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Volumn 49, Issue 2, 2006, Pages 169-176

Novel 99mTc labeled a receptor ligand as a potential tumor imaging agent

Author keywords

receptor; 99mTc; SPECT; Tumor

Indexed keywords

COMPLEXATION; IMAGING TECHNIQUES; LEAD COMPOUNDS; MODIFICATION; RHENIUM COMPOUNDS; TUMORS;

EID: 33745157528     PISSN: 10069291     EISSN: None     Source Type: Journal    
DOI: 10.1007/s11426-006-0169-z     Document Type: Article
Times cited : (22)

References (46)
  • 1
    • 0026567933 scopus 로고
    • A proposal for the classification of sigma binding sites
    • Quirion, R., Bowen, W. D., Itzhak, Y. et al., A proposal for the classification of sigma binding sites, Trends Pharmacol. Sci., 1992, 13: 85-86.
    • (1992) Trends Pharmacol. Sci. , vol.13 , pp. 85-86
    • Quirion, R.1    Bowen, W.D.2    Itzhak, Y.3
  • 2
    • 0025881278 scopus 로고
    • Sigma receptors: Putative links between nervous, endocrine and immune systems
    • Su, T. P., Sigma receptors: Putative links between nervous, endocrine and immune systems, Eur. J. Biochem., 1991, 200: 633-642.
    • (1991) Eur. J. Biochem. , vol.200 , pp. 633-642
    • Su, T.P.1
  • 3
    • 3843108019 scopus 로고    scopus 로고
    • Sigma receptors: Biology and therapeutic potential
    • Guitart, X., Codony, X., Monroy, X., Sigma receptors: Biology and therapeutic potential, Psychopharmacology, 2004, 174: 301-319.
    • (2004) Psychopharmacology , vol.174 , pp. 301-319
    • Guitart, X.1    Codony, X.2    Monroy, X.3
  • 4
    • 0028795145 scopus 로고
    • Sigma-1 and sigma-2 receptors are expressed in a wide variety of human and rodent tumor cell lines
    • Vilner, B. J., John, C. S., Bowen, W. D., Sigma-1 and sigma-2 receptors are expressed in a wide variety of human and rodent tumor cell lines, Cancer Res., 1995, 55: 408-413.
    • (1995) Cancer Res. , vol.55 , pp. 408-413
    • Vilner, B.J.1    John, C.S.2    Bowen, W.D.3
  • 5
    • 0031015053 scopus 로고    scopus 로고
    • 2 receptors as potential biomarkers of proliferation in breast cancer
    • 2 receptors as potential biomarkers of proliferation in breast cancer, Cancer Res., 1997, 57: 156-161.
    • (1997) Cancer Res. , vol.57 , pp. 156-161
    • Mach, R.H.1    Smith, C.R.2    al-Nabulsi, I.3
  • 6
    • 0030861403 scopus 로고    scopus 로고
    • 18F]fluorobenzamide: A potential ligand for PET imaging of σ receptors
    • 18F]fluorobenzamide: A potential ligand for PET imaging of σ receptors, Nucl. Med. Biol., 1997, 24: 671-676.
    • (1997) Nucl. Med. Biol. , vol.24 , pp. 671-676
    • Shiue, C.Y.1    Shiue, G.G.2    Zhang, S.X.3
  • 7
    • 0030611036 scopus 로고    scopus 로고
    • 18F] labeled benzamides: High affinity sigma receptor ligands for PET imaging
    • 18F] labeled benzamides: High affinity sigma receptor ligands for PET imaging, Nucl. Med. Biol., 1997, 24: 333-340.
    • (1997) Nucl. Med. Biol. , vol.24 , pp. 333-340
    • Dence, C.S.1    John, C.S.2    Bowen, W.D.3
  • 8
    • 0034528077 scopus 로고    scopus 로고
    • 18F]fluorobenzamide: A potential ligand for PET imaging of breast cancer
    • 18F]fluorobenzamide: A potential ligand for PET imaging of breast cancer, Nucl. Med. Biol., 2000, 27: 763-767.
