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Volumn 95, Issue 9, 2006, Pages 1994-2013

Physicochemical characterization of papain entrapped in ionotropically cross-linked kappa-carrageenan gel beads for stability improvement using Doehlert shell design

Author keywords

Composite index (CI); Doehlert shell design; DSC; FTIR; Ionotropic gelation; Mathematical models; Papain; Stability study; carrageenan

Indexed keywords

CARRAGEENAN; PAPAIN; POLYMER; POTASSIUM CHLORIDE;

EID: 33748932172     PISSN: 00223549     EISSN: 15206017     Source Type: Journal    
DOI: 10.1002/jps.20665     Document Type: Article
Times cited : (42)

References (50)
  • 1
    • 0343433408 scopus 로고    scopus 로고
    • Cysteine proteases and their inhibitors
    • Schirmeister T, Otto H-H. 1997. Cysteine proteases and their inhibitors. Chem Rev 97:133-171.
    • (1997) Chem Rev , vol.97 , pp. 133-171
    • Schirmeister, T.1    Otto, H.-H.2
  • 2
    • 0024393375 scopus 로고
    • Introduction of a cysteine protease active site into trypsin
    • Higaki JN, Evnin LB, Craik CS. 1989. Introduction of a cysteine protease active site into trypsin. Biochemistry 28:9256-9263.
    • (1989) Biochemistry , vol.28 , pp. 9256-9263
    • Higaki, J.N.1    Evnin, L.B.2    Craik, C.S.3
  • 3
    • 38349114375 scopus 로고    scopus 로고
    • Description of enzymes
    • New York, Singapore, Toronto: A Wiley-Intersciences Publication-John Wiley & Sons. Inc.
    • Uhlig H. 1998. Description of enzymes. Industrial enzymes and their applications, 1st ed., New York, Singapore, Toronto: A Wiley-Intersciences Publication-John Wiley & Sons. Inc., pp 37-202.
    • (1998) Industrial Enzymes and Their Applications, 1st Ed. , pp. 37-202
    • Uhlig, H.1
  • 4
    • 0001884120 scopus 로고    scopus 로고
    • Immobilization of enzymes and cells: Some practical considerations
    • Bickerstaff GF, editor. Totowa, New Jersey: Humana Press
    • Bickerstaff GF. 1997. Immobilization of enzymes and cells: Some practical considerations. In: Bickerstaff GF, editor. Immobilization of enzymes and cells, 1st ed., Totowa, New Jersey: Humana Press, pp 1-12.
    • (1997) Immobilization of Enzymes and Cells, 1st Ed. , pp. 1-12
    • Bickerstaff, G.F.1
  • 5
    • 0023876505 scopus 로고
    • The fate of multiple unit entric coated formulations in the stomach of the dog
    • Heinamaki J, Marvola M, Happonen I, Westemarck E. 1988. The fate of multiple unit entric coated formulations in the stomach of the dog. Int J Pharm 42:105-115.
    • (1988) Int J Pharm , vol.42 , pp. 105-115
    • Heinamaki, J.1    Marvola, M.2    Happonen, I.3    Westemarck, E.4
  • 6
    • 0027255271 scopus 로고
    • Release kinetics of drug from different combined retios of micropellets
    • Lin S-Y. 1993. Release kinetics of drug from different combined retios of micropellets. J Microencapsul 10:319-327.
    • (1993) J Microencapsul , vol.10 , pp. 319-327
    • Lin, S.-Y.1
  • 7
    • 0025837597 scopus 로고
    • Targeting in the gastrointestinal tract: New approaches
    • Ritschel WA. 1991. Targeting in the gastrointestinal tract: New approaches. Methods Find Exp Clin Pharmacol 13:313-336.
    • (1991) Methods Find Exp Clin Pharmacol , vol.13 , pp. 313-336
    • Ritschel, W.A.1
  • 8
    • 0030994401 scopus 로고    scopus 로고
    • Magnetically-responsive polymerized liposomes as potential oral delivery vehicles
    • Chen H, Langer R. 1997. Magnetically-responsive polymerized liposomes as potential oral delivery vehicles. Pharm Res 14:537-540.
