H., Kawashima A., Horii I., Ishitsuka H., and Shimma N. Bioorg. Med. Chem. Lett. 13 (2003) 867
35. Lee W.A., He G., Eisenberg E., Cihlar T., Swaminathan S., Mulato A., and Cundy K.C. Antimicrob. Agents Chemother. 49 (2005) 1898
36. Lin C., Yeh L., Vitarella D., Hong Z., and Erion M.D. Antivir. Chem. Chemother. 15 (2004) 307
37. Ciesla S.L., Trahan J., Wan W.B., Beadle J.R., Aldern K.A., Painter G.R., and Hostetler K.Y. Antivir. Res. 59 (2003) 163
38. Landowski C.P., Song X., Lorenzi P.L., Hilfinger J.M., and Amidon G.L. Pharmaceut. Res. 22 (2005) 1510
39. Song X., Lorenzi P.L., Landowski C.P., Vig B.S., Hilfinger J.M., and Amidon G.L. Mol. Pharmaceutics 2 (2005) 157
40. T. Piccariello, R. J. Kirk and L. P. Olon, US Patent 2004/0063628 A1, 2004.
41. J. Chen, D. F. Welty and D. D. Tang-Liu, US Patent 2005/0075371 A1, 2005.
42. K. C. Cundy, M. A. Gallop, C. X. Zhou, US Patent 2005/0272710 A1, 2005.
43. Rodriguez-Tellez M., Arguelles F., Herrerias Jr. J.M., Ledro D., Esteban J., and Herrerias J.M. Curr. Pharm. Design 7 (2001) 951
44. Sotbera L.A., Castaner J., and Garcia-Capdevila L. Drugs Fut. 30 (2005) 545
45. T. C. Mickle, S. Bera, S. Guenther, W. Hirschelman, S. Krishnan, C. Lauderback, S. Moncreif, J. Gill, D. Jones, D. Linn, A. Martin, C. Miller and D. Portlock, Abstracts of Paper, MEDI-246, 230th ACS National Meeting, Washington, DC, 2005.
46. T. Mickle, T. Piccariello, J. S. Moncrief, N. J. Boerth and B. Bishop, WO Patent 2004/062614 A2, 2004.