    • (2000) Nucl. Med. Biol. , vol.27 , pp. 763-767
    • Shiue, C.Y.1    Shiue, G.G.2    Benard, F.3
  • 9
    • 18144396486 scopus 로고    scopus 로고
    • Investigation of a new sigma-2 receptor ligand for detection of breast cancer
    • Rowland, D. J., Tu, Z., Mach, R. H. et al, Investigation of a new sigma-2 receptor ligand for detection of breast cancer, J. Labelled Cpd. Radiopharm., 2003, 46: S6.
    • (2003) J. Labelled Cpd. Radiopharm. , vol.46
    • Rowland, D.J.1    Tu, Z.2    Mach, R.H.3
  • 10
    • 0031004411 scopus 로고    scopus 로고
    • Sigma receptor imaging by means of 123-IDAB scintigraphy; clinical application in melanoma and non-small cell lung cancer
    • Everaert, H., Flamen, P., Franken, P. R. et al, Sigma receptor imaging by means of 123-IDAB scintigraphy; clinical application in melanoma and non-small cell lung cancer, Anticancer Res., 1997, 17: 1577-1582.
    • (1997) Anticancer Res. , vol.17 , pp. 1577-1582
    • Everaert, H.1    Flamen, P.2    Franken, P.R.3
  • 11
    • 0032054126 scopus 로고    scopus 로고
    • 125I]BP: A potential a receptor marker for human prostate tumors
    • 125I]BP: A potential a receptor marker for human prostate tumors, Nucl. Med. Biol., 1998, 25: 189-194.
    • (1998) Nucl. Med. Biol. , vol.25 , pp. 189-194
    • John, C.S.1    Gulden, M.E.2    Li, J.3
  • 12
    • 13844305877 scopus 로고    scopus 로고
    • 123I]-4-iodo-N - (4-(4-(2-me-thoxyphenyl)-piperazin-1-yl)butyl)-benzamide: A potential sigma receptor ligand for SPECT studies
    • 123I]-4-iodo-N - (4-(4-(2-me-thoxyphenyl)-piperazin-1-yl)butyl)-benzamide: A potential sigma receptor ligand for SPECT studies, Nucl. Med. Biol., 2005, 32: 193-200.
    • (2005) Nucl. Med. Biol. , vol.32 , pp. 193-200
    • Staelens, L.1    Oltenfreiter, R.2    Dumont, F.3
  • 14
    • 0032054096 scopus 로고    scopus 로고
    • 11C]NE-100 labeled in two different positions as a PET σ receptor ligand,
    • 11C]NE-100 labeled in two different positions as a PET σ receptor ligand, Nucl. Med. Biol., 1998, 25: 195-202.
    • (1998) Nucl. Med. Biol. , vol.25 , pp. 195-202
    • Ishiwata, K.1    Noguchi, J.2    Ishii, S.-I.3
  • 17
    • 0030610886 scopus 로고    scopus 로고
    • 18F]1-(3-fluoropropyl)-4-(4-cyanophenoxymethyl) piperidine: A selective sigma-1 receptor radioligand for PET
    • 18F]1-(3-fluoropropyl)-4-(4-cyanophenoxymethyl) piperidine: A selective sigma-1 receptor radioligand for PET, Nucl. Med. Biol., 1997, 24: 127-134.
    • (1997) Nucl. Med. Biol. , vol.24 , pp. 127-134
    • Waterhouse, R.N.1    Collier, T.L.2
  • 18
    • 0030220443 scopus 로고    scopus 로고
    • 125I]N-[2-(4-iodo-phen-yl)ethyl] - N-methyl-2-(1-piperidinyl)ethylamine: A high-affinity ligand for imaging sigma receptor positive tumors
    • 125I]N-[2-(4-iodo-phen-yl)ethyl]- N -methyl-2-(1-piperidinyl)ethylamine: A high-affinity ligand for imaging sigma receptor positive tumors, Nucl. Med. Biol., 1996, 23: 761-766.
    • (1996) Nucl. Med. Biol. , vol.23 , pp. 761-766
    • John, C.S.1    Gulden, M.E.2    Vilner, B.J.3
  • 19
    • 0030972783 scopus 로고    scopus 로고
    • 123I]-1-(iodopropen-2-yl)-4-[(4-cyanophenoxy)methyl] piperidine
    • 123I]-1-(iodopropen-2-yl)-4-[(4-cyanophenoxy)methyl] piperidine, J. Med. Chem., 1997, 40: 1657-1667.
