PEG-derivative effectively modifies the characteristics of indomethacin-PLGA microspheres destined to intra-articular administration

Journal of Microencapsulation

Volumn 22, Issue 7, 2005, Pages 793-808

  Puebla, Patricia ^a   Pastoriza, Pilar ^a   Barcia, Emilia ^a   Fernández Carballido, Ana ^a  

^a UNIVERSIDAD COMPLUTENSE DE MADRID   (Spain)

Author keywords

Indomethacin; Intra articular; Microspheres; PL PEG derivative; Rheumatoid arthritis

Indexed keywords

ANTIINFLAMMATORY AGENT; BIOPOLYMER; INDOMETACIN; MACROGOL; MICROSPHERE; OIL; POLYGLACTIN; SOLVENT; WATER;

ANGIOGENESIS; ANIMAL CELL; ANTIANGIOGENIC ACTIVITY; ANTIINFLAMMATORY ACTIVITY; ARTICLE; BIODEGRADABILITY; CELL VIABILITY; CONTROLLED STUDY; CRYSTALLIZATION; CYTOTOXICITY TEST; DRUG FORMULATION; DRUG RELEASE; DRUG SOLUBILITY; EVAPORATION; MICROENCAPSULATION; MICROMORPHOLOGY; NONHUMAN; RAT; RHEUMATOID ARTHRITIS; SPLEEN CELL;

ANTIRHEUMATIC AGENTS; DRUG ADMINISTRATION SCHEDULE; DRUG COMPOUNDING; INDOMETHACIN; INJECTIONS, INTRA-ARTICULAR; LACTIC ACID; MICROSPHERES; POLYETHYLENE GLYCOLS; POLYGLYCOLIC ACID; POLYMERS;

EID: 31544465524     PISSN: 02652048     EISSN: 14645246     Source Type: Journal    
DOI: 10.1080/02652040500273902     Document Type: Article

References (31)

