Chromatography studies on bio-affinity of nine ligands of α1-adrenoceptor to α1D subtypes overexpressed in cell membrane

Science in China, Series C: Life Sciences

Volumn 47, Issue 4, 2004, Pages 376-381

  Zhang, Dian ^a   Yuan, Bingxiang ^a   Deng, Xiuling ^a   Yang, Guangde ^a   He, Langchong ^a   Zhang, Youyi ^b   Han, Qide ^b  

^a XI'AN JIAOTONG UNIVERSITY   (China)

^b PEKING UNIVERSITY   (China)

Author keywords

1 adrenergic receptor; 1D adrenoceptor subtype; Cell membrane; Chromatography

Indexed keywords

AFFINITY CHROMATOGRAPHY; BIOASSAY; BIOLOGICAL MEMBRANES; BIOLOGICAL ORGANS; BIOMEDICAL ENGINEERING; CELLS;

1 ADRENERGIC RECEPTOR; 1D ADRENOCEPTOR SUBTYPE; CELL MEMBRANE; CELL MEMBRANE CHROMATOGRAPHY (CMC);

CELL MEMBRANES;

ALPHA 1 ADRENERGIC RECEPTOR; LIGAND;

AFFINITY CHROMATOGRAPHY; ARTICLE; CELL LINE; CELL MEMBRANE; CLASSIFICATION; DRUG SCREENING; GENE EXPRESSION; GENETIC TRANSFECTION; GENETICS; HUMAN; METABOLISM;

CELL LINE; CELL MEMBRANE; CHROMATOGRAPHY, AFFINITY; DRUG EVALUATION, PRECLINICAL; GENE EXPRESSION; HUMANS; LIGANDS; RECEPTORS, ADRENERGIC, ALPHA-1; TRANSFECTION;

EID: 32244444283     PISSN: 10069305     EISSN: None     Source Type: Journal    
DOI: 10.1360/03yc0109     Document Type: Article

References (17)

1. 2 -adrenoceptors, Eur. J. Pharmacol., 1998, 361: 1-15.
2. 1-Adrenoceptor subtypes linked to different mechanisms for increasing intracellular calcium in smooth muscle, Nature, 1987, 329: 333-335.
3. 1- and β-adrenoceptors, Basic Medical Sciences And Clinics (in Chinese), 1997, 17(4): 1-1.
4. 1-adrenergic receptor, Proc. Natl. Acad. Sci. USA, 1988, 85: 7159-7163.
5. 1-adrenergic receptor subtype, J. Biol. Chem., 1990, 265: 8183-8189.
6. 1dadrenergic receptor and inducible expression of three human subtypes in SK-N-MC cells, Mol. Pharmacol., 1995, 47: 977-985.
7. IUPHAR Committee of Receptor Nomenclature and Drug Classification, Trends Pharmacol. Sci., Nomenclature Suppl., 1995, 16-9.
8. He, L. C., Wang, S. C., Geng, X. D., Coating and fusing cell membranes onto a silica surface and their chromatographic characteristics, Chromatographia, 2001, 54: 71-76.
9. He, L. C., Yang, G D., Geng, X. D., Enzymatic activity and chromatography characteristics of the cell membrane immobilized on silica surface, Chinese Science Bulletin, 1999, 44(9): 826-830.
10. 1-adrenoceptor recognition sites by urapidil derivatives and other selective antagonists. Br. J. Pharmacol, 1989, 97: 691-695.
11. 1A- adrenergic receptor mediated the presser response to phenylephrine in anesthetized rat, Science in China, Ser. C, 2003, 33(2): 133-138.
12. 1d- adrenoceptor subtype is involved in the Noradrenaline-induced contractions of rat aorta, Life Sci., 1995, 57(13): 159-163.
13. 1d- adrenoceptor-induced contractility in rat aorta is mediated by the a1D subtype, Eur. J. Pharmacol., 1996, 297: 241-248.
14. 1 adrenoceptor subtype selective antagonists, Bioorg. Med. Chem., 2000, (8): 201-204.
15. Gao, K., He, L. C., Yang, G. D., Screening the effective component of Leontice robustum by cell membrane chromatography, Chin. Pharm. J. (in Chinese), 2003, 38(1): 14-16.
16. Zhao, H. R., Yang, G D., He, L. C. et al., Screening the effective component of Angelica sinensis by cell membrane chromatography, Chin. Pharm. J. (in Chinese), 2000, 35(1): 13-15.
17. Hou, J., Yuan, B.X., He, L.C. et al., Evaluation of drug-muscarinic receptor affinities by using cell membrane chromatography. Chin. J. Pharmacol. Toxicol., 2003, 17(1): 70-73.