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Volumn 8, Issue 3, 1997, Pages 304-309

99mTc-labeled σ-receptor-binding complex: Synthesis, characterization, and specific binding to human ductal breast carcinoma (T47D) cells

Author keywords

[No Author keywords available]

Indexed keywords

ALKYLATION; BIOACTIVITY; CELLS; CYTOLOGY; HIGH PERFORMANCE LIQUID CHROMATOGRAPHY; LIGANDS; PHARMACODYNAMICS; TUMORS;

EID: 0030609924     PISSN: 10431802     EISSN: None     Source Type: Journal    
DOI: 10.1021/bc9700087     Document Type: Article
Times cited : (37)

References (27)
  • 1
    • 0025180755 scopus 로고
    • A σ-like binding site in rat pheochromocytoma (PC12) cells: Decreased affinity for (+)-benzomorphans and lower molecular weight suggest a different σ-receptor form from that in guinea pig brain
    • (a) Hellewell, S. B., and Bowen, W. D. (1990) A σ-like binding site in rat pheochromocytoma (PC12) cells: Decreased affinity for (+)-benzomorphans and lower molecular weight suggest a different σ-receptor form from that in guinea pig brain. Brain Res. 527, 244-253.
    • (1990) Brain Res. , vol.527 , pp. 244-253
    • Hellewell, S.B.1    Bowen, W.D.2
  • 6
    • 0028795145 scopus 로고
    • σ-1 and σ-2 receptors are expressed in a wide variety of human and rodent tumor cell lines
    • Vilner, B. J., John, C. S., and Bowen, W. D. (1995) σ-1 and σ-2 receptors are expressed in a wide variety of human and rodent tumor cell lines. Cancer Res. 55, 408-413.
    • (1995) Cancer Res. , vol.55 , pp. 408-413
    • Vilner, B.J.1    John, C.S.2    Bowen, W.D.3
  • 9
    • 0000475641 scopus 로고    scopus 로고
    • Characterization of σ-receptor binding sites in human biopsied solid breast tumors
    • abstract
    • (c) John, C. S., Vilner, B. J., Schwartz, A. M., and Bowen, W. D. (1996) Characterization of σ-receptor binding sites in human biopsied solid breast tumors. J. Nucl. Med. 37, 267P (abstract).
    • (1996) J. Nucl. Med. , vol.37
    • John, C.S.1    Vilner, B.J.2    Schwartz, A.M.3    Bowen, W.D.4
  • 10
    • 0027141936 scopus 로고
    • A malignant melanoma imaging agent: Synthesis, characterization, in vitro binding and biodistribution of iodine-125-(2-piperidinyl-aminoethyl)-4-iodobenzamide
    • John, C. S., Bowen, W. D., Saga, T., Kinuya, S., Vilner, B. J., Baumgold, J., Paik, C. H., Reba R. C., Neumann, R. D., Varma, V. M., and McAfee, J. G. (1993) A malignant melanoma imaging agent: synthesis, characterization, in vitro binding and biodistribution of iodine-125-(2-piperidinyl-aminoethyl)-4-iodobenzamide. J. Nucl. Med. 34, 2169-2175.
    • (1993) J. Nucl. Med. , vol.34 , pp. 2169-2175
    • John, C.S.1    Bowen, W.D.2    Saga, T.3    Kinuya, S.4    Vilner, B.J.5    Baumgold, J.6    Paik, C.H.7    Reba, R.C.8    Neumann, R.D.9    Varma, V.M.10    McAfee, J.G.11
  • 11
    • 0028182454 scopus 로고
    • 125I]-N-(N-benzylpiperidin-4-yl)-4-iodobenzamide, a new σ-receptor radiopharmaceutical: High affinity binding to MCF-7 breast tumor cells
    • 125I]-N-(N-benzylpiperidin-4-yl)-4-iodobenzamide, a new σ-receptor radiopharmaceutical: high affinity binding to MCF-7 breast tumor cells. J. Med. Chem. 37, 1737-1739.
    • (1994) J. Med. Chem. , vol.37 , pp. 1737-1739
    • John, C.S.1    Vilner, B.J.2    Bowen, W.D.3
  • 13
    • 0029032044 scopus 로고
    • σ-Receptors are expressed in human non-small cell lung carcinoma
