SCOPUS 정보 검색 플랫폼

Volumn 1, Issue 9, 2006, Pages 997-1006

Conformationally constrained CCK8 analogues obtained from a rationally designed peptide library as ligands for cholecystokinin type B receptor

(9) De Luca, Stefania a Saviano, Michele a Della Moglie, Raffaella a Digilio, Giuseppe b Bracco, Chiara b Aloj, Luigi c Tarallo, Laura c Pedone, Carlo a Morelli, Giancarlo a

a CNR (Italy)

b Bioindustry Park del Canadese (Italy)

c NATIONAL CANCER INSTITUTE (Italy)

Author keywords

Cholecystokinin; Cyclic constraints; NMR structures; Peptides; Receptors

Indexed keywords

CHOLECYSTOKININ; CHOLECYSTOKININ RECEPTOR; DRUG DERIVATIVE; LIGAND; PEPTIDE; PEPTIDE LIBRARY;

ARTICLE; CHEMICAL STRUCTURE; CHEMISTRY; CONFORMATION; DRUG ANTAGONISM; DRUG DESIGN; NUCLEAR MAGNETIC RESONANCE SPECTROSCOPY; SYNTHESIS;

CHOLECYSTOKININ; DRUG DESIGN; LIGANDS; MAGNETIC RESONANCE SPECTROSCOPY; MODELS, MOLECULAR; MOLECULAR CONFORMATION; PEPTIDE LIBRARY; PEPTIDES; RECEPTORS, CHOLECYSTOKININ;

EID: 33749022768 PISSN: 18607179 EISSN: 18607187 Source Type: Journal
DOI: 10.1002/cmdc.200600054 Document Type: Article

Times cited : (12)

References (37)

1
- 0036968744
- D. Fourmy, C. Escrieut, E. Archer, C. Gales, V. Gigoux, B. Maigret, L. Moroder, S. Silvente-Poirot, J. Martinez, J. A. Fehrentz, L. Pradayrol, Pharmacol. Toxicol. 2002, 91, 313-320.
- (2002) Pharmacol. Toxicol. , vol.91 , pp. 313-320
- Fourmy, D.¹ Escrieut, C.² Archer, E.³ Gales, C.⁴ Gigoux, V.⁵ Maigret, B.⁶ Moroder, L.⁷ Silvente-Poirot, S.⁸ Martinez, J.⁹ Fehrentz, J.A.¹⁰ Pradayrol, L.¹¹

2
- 0033052520
- P. de Tullio, J. Delarge, B. Piroette, Curr. Med. Chem. 1999, 6, 433-455.
- (1999) Curr. Med. Chem. , vol.6 , pp. 433-455
- De Tullio, P.¹ Delarge, J.² Piroette, B.³

3
- 0040017647
- J. Anders, M. Blüggel, H. E. Meyer, R. Kühne, A. M. ter Laak, E. Kojro, F. Fahrenholz, Biochemistry 1999, 38, 6043-6055.
- (1999) Biochemistry , vol.38 , pp. 6043-6055
- Anders, J.¹ Blüggel, M.² Meyer, H.E.³ Kühne, R.⁴ Ter Laak, A.M.⁵ Kojro, E.⁶ Fahrenholz, F.⁷

4
- 0034699441
- C. M. R. Low, J. W. Black, H. B. Broughton, I. M. Buck, J. M. R. Davies, D. J. Dunstone, R. A. D. Hull, S. B. Kalindjian, I. M. McDonald, M. J. Pether, N. P. Shankley, K. I. M. Steel, J. Med. Chem. 2000, 43, 3505-3517.
- (2000) J. Med. Chem. , vol.43 , pp. 3505-3517
- Low, C.M.R.¹ Black, J.W.² Broughton, H.B.³ Buck, I.M.⁴ Davies, J.M.R.⁵ Dunstone, D.J.⁶ Hull, R.A.D.⁷ Kalindjian, S.B.⁸ McDonald, I.M.⁹ Pether, M.J.¹⁰ Shankley, N.P.¹¹ Steel, K.I.M.¹²

