The gatekeeper: Friend or foe in identifying the next generation of kinase inhibitors

ChemMedChem

Volumn 1, Issue 11, 2006, Pages 1195-1196

  Prien, Olaf ^a  

^a BAYER PHARMA AG   (Germany)

Author keywords

Antitumor agents; Drug design; Gatekeeper; Inhibitors; Mutation

Indexed keywords

PROTEIN KINASE INHIBITOR; PROTEIN TYROSINE KINASE;

CHEMICAL STRUCTURE; CHEMISTRY; DRUG ANTAGONISM; SHORT SURVEY;

MODELS, MOLECULAR; PROTEIN KINASE INHIBITORS; PROTEIN-TYROSINE KINASES;

EID: 33751246210     PISSN: 18607179     EISSN: 18607187     Source Type: Journal    
DOI: 10.1002/cmdc.200600163     Document Type: Short Survey

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