Synthesis and dipeptidyl peptidase inhibition of N-(4-substituted-2,4-diaminobutanoyl)piperidines

Bioorganic and Medicinal Chemistry Letters

Volumn 16, Issue 18, 2006, Pages 4777-4779

  Soroka, Anna ^a   der Veken, Pieter Van ^a   Meester, Ingrid De ^a   Lambeir, Anne Marie ^a   Maes, Marie Berthe ^a   Scharpé, Simon ^a   Haemers, Achiel ^a   Augustyns, Koen ^a  

^a UNIVERSITY OF ANTWERP   (Belgium)

Author keywords

2,4 Diaminoalkanoylpiperidines; Dipeptidyl peptidases; DPP II; Inhibitors

Indexed keywords

DIPEPTIDYL PEPTIDASE; ENZYME INHIBITOR; PIPERIDINE DERIVATIVE;

ARTICLE; DRUG ACTIVITY; DRUG SYNTHESIS; ENZYME ACTIVITY; ENZYME INHIBITION; SUBSTITUTION REACTION;

AMINATION; DIPEPTIDYL PEPTIDASES; INHIBITORY CONCENTRATION 50; MOLECULAR STRUCTURE; PIPERIDINES; PROTEASE INHIBITORS; STEREOISOMERISM;

EID: 33746810965     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2006.06.082     Document Type: Article

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