Evaluation of mismatch-binding ligands as inhibitors for Rev-RRE interaction

Bioorganic and Medicinal Chemistry

Volumn 14, Issue 15, 2006, Pages 5384-5388

  Nakatani, Kazuhiko ^a,b   Horie, Souta ^a   Goto, Yuki ^a   Kobori, Akio ^a   Hagihara, Shinya ^a  

^a KYOTO UNIVERSITY   (Japan)

^b OSAKA UNIVERSITY   (Japan)

Author keywords

Drug design; HIV 1 RRE; Inhibitors; RNA recognition

Indexed keywords

DOUBLE STRANDED DNA; FRAMYCETIN; NAPHTHYRIDINE DERIVATIVE; QUINOLONE DERIVATIVE; REV PROTEIN; REV RESPONSIBLE ELEMENT; UNCLASSIFIED DRUG; VIRUS RNA;

ARTICLE; COMPLEX FORMATION; DNA BINDING; HUMAN IMMUNODEFICIENCY VIRUS; LIGAND BINDING; PROTEIN RNA BINDING;

BASE PAIR MISMATCH; BASE SEQUENCE; BINDING SITES; BINDING, COMPETITIVE; DNA; DRUG EVALUATION, PRECLINICAL; FLUORESCENCE POLARIZATION; GENE PRODUCTS, REV; GENES, ENV; HIV-1; LIGANDS; MOLECULAR SEQUENCE DATA; MOLECULAR STRUCTURE; NAPHTHYRIDINES; NUCLEIC ACID CONFORMATION; POLYAMINES; PROTEIN BINDING; QUINOLONES; RNA, VIRAL; SURFACE PLASMON RESONANCE; TIME FACTORS;

HUMAN IMMUNODEFICIENCY VIRUS 1;

EID: 33745148276     PISSN: 09680896     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmc.2006.03.038     Document Type: Article

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