    • John, C. S., Bowen, W. D., Varma, V. M., McAfee, J. G., and Moody, T. W. (1995) σ-Receptors are expressed in human non-small cell lung carcinoma. Life Sci. 56, 2385-2392.
    • (1995) Life Sci. , vol.56 , pp. 2385-2392
    • John, C.S.1    Bowen, W.D.2    Varma, V.M.3    McAfee, J.G.4    Moody, T.W.5
  • 14
    • 0010556890 scopus 로고    scopus 로고
    • Characterization and targeting of σ-receptor binding sites in human prostate tumor cells
    • abstract
    • (a) John, C. S., Venugopal, R., Li, J., Bowen, W. D., Varma, V. M., and Thakur, M. L. (1996) Characterization and targeting of σ-receptor binding sites in human prostate tumor cells. J. Nucl. Med. 37, 205P (abstract).
    • (1996) J. Nucl. Med. , vol.37
    • John, C.S.1    Venugopal, R.2    Li, J.3    Bowen, W.D.4    Varma, V.M.5    Thakur, M.L.6
  • 16
    • 0026603216 scopus 로고
    • Technetium- and rhenium-labeled progestins: Synthesis, receptor binding and in-vivo distribution of an 111-substituted progestin labeled with technetium-99 and rhenium-186
    • (a) DiZio, J. P., Anderson, C. J., Davison, A., Ehrhardt, G. J., Carlson, K. E., Welch, M. J., and Katzenellenbogen, J. A. (1992) Technetium-and rhenium-labeled progestins: synthesis, receptor binding and in-vivo distribution of an 111-substituted progestin labeled with technetium-99 and rhenium-186. J. Nucl. Med. 33, 558-569.
    • (1992) J. Nucl. Med. , vol.33 , pp. 558-569
    • DiZio, J.P.1    Anderson, C.J.2    Davison, A.3    Ehrhardt, G.J.4    Carlson, K.E.5    Welch, M.J.6    Katzenellenbogen, J.A.7
  • 19
    • 0028255979 scopus 로고
    • Synthesis and in vivo evaluation of a 99m/99Tc-DADT-benzovesamicol: A potential marker for cholinergic neurons
    • Del Rosario, R. B., Jung, Y.-W., Baidoo, K. E., Lever, S. Z., and Wieland, D. M. (1994) Synthesis and in vivo evaluation of a 99m/99Tc-DADT-benzovesamicol: a potential marker for cholinergic neurons. Nucl. Med. Biol. 21, 197-203.
    • (1994) Nucl. Med. Biol. , vol.21 , pp. 197-203
    • Del Rosario, R.B.1    Jung, Y.-W.2    Baidoo, K.E.3    Lever, S.Z.4    Wieland, D.M.5
  • 20
    • 0026575012 scopus 로고
    • Synthesis, characterization and biological evaluation of a novel class of N-(arylethyl)-N-alkyl-2-(1-pyrrolidinyl)ethylamines: Structural requirements and binding affinity at the σ-receptors
    • de Costa, B. R., Radesca, L., Di Paolo, L., and Bowen, W. D. (1992) Synthesis, characterization and biological evaluation of a novel class of N-(arylethyl)-N-alkyl-2-(1-pyrrolidinyl)ethylamines: structural requirements and binding affinity at the σ-receptors. J. Med. Chem. 35, 38-47.
    • (1992) J. Med. Chem. , vol.35 , pp. 38-47
    • De Costa, B.R.1    Radesca, L.2    Di Paolo, L.3    Bowen, W.D.4
  • 21
    • 0026747748 scopus 로고
    • Synthesis and receptor binding properties of fluoro- and iodo-substituted high affinity σ-receptor ligands: Identification of potential PET and SPECT σ-receptor imaging agents
    • de Costa, B. R., Radesca, L., Dominguez, C., Di Paolo, L., and Bowen, W. D. (1992) Synthesis and receptor binding properties of fluoro-and iodo-substituted high affinity σ-receptor ligands: Identification of potential PET and SPECT σ-receptor imaging agents. J. Med. Chem. 35, 2221-2230.
    • (1992) J. Med. Chem. , vol.35 , pp. 2221-2230
    • De Costa, B.R.1    Radesca, L.2    Dominguez, C.3    Di Paolo, L.4    Bowen, W.D.5