5
- 0034609831
- B. Bellier, M. E. Million, S. DaNascimento, H. Meudal, S. Kellou, B. Maigret, C. Garbay, J. Med. Chem. 2000, 43, 3614-3623.
- (2000) J. Med. Chem. , vol.43 , pp. 3614-3623
- Bellier, B.¹ Million, M.E.² Danascimento, S.³ Meudal, H.⁴ Kellou, S.⁵ Maigret, B.⁶ Garbay, C.⁷

6
- 28144452231
- M. Martin-Martinez, N. De la Figuera, M. LaTorre, M. T. Garcia-Lopez, E. Cenarruzabeitia, J. Del Rio, R. Gonzales-Muñiz, J. Med. Chem. 2005, 48, 7667-7674.
- (2005) J. Med. Chem. , vol.48 , pp. 7667-7674
- Martin-Martinez, M.¹ De La Figuera, N.² Latorre, M.³ Garcia-Lopez, M.T.⁴ Cenarruzabeitia, E.⁵ Del Rio, J.⁶ Gonzales-Muñiz, R.⁷

7
- 33749038154
- S. Silvente-Poirot, S. A. Wank, J. Biol. Chem. 1996, 271, 1468-14706.
- (1996) J. Biol. Chem. , vol.271 , pp. 1468-14706
- Silvente-Poirot, S.¹ Wank, S.A.²

8
- 33749007760
- F. Schmitz, D. S. Pratt, M. J. Wu, L. F. Kolakowski, M. Beinborn, A. Kopin, Mol. Pharmacol. 1996, 50, 3804-3809.
- (1996) Mol. Pharmacol. , vol.50 , pp. 3804-3809
- Schmitz, F.¹ Pratt, D.S.² Wu, M.J.³ Kolakowski, L.F.⁴ Beinborn, M.⁵ Kopin, A.⁶

9
- 0031818991
- S. Silvente-Poirot, C. Escrieut, S.A. Wank, Mol. Pharmacol. 1998, 54, 364-371.
- (1998) Mol. Pharmacol. , vol.54 , pp. 364-371
- Silvente-Poirot, S.¹ Escrieut, C.² Wank, S.A.³

10
- 0033551809
- S. Silvente-Poirot, C. Escrieut, C. Gales, J. A. Fehrentz, A. Escherich, S.A. Wank, J. Martinez, L. Moroder, B. Maigret, M. Bouisson, N. Vaysse, D. Fourmy, J. Biol. Chem. 1999, 274, 23191-23197.
- (1999) J. Biol. Chem. , vol.274 , pp. 23191-23197
- Silvente-Poirot, S.¹ Escrieut, C.² Gales, C.³ Fehrentz, J.A.⁴ Escherich, A.⁵ Wank, S.A.⁶ Martinez, J.⁷ Moroder, L.⁸ Maigret, B.⁹ Bouisson, M.¹⁰ Vaysse, N.¹¹ Fourmy, D.¹²

11
- 12144268032
- E. Archer-Lahlou, I. Tikhonova, C. Escrieut, M. Dufresne, C. Seva, L. Pradayrol, L. Moroder, B. Maigret, D. Fourmy, J. Med. Chem. 2005, 48, 180-191.
- (2005) J. Med. Chem. , vol.48 , pp. 180-191
- Archer-Lahlou, E.¹ Tikhonova, I.² Escrieut, C.³ Dufresne, M.⁴ Seva, C.⁵ Pradayrol, L.⁶ Moroder, L.⁷ Maigret, B.⁸ Fourmy, D.⁹

12
- 0033539640
- M. Pellegrini, D. F. Mierke, Biochemistry 1999, 38, 14775-14783.
- (1999) Biochemistry , vol.38 , pp. 14775-14783
- Pellegrini, M.¹ Mierke, D.F.²

13
- 0035799326
- C. Giragossian, D. F. Mierke, Biochemistry 2001, 40, 3804-3809.
- (2001) Biochemistry , vol.40 , pp. 3804-3809
- Giragossian, C.¹ Mierke, D.F.²

14
- 0037046144
- C. Giragossian, D. F. Mierke, Biochemistry 2002, 41, 4560-4566.
- (2002) Biochemistry , vol.41 , pp. 4560-4566
- Giragossian, C.¹ Mierke, D.F.²

