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Volumn 16, Issue 7, 2006, Pages 1965-1968

A novel series of urea-based peptidomimetic calpain inhibitors

Author keywords

Calpain inhibitors; Peptidomimetic; Peptidyl aldehyde inhibitors; Urea based calpain inhibitors

Indexed keywords

[1 [(1 FORMYL 2 PHENYLETHYL)CARBAMOYL] 2 METHYLPROPYL]CARBAMIC ACID BENZYL ESTER; ALDEHYDE DERIVATIVE; CALPAIN; CALPASTATIN; CARBON; CATHEPSIN B; NITROGEN; PEPTIDE DERIVATIVE; UREA DERIVATIVE;

EID: 33144476326     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2005.12.068     Document Type: Article
Times cited : (9)

References (29)
  • 22
    • 33144462718 scopus 로고    scopus 로고
    • note
    • i values are the average of duplicate determinations.
  • 23
    • 33144484824 scopus 로고    scopus 로고
    • note
    • i values for inhibition of human liver cathepsin B were determined as described for calpain using a reaction mixture containing 14 ng human liver cathepsin B (Calbiochem), 20 mM NaOAc (pH 6.0), 1 mM EDTA, 0.5 mM DTT, 50 μM or 250 μM Z-Arg-Arg-AMC, and varying concentrations of inhibitor dissolved in DMSO (2% total concentration) in a final volume of 200 μL.


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.