    • (1997) Pharm Res , vol.14 , pp. 537-540
    • Chen, H.1    Langer, R.2
  • 9
    • 0031469673 scopus 로고    scopus 로고
    • The mechanism of uptake of biodegradable microparticles in Caco-2 cells is size dependent
    • Desai MP, Labhasetwar V, Walter E, Levy RJ, Amidon GL. 1997. The mechanism of uptake of biodegradable microparticles in Caco-2 cells is size dependent. Pharm Res 14:1568-1573.
    • (1997) Pharm Res , vol.14 , pp. 1568-1573
    • Desai, M.P.1    Labhasetwar, V.2    Walter, E.3    Levy, R.J.4    Amidon, G.L.5
  • 10
    • 0033046738 scopus 로고    scopus 로고
    • Matrix tablets of carrageenans. II. Release behavior and effect of added cations
    • Picker KM. 1999. Matrix tablets of carrageenans. II. Release behavior and effect of added cations. Drug Dev Ind Pharm 25:339-346.
    • (1999) Drug Dev Ind Pharm , vol.25 , pp. 339-346
    • Picker, K.M.1
  • 11
    • 0028202079 scopus 로고
    • Microencapsulation with carrageenan-locust bean gum in a multiphase emulsification technique for sustained drug release
    • Suzuki S, Lim JK. 1994. Microencapsulation with carrageenan-locust bean gum in a multiphase emulsification technique for sustained drug release. J Microencapsul 11:197-203.
    • (1994) J Microencapsul , vol.11 , pp. 197-203
    • Suzuki, S.1    Lim, J.K.2
  • 12
    • 0035834183 scopus 로고    scopus 로고
    • Preparation and in vitro evaluation of verapamil HCl and ibuprofen containing carrageenan beads
    • Sipahigil O, Dortunc B. 2001. Preparation and in vitro evaluation of verapamil HCl and ibuprofen containing carrageenan beads. Int J Pharm 228: 119-128.
    • (2001) Int J Pharm , vol.228 , pp. 119-128
    • Sipahigil, O.1    Dortunc, B.2
  • 13
    • 0029922796 scopus 로고    scopus 로고
    • Preliminary spherical agglomerates of water soluble drug using natural polymer and cross-linking technique
    • Garcia AM, Ghaly ES. 1996. Preliminary spherical agglomerates of water soluble drug using natural polymer and cross-linking technique. J Control Release 40:179-186.
    • (1996) J Control Release , vol.40 , pp. 179-186
    • Garcia, A.M.1    Ghaly, E.S.2
  • 14
    • 0034891985 scopus 로고    scopus 로고
    • Sol-gel transition behavior of pure ι-carrageenan in both salt-free and added salt states
    • Hossain KS, Miyanaga K, Maeda H, Nemoto N. 2001. Sol-gel transition behavior of pure ι-carrageenan in both salt-free and added salt states. Biomacromolecules 2:442-449.
    • (2001) Biomacromolecules , vol.2 , pp. 442-449
    • Hossain, K.S.1    Miyanaga, K.2    Maeda, H.3    Nemoto, N.4
  • 17
    • 23144433478 scopus 로고    scopus 로고
    • Effect of potassium chloride and cationic drug on swelling, erosion and release from kappa-carrageenan matrices
    • Naim S, Samuel B, Chauhan B, Paradkar A. 2004. Effect of potassium chloride and cationic drug on swelling, erosion and release from kappa-carrageenan matrices. AAPS Pharm Sci Tech 5:e25.
    • (2004) AAPS Pharm Sci Tech , vol.5
    • Naim, S.1    Samuel, B.2    Chauhan, B.3    Paradkar, A.4
  • 18
    • 0343036312 scopus 로고    scopus 로고
    • Response surface analysis of chlortetracycline and tetracycline production with K-carrageenan immobilized Streptomyces aureofaciens
    • Asanza Teruel ML, Gontier E, Bienaime C, Nava Saucedo JE, Barbotin JN. 1997. Response surface analysis of chlortetracycline and tetracycline production with K-carrageenan immobilized Streptomyces aureofaciens. Enzyme Microb Technol 21: 314-320.
    • (1997) Enzyme Microb Technol , vol.21 , pp. 314-320
    • Asanza Teruel, M.L.1    Gontier, E.2    Bienaime, C.3    Nava Saucedo, J.E.4    Barbotin, J.N.5
  • 19
    • 0000532112 scopus 로고
    • Multi-factorial designs for exploring response surfaces
    • Box GEP, Hunter JS. 1957. Multi-factorial designs for exploring response surfaces. Ann Math Stat 28: 195-241.