15
- 12544254799
- K. G. Harikumar, J. Clain, D. I. Pinon, M. Dong, L. J. Miller, J. Biol. Chem. 2005, 280, 10441050.
- (2005) J. Biol. Chem. , vol.280 , pp. 10441050
- Harikumar, K.G.¹ Clain, J.² Pinon, D.I.³ Dong, M.⁴ Miller, L.J.⁵

16
- 0344875561
- S. De Luca, R. Ragone, C. Bracco, G. Digilio, L. Aloj, D. Tesauro, M. Saviano, C. Pedone, G. Morelli, ChemBioChem 2003, 4, 1176-1187.
- (2003) ChemBioChem , vol.4 , pp. 1176-1187
- De Luca, S.¹ Ragone, R.² Bracco, C.³ Digilio, G.⁴ Aloj, L.⁵ Tesauro, D.⁶ Saviano, M.⁷ Pedone, C.⁸ Morelli, G.⁹

17
- 33749012067
- L. Aloj, C. Caracò, M. Panico, A. Zannetti, S. Del Vecchio, D. Tesauro, S. De Luca, C. Arra, C. Pedone, G. Morelli, M. Salvatore, J. Nucl. Med. 2003, 44, 485-494.
- (2003) J. Nucl. Med. , vol.44 , pp. 485-494
- Aloj, L.¹ Caracò, C.² Panico, M.³ Zannetti, A.⁴ Del Vecchio, S.⁵ Tesauro, D.⁶ De Luca, S.⁷ Arra, C.⁸ Pedone, C.⁹ Morelli, G.¹⁰ Salvatore, M.¹¹

18
- 0003919736
- Wiley, New York
- K. Wüthrich, NMR of proteins and nucleic acids, Wiley, New York 1986.
- (1986) NMR of Proteins and Nucleic Acids
- Wüthrich, K.¹

19
- 0027742024
- L. Moroder, R. Romano, W. Guba, D. F. Mierke, H. Kessler, C. Delporte, J. Winand, J. Christophe, Biochemistry 1993, 32, 13551-13559.
- (1993) Biochemistry , vol.32 , pp. 13551-13559
- Moroder, L.¹ Romano, R.² Guba, W.³ Mierke, D.F.⁴ Kessler, H.⁵ Delporte, C.⁶ Winand, J.⁷ Christophe, J.⁸

20
- 33644787399
- S. Lifson, A. T. Hagler, P. J. Dauber, J. Am. Chem. Soc. 1979, 101, 5111-5121.
- (1979) J. Am. Chem. Soc. , vol.101 , pp. 5111-5121
- Lifson, S.¹ Hagler, A.T.² Dauber, P.J.³

21
- 6344256147
- A. T. Hagler, S. Lifson, P. J. Dauber, J. Am. Chem. Soc. 1979, 101, 5122-5130.
- (1979) J. Am. Chem. Soc. , vol.101 , pp. 5122-5130
- Hagler, A.T.¹ Lifson, S.² Dauber, P.J.³

22
- 33845560932
- A. T. Hagler, A. T. Hagler, S. Lifson, J. Am. Chem. Soc. 1979, 101, 5131-5140.
- (1979) J. Am. Chem. Soc. , vol.101 , pp. 5131-5140
- Hagler, A.T.¹ Hagler, A.T.² Lifson, S.³

23
- 0014772602
- E. Kaiser, R. L. Colescott, C. D. Bossinger, P. I. Cook, Anal. Biochem. 1970, 34, 595-598.
- (1970) Anal. Biochem. , vol.34 , pp. 595-598
- Kaiser, E.¹ Colescott, R.L.² Bossinger, C.D.³ Cook, P.I.⁴

24
- 0020214402
- R. C. Sheppard, B. J. Williams, Int. J. Pept. Protein Res. 1982, 20, 451-454.
- (1982) Int. J. Pept. Protein Res. , vol.20 , pp. 451-454
- Sheppard, R.C.¹ Williams, B.J.²

25
- 0026951903
- M. Piotto, V. Saudek, V. Sklenar, J. Biomol. NMR 1992, 2, 661-666.
- (1992) J. Biomol. NMR , vol.2 , pp. 661-666
- Piotto, M.¹ Saudek, V.² Sklenar, V.³