  • 22
    • 4244000670 scopus 로고
    • Synthesis, binding characteristics and in-vivo clearance of 4-[I-125]PEMP: A σ-receptor ligand for imaging tumors
    • abstract
    • (a) John, C. S., Vilner, B. J., and Bowen, W. D. (1995) Synthesis, binding characteristics and in-vivo clearance of 4-[I-125]PEMP: a σ-receptor ligand for imaging tumors. J. Nucl. Med. 36, 6P (abstract).
    • (1995) J. Nucl. Med. , vol.36
    • John, C.S.1    Vilner, B.J.2    Bowen, W.D.3
  • 23
    • 0030220443 scopus 로고    scopus 로고
    • 125I]N-[2-(4-iodophenyl)ethyl]-N-methyl-2-(1-piperidinyl)ethylamine: A high affinity ligand for imaging σ-receptor-positive tumors
    • 125I]N-[2-(4-iodophenyl)ethyl]-N-methyl-2-(1-piperidinyl)ethylamine: a high affinity ligand for imaging σ-receptor-positive tumors. Nucl. Med. Biol. 23, 761-766.
    • (1996) Nucl. Med. Biol. , vol.23 , pp. 761-766
    • John, C.S.1    Gulden, M.E.2    Vilner, B.J.3    Bowen, W.D.4
  • 24
    • 0001528499 scopus 로고
    • Transannular cyclizations of 1,2-dithia-5,8-diazacyclodeca-4,8-dienes during borohydride reduction
    • Joshua, A. V., Scott, J. R., Sondhi, S. M., Ball, R. G., and Lown, J. W. (1987) Transannular cyclizations of 1,2-dithia-5,8-diazacyclodeca-4,8-dienes during borohydride reduction. J. Org. Chem. 52, 2447-2451.
    • (1987) J. Org. Chem. , vol.52 , pp. 2447-2451
    • Joshua, A.V.1    Scott, J.R.2    Sondhi, S.M.3    Ball, R.G.4    Lown, J.W.5
  • 25
    • 0026215304 scopus 로고
    • Progestin-rhenium complexes: Metal-labeled steroids with high receptor binding affinity, potential receptor-directed agents for diagnostic imaging or therapy
    • (a) DiZio, J. P., Fiaschi, R., Davison, A., Jones, A. G., and Katzenellenbogen, J. A. (1991) Progestin-rhenium complexes: metal-labeled steroids with high receptor binding affinity, potential receptor-directed agents for diagnostic imaging or therapy. Bioconjugate Chem. 2, 353-366.
    • (1991) Bioconjugate Chem. , vol.2 , pp. 353-366
    • DiZio, J.P.1    Fiaschi, R.2    Davison, A.3    Jones, A.G.4    Katzenellenbogen, J.A.5
  • 26
    • 0001636391 scopus 로고
    • Stereoisomers of neutral oxotechnetium(V) and oxorhenium(V) complexes
    • (M. Nicolini, G. Bandoli, and U. Mazzi, Eds.) Cortina International, Verona
    • (b) Mahmood, A., Baidoo, K. E., and Lever, S. Z. (1990) Stereoisomers of neutral oxotechnetium(V) and oxorhenium(V) complexes. In Techneium in Chemistry and Nuclear Medicine (M. Nicolini, G. Bandoli, and U. Mazzi, Eds.) Vol. 3, pp 119-124, Cortina International, Verona.
    • (1990) Techneium in Chemistry and Nuclear Medicine , vol.3 , pp. 119-124
    • Mahmood, A.1    Baidoo, K.E.2    Lever, S.Z.3
  • 27
    • 0028180570 scopus 로고
    • Rat liver and kidney contain high densities of σ-1 and σ-2 receptors: Characterization by ligand binding and photoaffinity labeling
    • Hellewell, S. B., Bruce, A., Feinstein, G., Orringer, J., Williams, W., and Bowen, W. D. (1994) Rat liver and kidney contain high densities of σ-1 and σ-2 receptors: characterization by ligand binding and photoaffinity labeling. Eur. J. Pharmacol., Mol. Pharmacol. Sect. 268, 9-18.
    • (1994) Eur. J. Pharmacol., Mol. Pharmacol. Sect. , vol.268 , pp. 9-18
    • Hellewell, S.B.1    Bruce, A.2    Feinstein, G.3    Orringer, J.4    Williams, W.5    Bowen, W.D.6


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.