Synthesis of potential biologically active 1,2-benzothiazin-3-yl- quinazolin-4(3H)-ones

Chemical and Pharmaceutical Bulletin

Volumn 54, Issue 8, 2006, Pages 1175-1178

  Zia Ur Rehman, Muhammad ^a,b   Choudary, Jamil Anwar ^b   Ahmad, Saeed ^a   Siddiqui, Hamid Latif ^b  

^a PCSIR LABORATORIES COMPLEX   (Pakistan)

^b UNIVERSITY OF THE PUNJAB   (Pakistan)

Author keywords

1,2 benzothiazin 3 yl quinazolin 4(3H) one; 1,2 benzothiazine 3 carboxamide; Anthranilamide; Antibacterial agent; Potassium tertiary butoxide

Indexed keywords

2 (4 HYDROXY 1,1 DIOXIDO 2H 1,2 BENZOTHIAZIN 3 YL)QUINAZOLIN 4(3H) ONES; 2 AMINOBENZAMIDE; 4 HYDROXY 1,2 BENZOTHIAZINE 1,1 DIOXIDE DERIVATIVE; N [2 (AMINOCARBONYL)PHENYL] 4 HYDROXY 1,2 BENZOTHIAZINE 3 CARBOXAMIDE 1,1 DIOXIDE DERIVATIVE; OXIDE; QUINAZOLINE DERIVATIVE; UNCLASSIFIED DRUG;

ANTIMICROBIAL ACTIVITY; ARTICLE; BACILLUS SUBTILIS; DRUG ACTIVITY; DRUG DESIGN; DRUG SYNTHESIS; GRAM NEGATIVE BACTERIUM; GRAM POSITIVE BACTERIUM; NONHUMAN;

ANTHRANILIC ACIDS; ANTI-BACTERIAL AGENTS; BACILLUS SUBTILIS; DRUG EVALUATION, PRECLINICAL; MOLECULAR STRUCTURE; QUINAZOLINES; THIAZINES;

EID: 33746700268     PISSN: 00092363     EISSN: 13475223     Source Type: Journal    
DOI: 10.1248/cpb.54.1175     Document Type: Article

References (26)

1. Vidal A., Madelmont J. C., Mounetou E., Synthesis, 2006, 591-594 (2006).
2. Lombardino J. G., Wiseman E. H., Mclamore W., J. Med. Chem., 14, 1171-1175 (1971).
3. Marfat A., Annual Drug Report, 1987, 202; US Patent, 4551452 (1985).
4. Turck D., Busch U., Heinzel G., Narjes H., Nehmiz G., Clin. Pharmacol., 36, 79-84 (1996).
5. Bihovsky R., Tao M., Mallamo J. P., Wells G. J., Bioorg. Med. Chem. Lett., 14, 1035-1038 (2004).
6. Bihovsky R., Tao M., Mallamo J. P., Wells G. J., J. Med. Chem., 44, 3488-3503 (2001).
7. Baruffini A., Pagani G., Amoretti L., Il Farmaco, 22, 528-534 (1967).
8. Fringuelli R., Schiaffella F., Vecchiarelli A., J. Chemother., 13, 9-14 (2001).
9. Bekhit A. A., Habbib N. S., Bekhit A. El., Boll. Chim. Farm., 140, 297-301 (2001).
10. Jiang J. B., Hesson D. P., Dusak B. A., Dexter D. L., Kang G. T., J. Med. Chem., 33, 1721-1728 (1990).
11. Tani J., Yamada Y., Oine T., Ochiai T., Ishida R., Inoue I., J. Med. Chem., 22, 95-99 (1979).
12. Ochiai T., Ishida R., Jpn. J. Pharmacol., 32, 427-438 (1982).
13. Raffa D., Daidone G., Schillaci D., Maggio B., Plescia F., Pharmazie, 54, 251-254 (1999).
14. Robert J. A., Russell H. E., J. Med. Chem., 15, 335-336 (1972).
15. Jantova S., Greif G., Spirkova K., Stankovsky S., Oravcova M., Folia Microbiol. (Praha), 45, 133-137 (2000).
16. Guersoy A., Illhan N., Farmaco, 50, 559-562 (1995).
17. Pandeya S. N., Sriram D., Nath G., DeClereq E., Pharm. Acta Helv., 74, 11-17 (1999).
18. Caroll S. S., Stahlhut M., Greb J., Olsen D. B., J. Biol. Sci., 269, 32351-32359 (1994).
19. Lopez S. E., Rosales M. E., Canelon C. E., Valverode E. A., Narvaez R. C., Charris J. E., Giannini F. A., Enriz R. D., Carrasco M., Zacchino S., Hetrocycl. Commun., 7, 473-480 (2000).
20. Farghaly A. O., Moharram A. M., Boll. Chim. Farm., 138, 280-289 (1999).
21. Kwon S. K., Park M. S., Arzneium-Forsch./Drug Res., 46, 966-971 (1996).
22. Rehman M. Z., Anwar J., Ahmad S., Bull. Korean Chem. Soc., 26, 1771-1775 (2005).
23. Nunomoto S., Kawakami Y., Yamashita Y., Takeuchi H., Eguchi S., J. Chem. Soc., Perkin Trans. 1, 1990, 111-114 (1990).
24. Le Z. G., Chen Z. C., Hu Y., Zheng Q. G., Synthesis, 2004, 208-212 (2004).
25. Colle J. G., Duguid J. P., Fraser A. G., Marmion B. P., "Practical Medical Biology," 13th ed., ed. by Mackie T. J., McCartney J. E., Churchill Livingstone, London, UK, 1989.
26. Owens G. S., Abu-Omer M. M., J. Mol. Catal. A: Chem., 187, 215-221 (2002).