26
- 0001350902
- V. Sklenar, M. Piotto, R. Leppik, V. Saudek, J. Magn. Keson. Ser. A 1993, 102, 241-245.
- (1993) J. Magn. Keson. Ser. A , vol.102 , pp. 241-245
- Sklenar, V.¹ Piotto, M.² Leppik, R.³ Saudek, V.⁴

27
- 0344448273
- L. Braunschweiler, R. R. Ernst, J. Magn. Reson. 1983, 53, 521-528.
- (1983) J. Magn. Reson. , vol.53 , pp. 521-528
- Braunschweiler, L.¹ Ernst, R.R.²

28
- 5144233105
- (28] A. Bax, D. G. Davis, J. Magn. Reson. 1985, 65, 355-360.
- (1985) J. Magn. Reson. , vol.65 , pp. 355-360
- Bax, A.¹ Davis, D.G.²

29
- 0343359244
- J. Jeener, B. H. Meier, P. Bachmann, R. R. Ernst, J. Chem. Phys. 1979, 71, 4546-4553.
- (1979) J. Chem. Phys. , vol.71 , pp. 4546-4553
- Jeener, J.¹ Meier, B.H.² Bachmann, P.³ Ernst, R.R.⁴

30
- 0005963761
- U. Piantini, O. W. Sørensen, R. R. Ernst, J. Am. Chem. Soc. 1982, 104, 6800-6801.
- (1982) J. Am. Chem. Soc. , vol.104 , pp. 6800-6801
- Piantini, U.¹ Sørensen, O.W.² Ernst, R.R.³

31
- 0343459675
- C. H. Bartels, T.-H. Xia, M. Billeter, P. Güntert, K. Wüthrich, J. Biomol. NMR 1995, 6, 1-10.
- (1995) J. Biomol. NMR , vol.6 , pp. 1-10
- Bartels, C.H.¹ Xia, T.-H.² Billeter, M.³ Güntert, P.⁴ Wüthrich, K.⁵

32
- 0031576336
- P. Güntert, C. Mumenthaler, K. Wüthrich, J. Mol. Biol. 1997, 273, 283-298.
- (1997) J. Mol. Biol. , vol.273 , pp. 283-298
- Güntert, P.¹ Mumenthaler, C.² Wüthrich, K.³

33
- 0029881007
- R. Koradi, M. Billeter, K. Wüthrich, J. Mol. Graphics 1996, 14, 51-55.
- (1996) J. Mol. Graphics , vol.14 , pp. 51-55
- Koradi, R.¹ Billeter, M.² Wüthrich, K.³

34
- 33845550595
- G. Nèmethy, M. S. Pottle, H. A. Scheraga, J. Phys. Chem. 1983, 87, 1883-1887.
- (1983) J. Phys. Chem. , vol.87 , pp. 1883-1887
- Nèmethy, G.¹ Pottle, M.S.² Scheraga, H.A.³

35
- 84986437005
- F. Mohamadi, N. G. J. Richards, W. C. Guida, R. Liskamp, M. Lipton, C. Caufield, G. Chang, T. Hendrickson, W. C. Still, J. Comput. Chem. 1990, 11, 440-467.
- (1990) J. Comput. Chem. , vol.11 , pp. 440-467
- Mohamadi, F.¹ Richards, N.G.J.² Guida, W.C.³ Liskamp, R.⁴ Lipton, M.⁵ Caufield, C.⁶ Chang, G.⁷ Hendrickson, T.⁸ Still, W.C.⁹

36
- 0021757436
- S. J. Weiner, P. A. Kollman, D. A. Case, U. C. Singh, C. Chio, G. Alagona, S. Profeta, P. Weiner, J. Am. Chem. Soc. 1984, 106, 765-784.
- (1984) J. Am. Chem. Soc. , vol.106 , pp. 765-784
- Weiner, S.J.¹ Kollman, P.A.² Case, D.A.³ Singh, U.C.⁴ Chio, C.⁵ Alagona, G.⁶ Profeta, S.⁷ Weiner, P.⁸

37
- 0026620007
- D. Q. McDonald, W. C. Still, Tetrahedron Lett. 1992, 33, 7743-7746.
- (1992) Tetrahedron Lett. , vol.33 , pp. 7743-7746
- McDonald, D.Q.¹ Still, W.C.²

* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.