Novel T-type calcium channel blockers: Dioxoquinazoline carboxamide derivatives

Bioorganic and Medicinal Chemistry

Volumn 15, Issue 1, 2007, Pages 365-373

  Jo, Mi Na ^a   Seo, Hee Jeong ^a   Kim, Yoonji ^a   Seo, Seon Hee ^a   Rhim, Hyewhon ^a   Cho, Yong Seo ^a   Cha, Joo Hwan ^a   Koh, Hun Yeong ^b   Choo, Hyunah ^a   Pae, Ae Nim ^a  

^a Korea Institute of Science and Technology   (South Korea)

^b Inha University   (South Korea)

Author keywords

Dioxoquinazoline carboxamide derivatives; T type calcium channel blockers

Indexed keywords

3 (4 CHLOROBENZYL) N [3 (2 ETHYLPIPERIDIN 1 YL)PROPYL] 2,4 DIOXOQUINAZOLINE 7 CARBOXAMIDE; CALCIUM CHANNEL BLOCKING AGENT; CALCIUM CHANNEL T TYPE; DIOXOQUINAZOLINE CARBOXAMIDE DERIVATIVE; QUINAZOLINE DERIVATIVE; UNCLASSIFIED DRUG;

ARTICLE; CELL STRAIN HEK293; CONTROLLED STUDY; DRUG ACTIVITY; DRUG DESIGN; DRUG POTENCY; DRUG SCREENING; DRUG SYNTHESIS; EMBRYO; HUMAN; HUMAN CELL; IC 50; MOLECULAR LIBRARY;

AMIDES; CALCIUM CHANNEL BLOCKERS; CALCIUM CHANNELS, T-TYPE; CELL LINE; DRUG DESIGN; DRUG EVALUATION, PRECLINICAL; HUMANS; MOLECULAR STRUCTURE; QUINAZOLINES; STEREOISOMERISM; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 33750952104     PISSN: 09680896     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmc.2006.09.051     Document Type: Article

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