1. Blanco-Prieto, MJ and Besseghir, K and Zerbe, O and Andris, D and Orsolini, F and Heingartiner, P and Merkle, HP and Gander, B. (2000) In vitro and in vivo evaluation of a somatostatin analogue released from PLGA microspheres Journal of Controlled Release, 67, pp. 19 - 28.
2. Capsoni, F and Sarzi-Puttini, P and Atzeri, F and Minonzio, F and Bonara, P and Doria, A and Carraba, M. (2005) Effect of adalimumad on neutrofil function in patients with rheumatoid arthritis Arthritis Research and Therapy, 7, pp. R250 - R255.
3. Choi, Y and Kim, SY and Kim, SH and Lee, KS and Kim, C and Byun, Y. (2001) Long-term delivery of all-trans-retinoic acid using biodegradable PLLA/PEG-PLLA blended microspheres International Journal of Pharmaceutics, 215, pp. 67 - 81.
4. Elmquist, WF and Keith, KH and Sawchuk, RJ. (1994) Transsynovial drug distribution: Synovial mean transit time of diclofenac and other nonsteroidal antiinflammatory drugs Pharmaceutical Research, 11, pp. 1689 - 1699.
5. Fernández-Carballido, A and Herrero-Vanrell, R and Molina-Martínez, IT and Pastoriza, P. (2004a) Sterilizad ibuprofen-loaded poly(D,L-lactide-co-glycolide) microspheres for intraarticular administration: Effect of γ-irradiation and storage Journal of Microencapsulation, 21, pp. 653 - 665.
6. Fernández-Carballido, A and Herrero-Vanrell, R and Molina-Martínez, IT and Pastoriza, P. (2004b) Biodegradable ibuprofen loaded PLGA microspheres for intraarticular administration. Effect of Labrafil addition on release in vitro International Journal of Pharmaceutics, 27, pp. 33 - 41.
7. Fini, A and Rodriguez, L and Cavallari, C and Albertini, B and Passerini, N. (2002) Utrasound-compacted and spray-congealed indomethacin/polyethyleneglycol systems International Journal of Pharmaceutics, 247, pp. 11 - 22.
8. Gao, Z and Crowley, WR and Shukla, AJ and Johnson, JR and Reger, JF. (1995) Controlled release of contraceptive steroids from biodegradable and injectable gel formulations: In vivo evaluation Pharmaceutical Research, 12, pp. 864 - 868.
9. Gasparini, G and Longo, R and Sarmiento, R and Morabito, A. (2003) Inhibitors of cyclooxygenase 2: A new class of anticancer agents? Oncology, 4, pp. 605 - 615.
10. Ghosh, AK and Hirasawa, N and Niki, H and Ohuchi, K. (2000) Cyclooxygenase-2-mediated angiogenesis in carrageenin-induced granulation tissue in rats Journal of Pharmacology and Experimental Therapeutics, 295, pp. 802 - 809.
11. Hedberg, EL and Tang, A and Crowther, RS and Carney, DH and Mikos, A. (2002) Controlled release of an osteogenic peptide from injectable biodegradable polymeric composites Journal of Controlled Release, 84, pp. 137 - 150.
12. Herrero-Vanrell, R and Ramírez, L and Fernández-Carballido, A and Refojo, MF. (2000) Biodegradable PLGA microspheres loaded with Ganciclovir for intraocular administration Encapsulation technique, in-vitro release profiles, and sterilization process Pharmaceutical Research, 17, pp. 1323 - 1328.
13. Iñiguez, MA and Rodriguez, A and Volpert, O and Fresno, M and Redondo, JM. (2003) Cyclooxygenase-2: A therapeutic target in angiogenesis Trends in Molecular Medicine, 9, pp. 73 - 78.
14. Karasulu, E and Karasulu, HY and Ertan, G and Kirilmaz, L and Güneri, T. (2003) Extended release lipophilic indomethacin microspheres: Formulation factors and mathematical equation fitted drug release rate European Journal of Pharmaceutical Science, 19, pp. 99 - 104.
15. Kim, JH and Choi, HK. (2002) Effect of additives on the crystallization and the permeation of ketoprofen from adhesive matrix International Journal of Pharmaceutics, 236, pp. 81 - 85.
16. Lemaire, V and Belair, J and Hildgen, P. (2003) Structural modelling of drug release from biodegradable porous matrices based on a combined diffusion/erosion process International Journal of Pharmaceutics, 258, pp. 95 - 107.
17. Li, G and Yang, T and Yan, J. (2002) Cyclooxygenase-2 increased the angiogenic and metastatic potential of tumour cells Biochemical and Biophysical Research Communications, 299, pp. 886 - 890.
18. Lin, SY and Chen, KS and Teng, HH and Li, MJ. (2000) In vitro degradation and dissolution behaviours of microspheres prepared by three low molecular weight polyesters Journal of Microencapsulation, 17, pp. 577 - 586.
19. Mallard, C and Coudane, J and Rault, I and Vert, M. (2000) The use of additives to modulate the release of sparingly water soluble drug entrapped in PLA50 microparticles Journal of Microencapsulation, 17, pp. 81 - 93.
20. Martinez-Sancho, C and Herrero-Vanrell, R and Negro, S. (2004) Optimisation of aciclovir poly (D,L-lactide-co-glycolide) microspheres for intravitreal administration using a factorial design study International Journal of Pharmaceutics, 273, pp. 45 - 56.
21. Martinez-Sancho, C and Herrero-Vanrell, R and Negro, S. (2003) Poly (D, L, lactide-co-glycolide) microspheres for long-term intravitreal delivery of aciclovir: Influence of fatty and non fatty additives Journal of Microencapsulation, 20, pp. 799 - 810.
22. Ruan, G and Feng, S. (2003) Preparation and characterization of poly(lactic-acid)-polyethy(eneglycol)-poly(lactic acid) (PLA-PEG-PLA) microspheres for controlled release of paclitaxel Biomaterials, 24, pp. 5037 - 5044.
23. Sales, KJ and Katz, AA and Howard, B and Soeters, RP and Millar, RP and Jabbour, HN. (2002) Cyclooxygenase-1 is upregulated in cervical carcinomas Autocrine/paracrine regulation of cyclooxygenase-2, prostaglandin E receptors, and antiangiogenic factors by cyclooxygenase-1. Cancer Research, 62, pp. 424 - 432.
24. Sato, Y and Kawashima, Y and Takeuchi, H and Yamamoto, H. (2004) In vitro evaluation of floating and drug releasing behaviors of hollow microspheres (microballoons) prepared by emulsion solvent diffusion method European Journal of Pharmaceutics and Biopharmaceutics, 57, pp. 235 - 243.
25. Siepmann, J and Peppas, NA. (2000) Hydrophilic matrices for controlled drug delivery: An improved mathematical model to predict the resulting drug release kinetics (the 'sequential layer' model) Pharmaceutical Research, 17, pp. 1290 - 1298.
26. Steinmeyer, J. (2001) Pharmacotherapy in osteoarthritis Orthopade, 30, pp. 856 - 865.
27. Suzuki, N and Takahashi, S and Okade, S. (1998) Relationship between vascular endothelial growth factor and angiogenesis in spontaneous and indomethacin-delayed healing of acetic acid-induced gastric ulcer in rats Journal of Physiology and Pharmacology, 49, pp. 515 - 527.
28. Terada, K and Kitano, H and Yoshihashi, Y and Yonemochi, E. (2000) Quantitative correlation between initial dissolution rate and heat of solution of drug Pharmaceutical Research, 17, pp. 920 - 924.
29. 2α-induced vascular endhotelial growth factor synthesis in osteoblasts Enhancement of MAPK activity. Journal of Biological Chemistry, 278, pp. 18930 - 18937.
30. Tunçay, M and Calis, S and Kas, HS and Ercan, MT and Peksoy, I and Hincal, AA. (2000) Diclofenac sodium incorporated PLGA (50:50) microspheres: Formulations considerations and in vitro/in vivo evaluation International Journal of Pharmaceutics, 17, pp. 179 - 188.
31. Villaseñor-Garcia, MM and Puebla-Perez, AM and Sandoval-Ramirez, L and Lozoya, X. (2000) Phenytoin and electric shock-induced apoptosis in rat peripheral blood lymphocytes International Journal of Immunopharmacology, 22, pp. 143 - 150.