Novel approach to DPI carrier lactose with mechanofusion process with additives and evaluation by IGC

Chemical and Pharmaceutical Bulletin

Volumn 54, Issue 11, 2006, Pages 1508-1514

  Kumon, Michiko ^a   Suzuki, Masahiko ^a   Kusai, Akira ^a   Yonemochi, Etsuo ^b   Terada, Katsuhide ^b  

^a DAIICHI SANKYO CO   (Japan)

^b TOHO UNIVERSITY   (Japan)

Author keywords

Dry powder inhaler; Inverse gas chromatography; Lactose; Magnesium stearate; Mechanofusion; Sucrose stearate

Indexed keywords

LACTOSE PERMEASE; MAGNESIUM STEARATE; STEARIC ACID; SUCROSE;

ACIDITY; ARTICLE; CHEMICAL INTERACTION; DISPERSION; DRY POWDER; INHALER; INVERSE GAS CHROMATOGRAPHY; SCANNING ELECTRON MICROSCOPY;

CHROMATOGRAPHY, GAS; DRUG CARRIERS; DRUG DELIVERY SYSTEMS; EQUIPMENT DESIGN; ETHERS; HYDROCARBONS, FLUORINATED; LACTOSE; MICROSCOPY, ELECTRON, SCANNING; PARTICLE SIZE; POWDERS; SENSITIVITY AND SPECIFICITY; SURFACE PROPERTIES;

EID: 33750741095     PISSN: 00092363     EISSN: 13475223     Source Type: Journal    
DOI: 10.1248/cpb.54.1508     Document Type: Article

References (32)

1. Dunbar C., Scheuch G., Sommerer K., DeLong M., Verma A., Batycky R., Int. J. Pharm., 245, 179-189 (2002).
2. Schiavone H., Palakodaty S., Clark A., York P., Tzannis S. T., Int. J. Pharm., 281, 55-66 (2004).
3. Yamashita C., Pharm Stage, 4, 59-65 (2004).
4. Steckel H., Muller B. W., Int. J. Pharm., 154, 19-29 (1997).
5. Zeng X. M., Martin G. P., Marriott C., Pritchard J., Int. J. Pharm., 200, 93-106 (2000).
6. Chan L. W., Lim L. T., Heng P. W. S., J. Pharm. Sci., 92, 975-984 (2003).
7. Kawashima Y., Serigano T., Hino T., Yamamoto H., Takeuchi H., Int. J. Pharm., 172, 179-188 (1998).
8. Yamamoto H., Kurashima H., Katagiri D., Yang M., Takeuchi H., Kawashima Y., Yokoyama T., Tsujimoto H., Yakuzaigaku, 64, 245-253 (2004).
9. Concessio N. M., VanOort M. M., Knowles M. R., Hickey A. J., Pharm. Res., 16, 828-834 (1999).
10. Bérard V., Lesniewska E., Andrès C., Pertuy D., Laroche C., Pourcelot Y., Int. J. Pharm., 232, 213-224 (2002).
11. Price R., Young P. M., Edge S., Staniforth J. N., Int. J. Pharm., 246, 47-59 (2002).
12. Chew N. Y. K., Bagster D. F., Chan H. K., Int. J. Pharm., 206, 75-83 (2000).
13. Chew N. Y. K., Chan H. K., Pharm. Res., 16, 1098-1103 (1999).
14. Steckel H., Muller B. W., Int. J. Pharm., 154, 31-37 (1997).
15. de Boer H. A., Hagedoorn P., Gjaltema D., Goede J., Kussendrager K. D., Frijlink H. W., Int. J. Pharm., 260, 201-216 (2003).
16. Newell H. E., Buckton G., Butler D. A., Thielmann F., Williams D. R., Pharm. Res., 18, 662-666 (2001).
17. Newell H. E., Buckton G., Butler D. A., Thielmann F., Williams D. R., Int. J. Pharm., 217, 45-56 (2001).
18. Cline D., Dalby R., Pharm. Res., 19, 1274-1277 (2002).
19. Newell H. E., Buckton G., Pharm. Res., 21, 1440-1444 (2004).
20. Planinsek O., Buckton G., J. Pharm. Sci., 92, 1286-1294 (2003).
21. Schultz J., Lavielle L., Martin C., J. Adhes., 23, 45-60 (1987).
22. Grimsey I. M., Feeley J. C., York P., J. Pharm. Sci., 91, 571-583 (2002).
23. Nardin M., Papirer E., J. Colloid. Interf. Sci., 137, 534-545 (1990).
24. Gutmann V., "The Donor-Acceptor Approach to Molecular Interactions," Chap. 2, Plenum Press, New York, 1978.
25. Riddle F. L., Fowkes F. M., J. Am. Chem. Soc., 112, 3259-3264 (1990).
26. Zeng X. M., Martin G. P., Tee S. K., Ghoush A. A., Marriott C., Int. J. Pharm., 182, 133-144 (1999).
27. Louey M. D., Stewart P. J., Pharm. Res., 19, 1524-1531 (2002).
28. Chan H. K., Chew N. Y., Adv. Drug Deliv. Rev., 55, 793-805 (2003).
29. Harjunen P., Lankinen T., Salonen H., Lehto V.-P., Järvinen K., Int. J. Pharm., 263, 151-163 (2003).
30. Staniforth J. N., Rees J. E., Lai F. K., Hersey J. A., J. Pharm. Pharmacol., 34, 141-145 (1982).
31. Podczeck F., Aerosol Sci. Technol., 31, 301-321 (1999).
32. Zeng X. M., Martin G. P., Marriott C., Pritchard J., J. Pharm. Sci., 90, 1424-1434 (2001).