    • (1997) J. Med. Chem. , vol.40 , pp. 1657-1667
    • Waterhouse, R.N.1    Mardon, K.2    Giles, K.M.3
  • 20
    • 0030907267 scopus 로고    scopus 로고
    • 123I]1-(4-cyanobenzyl)- 4 -[[(trans-iodopropen-2-yl)oxy]-methyl] piperidine: A novel high affinity sigma receptor radioligand for SPECT
    • 123I]1-(4-cyanobenzyl)- 4 -[[(trans-iodopropen-2-yl)oxy]-methyl] piperidine: A novel high affinity sigma receptor radioligand for SPECT, Nucl. Med. Biol., 1997, 24: 45-51.
    • (1997) Nucl. Med. Biol. , vol.24 , pp. 45-51
    • Waterhouse, R.N.1    Mardon, K.2    O'Brien, J.C.3
  • 21
    • 0030608888 scopus 로고    scopus 로고
    • 123I-labeled piperidine-based sigma receptor ligands as potential melanoma imaging agents: Initial studies in mouse tumor models
    • 123I-labeled piperidine-based sigma receptor ligands as potential melanoma imaging agents: Initial studies in mouse tumor models, Nucl. Med. Biol., 1997, 24: 587-593.
    • (1997) Nucl. Med. Biol. , vol.24 , pp. 587-593
    • Waterhouse, R.N.1    Chapman, J.2    Izard, B.3
  • 22
    • 33745120413 scopus 로고    scopus 로고
    • 125I-4-(N-benzyIpiperidin)-4-iodo-phenylsulfonamide
    • Chinese source
    • 125I-4-(N-benzyIpiperidin)-4-iodo-phenylsulfonamide, J. Isotopes (in Chinese), 2004, 17: 198-203.
    • (2004) J. Isotopes , vol.17 , pp. 198-203
    • Zhang, C.1    Liu, Q.2    Wang, R.3
  • 23
    • 0037122746 scopus 로고    scopus 로고
    • Novel spiropiperidines as highly potent and subtype selective sigma-receptor ligands. Part 1
    • Maier, C. A., Wünsch, B., Novel spiropiperidines as highly potent and subtype selective sigma-receptor ligands, Part 1, J. Med. Chem., 2002, 45: 438-448.
    • (2002) J. Med. Chem. , vol.45 , pp. 438-448
    • Maier, C.A.1    Wünsch, B.2
  • 24
    • 0037168069 scopus 로고    scopus 로고
    • Novel sigma receptor ligands, Part 2. SAR of spiro[[2]benzopyran-1,4'-piperidines] and spiro[[2]ben-zofuran-1,4'-piperidines] with carbon substituents in position 3
    • Maier, C. A., Wiinsch, B., Novel sigma receptor ligands, Part 2. SAR of spiro[[2]benzopyran-1,4'-piperidines] and spiro[[2]ben-zofuran-1,4'-piperidines] with carbon substituents in position 3, J. Med. Chem., 2002, 45: 4923-4930.
    • (2002) J. Med. Chem. , vol.45 , pp. 4923-4930
    • Maier, C.A.1    Wiinsch, B.2
  • 25
    • 0027439763 scopus 로고
    • Synthesis and PET studies of fluorine-18-BMY 14802: A potential antipsychotic drug
    • Ding, Y. S., Fowler, J. S., Dewey, S. L. et al., Synthesis and PET studies of fluorine-18-BMY 14802: A potential antipsychotic drug, J. Nucl. Med., 1993, 34: 246-254.
    • (1993) J. Nucl. Med. , vol.34 , pp. 246-254
    • Ding, Y.S.1    Fowler, J.S.2    Dewey, S.L.3
  • 26
    • 0027271963 scopus 로고
    • 4-2-([3,4-dichlorophenyl]ethyl)piperazine, a high affinity ligand for sigma receptor
    • 4-2-([3,4-dichlorophenyl]ethyl)piperazine, a high affinity ligand for sigma receptor, J. Labelled Cpd. Radiopharm., 1993, 33: 639-643.