    • (1957) Ann Math Stat , vol.28 , pp. 195-241
    • Box, G.E.P.1    Hunter, J.S.2
  • 20
    • 0001131698 scopus 로고
    • The design of optimum multifactorial experiments
    • Plackett RL, Burman JP. 1946. The design of optimum multifactorial experiments. Biometrika 33: 305-325.
    • (1946) Biometrika , vol.33 , pp. 305-325
    • Plackett, R.L.1    Burman, J.P.2
  • 21
    • 84946657020 scopus 로고
    • Some new three level desings for the study of quantitative variables
    • Box GEP, Behnken DW. 1960. Some new three level desings for the study of quantitative variables. Technometrics 2:455-476.
    • (1960) Technometrics , vol.2 , pp. 455-476
    • Box, G.E.P.1    Behnken, D.W.2
  • 22
    • 0000495517 scopus 로고
    • Uniform shell designs
    • Doehlert DH. 1970. Uniform shell designs. Appl Stat 19:231-239.
    • (1970) Appl Stat , vol.19 , pp. 231-239
    • Doehlert, D.H.1
  • 23
    • 0030573074 scopus 로고    scopus 로고
    • Doehlert experimental design applied to optimization and quality control of a granulation process in a high shear mixer
    • Vojnovic D, Chicoo D, Zenary HE. 1996. Doehlert experimental design applied to optimization and quality control of a granulation process in a high shear mixer. Int J Pharm 145:203-213.
    • (1996) Int J Pharm , vol.145 , pp. 203-213
    • Vojnovic, D.1    Chicoo, D.2    Zenary, H.E.3
  • 25
    • 0344061524 scopus 로고    scopus 로고
    • Development of 5-iodo-2′-deoxyuridine milling process to reduce initial burst release from PLGA microparticles
    • Geze A, Venier-Julienne MC, Mathieu D, Filmon R, Phan-Tan-Luu R, Benoit JP. 1999. Development of 5-iodo-2′-deoxyuridine milling process to reduce initial burst release from PLGA microparticles. Int J Pharm 178:257-268.
    • (1999) Int J Pharm , vol.178 , pp. 257-268
    • Geze, A.1    Venier-Julienne, M.C.2    Mathieu, D.3    Filmon, R.4    Phan-Tan-Luu, R.5    Benoit, J.P.6
  • 26
    • 0344241932 scopus 로고    scopus 로고
    • Computational program for evaluating and optimizing response-surface curves based on uniform shell designs
    • Gustavo Gonzalez A, Gonzalez-Arjona D. 1999. Computational program for evaluating and optimizing response-surface curves based on uniform shell designs. Talanta 49:433-439.
    • (1999) Talanta , vol.49 , pp. 433-439
    • Gustavo Gonzalez, A.1    Gonzalez-Arjona, D.2
  • 27
    • 85030598611 scopus 로고    scopus 로고
    • Kaysville, Utah: Number Cruncher Statistical Systems
    • Hintze J. 2003. NCSS and PASS. 2003 ed., Kaysville, Utah: Number Cruncher Statistical Systems.
    • (2003) NCSS and PASS. 2003 Ed.
    • Hintze, J.1
  • 28
    • 0000432952 scopus 로고
    • Simultaneous optimization of several responses variables
    • Derringer G, Suich R. 1980. Simultaneous optimization of several responses variables. J Qual Technol 2:214-219.
    • (1980) J Qual Technol , vol.2 , pp. 214-219
    • Derringer, G.1    Suich, R.2
  • 29
    • 0030853835 scopus 로고    scopus 로고
    • Optimization of hydrophilic matrix tablets using a D-optimal design
    • Bodeam X, Leucata SE. 1997. Optimization of hydrophilic matrix tablets using a D-optimal design. Int J Pharm 153:247-255.
    • (1997) Int J Pharm , vol.153 , pp. 247-255
    • Bodeam, X.1    Leucata, S.E.2
  • 30
    • 0037570797 scopus 로고    scopus 로고
    • Development of modified release diltiazem HCl tablets using composite index to identify optimal formulation
    • Gohel MC, Patel MM, Amin AF. 2003. Development of modified release diltiazem HCl tablets using composite index to identify optimal formulation. Drug Dev Ind Pharm 29:565-574.
    • (2003) Drug Dev Ind Pharm , vol.29 , pp. 565-574
    • Gohel, M.C.1    Patel, M.M.2    Amin, A.F.3
  • 31
    • 0028358848 scopus 로고
    • A new attempt to solve the scale up problem for granulation using response surface methodology
    • Shigeo O, Toshihiko K, Yousuke M, Horoshima S, Kozo T, Nagai T. 1994. A new attempt to solve the scale up problem for granulation using response surface methodology. J Pharm Sci 83:439-443.
    • (1994) J Pharm Sci , vol.83 , pp. 439-443
    • Shigeo, O.1    Toshihiko, K.2    Yousuke, M.3    Horoshima, S.4    Kozo, T.5    Nagai, T.6
  • 32
    • 23144449203 scopus 로고    scopus 로고
    • Composite method to quantify powder flow as a screening method in early tablet or capsule formulation development
    • article 18
    • Taylor MK, Ginsburg J, Hickey AJ, Gheyas F. 2000. Composite method to quantify powder flow as a screening method in early tablet or capsule formulation development. AAPS Pharm Sci Tech 1:(3). article 18.
    • (2000) AAPS Pharm Sci Tech , vol.1 , Issue.3
    • Taylor, M.K.1    Ginsburg, J.2    Hickey, A.J.3    Gheyas, F.4
  • 33
    • 0014138173 scopus 로고
    • Establishment of sink conditions in dissolution rate determinations- theoretical considerations and application to non-disintegrating dosage forms
    • Gibaldi M, Feldman S. 1967. Establishment of sink conditions in dissolution rate determinations-theoretical considerations and application to non-disintegrating dosage forms. J Pharm Sci 56:1238-1242.
    • (1967) J Pharm Sci , vol.56 , pp. 1238-1242
    • Gibaldi, M.1    Feldman, S.2
  • 34
    • 0014592606 scopus 로고
    • Interpretation of percent dissolved-time plots derived from in vitro testing of conventional tablets and capsules
    • Wagner JG. 1969. Interpretation of percent dissolved-time plots derived from in vitro testing of conventional tablets and capsules. J Pharm Sci 58: 1253-1257.
    • (1969) J Pharm Sci , vol.58 , pp. 1253-1257
    • Wagner, J.G.1
  • 35
    • 0344893332 scopus 로고
    • Mechanism of sustained-action medication. Theoretical analysis of rate of release of solid drugs dispersed in solid matrices
    • Higuchi T. 1963. Mechanism of sustained-action medication. Theoretical analysis of rate of release of solid drugs dispersed in solid matrices. J Pharm Sci 52:1145-1149.
    • (1963) J Pharm Sci , vol.52 , pp. 1145-1149
    • Higuchi, T.1
  • 37
    • 0021904208 scopus 로고
    • Analysis of Fickian and non-Fickian drug release from polymers
    • Peppas NA. 1985. Analysis of Fickian and non-Fickian drug release from polymers. Pharm Acta Helv 60:110-111.
    • (1985) Pharm Acta Helv , vol.60 , pp. 110-111
    • Peppas, N.A.1
  • 38
    • 84887725686 scopus 로고
    • Dependence of reaction velocity upon surface and agitation
    • Hixson AW, Crowell JH. 1931. Dependence of reaction velocity upon surface and agitation. Ind Eng Chem 23:923-931.
    • (1931) Ind Eng Chem , vol.23 , pp. 923-931
    • Hixson, A.W.1    Crowell, J.H.2
  • 39
    • 0032513508 scopus 로고    scopus 로고
    • Sustained release theophylline tablets by direct compression Part 1: Formulation and in vitro testing
    • Pather SI, Russell I, Syce JA, Neau SH. 1998. Sustained release theophylline tablets by direct compression Part 1: Formulation and in vitro testing. Int J Pharm 164:1-10.
    • (1998) Int J Pharm , vol.164 , pp. 1-10
    • Pather, S.I.1    Russell, I.2    Syce, J.A.3    Neau, S.H.4
  • 40
    • 0025760914 scopus 로고
    • Evaluation of release from selected thermosoftening vehicles
    • Kopcha M, Lordi N, Tojo KJ. 1991. Evaluation of release from selected thermosoftening vehicles. J Pharm Pharmacol 43:382-387.