    • (1993) J. Labelled Cpd. Radiopharm. , vol.33 , pp. 639-643
    • Kiesewetter, D.O.1    de Costa, B.2
  • 29
    • 33745146081 scopus 로고    scopus 로고
    • 11C-labeled SA4503, SA5845, and their ethyl derivatives as PET sigma receptor ligands
    • 11C-labeled SA4503, SA5845, and their ethyl derivatives as PET sigma receptor ligands, J. Labelled Cpd. Radiopharm., 2001, 44(Suppl.1): S233-S235.
    • (2001) J. Labelled Cpd. Radiopharm. , vol.44 , Issue.SUPPL.1
    • Kawamura, K.1    Ishii, S.2    Kobayashi, T.3
  • 32
    • 0038397216 scopus 로고    scopus 로고
    • 18F-labeled 1-[2-(4-alkoxy-3-methoxy-phenyl)ethyl]-4-(3-phenylpropyl)piperazines as sigma receptor ligands for positron emission tomography studies
    • 18F-labeled 1-[2-(4-alkoxy-3-methoxy-phenyl)ethyl]-4-(3-phenylpropyl)piperazines as sigma receptor ligands for positron emission tomography studies, Nucl. Med. Biol., 2003, 30: 273-284.
    • (2003) Nucl. Med. Biol. , vol.30 , pp. 273-284
    • Kawamura, K.1    Elsinga, P.H.2    Kobayashi, T.3
  • 33
    • 0030609924 scopus 로고    scopus 로고
    • 99mTc-labeled σ-receptor-binding complex: Synthesis, characterization, and specific binding to human ductal breast carcinoma (T47D) cells
    • 99mTc-labeled σ-receptor-binding complex: Synthesis, characterization, and specific binding to human ductal breast carcinoma (T47D) cells, Bioconj. Chem., 1997, 8: 304-309.
    • (1997) Bioconj. Chem. , vol.8 , pp. 304-309
    • John, C.S.1    Lim, B.B.2    Geyer, B.C.3
  • 34
    • 0034886265 scopus 로고    scopus 로고
    • Development of a Tc-99 m labeled sigma-2 receptor-specific ligand as a potential breast tumor imaging agent
    • Choi, S-R., Yang, B. Plossl, K. et al., Development of a Tc-99m labeled sigma-2 receptor-specific ligand as a potential breast tumor imaging agent, Nucl. Med. Biol., 2001, 28: 657-666.
    • (2001) Nucl. Med. Biol. , vol.28 , pp. 657-666
    • Choi, S.-R.1    Yang, B.2    Plossl, K.3
  • 35
    • 0032480908 scopus 로고    scopus 로고
    • Characterization of novel N,N'-disubstituted piperazines as sigma receptor ligands
    • Zhang, Y., Williams, W., Torrence-Campbell, C. et al., Characterization of novel N,N'-disubstituted piperazines as sigma receptor ligands, J. Med. Chem., 1998, 41: 4950-4957.
    • (1998) J. Med. Chem. , vol.41 , pp. 4950-4957
    • Zhang, Y.1    Williams, W.2    Torrence-Campbell, C.3
  • 36
    • 0037059866 scopus 로고    scopus 로고
    • N-arylalkylpiperidines as high-affinuty sigma-1 and sigma-2 receptor ligands: Phenylpropylamine as potential leads for selective sigma-2 agents
    • Maeda, D. N., Williams, W., Kim, W. E. et al., N-arylalkylpiperidines as high-affinuty sigma-1 and sigma-2 receptor ligands: Phenylpropylamine as potential leads for selective sigma-2 agents, Bioorg. Med. Chem. Lett., 2002, 12: 497-500.
    • (2002) Bioorg. Med. Chem. Lett. , vol.12 , pp. 497-500
    • Maeda, D.N.1    Williams, W.2    Kim, W.E.3
  • 37
    • 0001811914 scopus 로고
    • N-substituted derivatives of piperazine and ethylenediamine. Part I. The preparation of N-monosubstituted derivatives
    • Moore, T. S., Boyle, M., Thorn, V. M. et al., N-substituted derivatives of piperazine and ethylenediamine, Part I. The preparation of N-monosubstituted derivatives, J. Chem. Soc., 1929: 39. 38.