    • (1991) J Pharm Pharmacol , vol.43 , pp. 382-387
    • Kopcha, M.1    Lordi, N.2    Tojo, K.J.3
  • 41
    • 84985287392 scopus 로고
    • Assay systems and characterization of Pacific whiting (Merluccius productus) protease
    • An H, Seymour TA, Wu JW, Morrissey MT. 1994. Assay systems and characterization of Pacific whiting (Merluccius productus) protease. J Food Sci 59:277-281.
    • (1994) J Food Sci , vol.59 , pp. 277-281
    • An, H.1    Seymour, T.A.2    Wu, J.W.3    Morrissey, M.T.4
  • 42
    • 27744601951 scopus 로고    scopus 로고
    • Papain entrapment in alginate beads for stability improvement and site specific delivery: Physicochemical characterization and factorial optimization using neural network modeling
    • Sankalia MG, Mashru RC, Sankalia JM, Sutariya VB. 2005. Papain entrapment in alginate beads for stability improvement and site specific delivery: Physicochemical characterization and factorial optimization using neural network modeling. AAPS Pharm Sci Tech 6(2): E209-E222.
    • (2005) AAPS Pharm Sci Tech , vol.6 , Issue.2
    • Sankalia, M.G.1    Mashru, R.C.2    Sankalia, J.M.3    Sutariya, V.B.4
  • 44
    • 0027298603 scopus 로고
    • Microencapsulation of drugs with aqueous colloidal polymer dispersions
    • Bodmeier R, Wang J. 1993. Microencapsulation of drugs with aqueous colloidal polymer dispersions. J Pharm Sci 82:191-194.
    • (1993) J Pharm Sci , vol.82 , pp. 191-194
    • Bodmeier, R.1    Wang, J.2
  • 45
    • 0028960948 scopus 로고
    • Effect of varying drug loading on particle size distribution and drug release kinetics of verapamil hydrochloride microspheres prepared with cellulose esters
    • Bhardwaj SB, Shukia AJ, Collins CC. 1995. Effect of varying drug loading on particle size distribution and drug release kinetics of verapamil hydrochloride microspheres prepared with cellulose esters. J Microencapsul 12:71-81.
    • (1995) J Microencapsul , vol.12 , pp. 71-81
    • Bhardwaj, S.B.1    Shukia, A.J.2    Collins, C.C.3
  • 46
    • 0028306685 scopus 로고
    • On the employment of λ carrageenan in a matrix system. II: λ carrageenan and hydroxypropyl-methylcellulose mixtures
    • Bonferoni MC, Rossi S, Tamayo M, Pedraz JL, Dominguez Gil A, Caramella C. 1994. On the employment of λ carrageenan in a matrix system. II: λ carrageenan and hydroxypropyl-methylcellulose mixtures. J Control Release 30: 175-182.
    • (1994) J Control Release , vol.30 , pp. 175-182
    • Bonferoni, M.C.1    Rossi, S.2    Tamayo, M.3    Pedraz, J.L.4    Dominguez Gil, A.5    Caramella, C.6
  • 47
    • 0033152277 scopus 로고    scopus 로고
    • Mechanisms of solute and drug transport in relaxing, swellable, hydrophilic glassy polymers
    • Brazel CS, Peppas NA. 1999. Mechanisms of solute and drug transport in relaxing, swellable, hydrophilic glassy polymers. Polymers 40:3383-3398.
    • (1999) Polymers , vol.40 , pp. 3383-3398
    • Brazel, C.S.1    Peppas, N.A.2
  • 48
    • 0037122675 scopus 로고    scopus 로고
    • Hydrogels for biomedical applications
    • Hoffman AS. 2002. Hydrogels for biomedical applications. Adv Drug Del Rev 43:3-12.
    • (2002) Adv Drug del Rev , vol.43 , pp. 3-12
    • Hoffman, A.S.1
  • 49
  • 50
    • 0032482180 scopus 로고    scopus 로고
    • Inclusion and release of proteins from polysaccharide-based polyion complexs
    • Severian D, Esteban C. 1998. Inclusion and release of proteins from polysaccharide-based polyion complexs. Adv Drug Deliv Rev 31:223-246.
    • (1998) Adv Drug Deliv Rev , vol.31 , pp. 223-246
    • Severian, D.1    Esteban, C.2


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