    • (1929) J. Chem. Soc. , vol.39 , pp. 38
    • Moore, T.S.1    Boyle, M.2    Thorn, V.M.3
  • 38
    • 33947434905 scopus 로고
    • Experimental chemotherapy of filariasis. IV. The preparation of derivatives of piperazine
    • Stewart, H. W., Turner, R. J., Denton, J. J. et al., Experimental chemotherapy of filariasis, IV. The preparation of derivatives of piperazine, J. Org. Chem., 1948, 13: 134-143.
    • (1948) J. Org. Chem. , vol.13 , pp. 134-143
    • Stewart, H.W.1    Turner, R.J.2    Denton, J.J.3
  • 39
    • 0001666244 scopus 로고
    • Preparation and structural characterization of monoamine-monoamide bis(thio) oxo complexes of technetium(V) and rhenium(V)
    • O'Neil, J. P., Wilson, S. R., Katzenellenbogen, J. A., Preparation and structural characterization of monoamine-monoamide bis(thio) oxo complexes of technetium(V) and rhenium(V), Inorg. Chem., 1994, 33: 319-323.
    • (1994) Inorg. Chem. , vol.33 , pp. 319-323
    • O'Neil, J.P.1    Wilson, S.R.2    Katzenellenbogen, J.A.3
  • 40
    • 0034080806 scopus 로고    scopus 로고
    • Sigma receptors: Recent advances and new clinical potentials
    • Bowen, W. D., Sigma receptors: Recent advances and new clinical potentials, Pharm. Acta Helv., 2000, 74: 211-218.
    • (2000) Pharm. Acta Helv. , vol.74 , pp. 211-218
    • Bowen, W.D.1
  • 41
    • 5044235132 scopus 로고    scopus 로고
    • Norchloro-fluoro-homoepibatidine: Specificity to neuronal nicotinic acetylcholine receptor subtypes in vitro
    • Deuther-Conrad, W., Patt, J. T., Feuerbach, D. et al., Norchloro-fluoro-homoepibatidine: Specificity to neuronal nicotinic acetylcholine receptor subtypes in vitro, IL Farmaco, 2004, 59: 785-792.
    • (2004) IL Farmaco , vol.59 , pp. 785-792
    • Deuther-Conrad, W.1    Patt, J.T.2    Feuerbach, D.3
  • 42
    • 0034053453 scopus 로고    scopus 로고
    • Modulation of cellular calcium by sigma-2 receptors: Release form intracellular stores in human SK-N-SH neuroblastoma cells
    • Vilner, B. J., Bowen, W. D., Modulation of cellular calcium by sigma-2 receptors: Release form intracellular stores in human SK-N-SH neuroblastoma cells, J. Pharmacol. Exp. Ther., 2000, 292: 900-911.
    • (2000) J. Pharmacol. Exp. Ther. , vol.292 , pp. 900-911
    • Vilner, B.J.1    Bowen, W.D.2
  • 44
    • 0029957462 scopus 로고    scopus 로고
    • Imaging of dopamine transporters in humans with technetium-99 m TRODAT-1
    • Kung, H. F, Kim, H-J., Kung, M-P. et al., Imaging of dopamine transporters in humans with technetium-99 m TRODAT-1, Eur. J. Nucl. Med., 1996,23: 1527-1530.
    • (1996) Eur. J. Nucl. Med. , vol.23 , pp. 1527-1530
    • Kung, H.F.1    Kim, H.-J.2    Kung, M.-P.3
  • 45
    • 33745164539 scopus 로고    scopus 로고
    • A phase I clinical trial of the DAT ligand 99 mTc-O1505T
    • Callahan, R. J., Dragotakes, S. C., Barrow, S. A. et al, A phase I clinical trial of the DAT ligand 99 mTc-O1505T, J. Med. Chem., 2003, 46: 3483-3496.
    • (2003) J. Med. Chem. , vol.46 , pp. 3483-3496
    • Callahan, R.J.1    Dragotakes, S.C.2    Barrow, S.A.3


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