Correlation between in vitro release from topical delivery vehicles and microbicidal activity of triclosan

Pharmazie

Volumn 61, Issue 1, 2006, Pages 35-40

  Swart, H C ^a   Du Preez, J L ^a   De Villiers, M M ^b   Lotter A P ^a   Liebenberg, Wilna ^a  

^a NORTH WEST UNIVERSITY   (South Africa)

^b UNIVERSITY OF LOUISIANA AT MONROE   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

AEROSIL; ANTIINFECTIVE AGENT; ARACHIS OIL; CASTOR OIL; CETYL STEARY 2 ETHYL HEXANOATE; CITRIC ACID; EXCIPIENT; GLYCEROL STEARATE; GUAIACOL; LIQUID PARAFFIN; METHYL HYDROXYBENZOATE; MICROBICIDE; MYRISTYL ETHER PROPIONATE; POLYOXYETHYLENE SORBITAN MONOLEATE; PROPOLIS; PROPYL PARABEN; PROPYLENE GLYCOL; SILICON DIOXIDE; SORBITAN OLEATE; SORBITOL; STEARIC ACID; TRICLOSAN; UNCLASSIFIED DRUG;

AEROSOL; ANTIMICROBIAL ACTIVITY; ARTICLE; CREAM; DRUG DELIVERY SYSTEM; DRUG FORMULATION; DRUG RELEASE; DRUG STABILITY; EMULSION; GEL; GRAM NEGATIVE BACTERIUM; GRAM POSITIVE BACTERIUM; IN VITRO STUDY; NONHUMAN; STORAGE TEMPERATURE;

ADMINISTRATION, TOPICAL; ANTI-INFECTIVE AGENTS, LOCAL; BACTERIA; CHEMISTRY, PHARMACEUTICAL; CHROMATOGRAPHY, HIGH PRESSURE LIQUID; DRUG STABILITY; MICROBIAL SENSITIVITY TESTS; SPECTROPHOTOMETRY, ULTRAVIOLET; TRICLOSAN; VEHICLES;

EID: 31144473570     PISSN: 00317144     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Article

References (19)

1. Borsadia S, Ghanem AH, Seta Y, Higuchi WI, Flynn GL, Behl CR, Shah VP (1992) Factors to be considered in the evaluation of bioavailability and bioequivalence of topical formulations. Skin Pharmacol 5: 129-145.
2. Grove C, Liebenberg W, Du Preez JL, Yang W, De Villiers MM (2003) Improving the aqueous solubility of triclosan by solubilization, complexation and in-situ salt formation. J Cosmet Sci 54: 537-550.
3. Guillen J, Bernabeu A, Shapiro S, Villalain J (2004) Location and orientation of triclosan in phospholipid model membranes. Eur Biophys J 33: 448-453.
4. Higuchi T (1960) Physical chemical analysis of percutaneous absorption process from creams and ointments. J Soc Cosmet Chem 11: 85-97.
5. ICH-Q2A (1995) Text on validation of analytical procedures. ICH Secretariat, Geneva, Switzerland.
6. Jones RD, Jampani HB, Newman JL, Lee AS (2000) Triclosan: a review of effectiveness and safety in health care settings. Am J Infect Control 28: 184-196.
7. Loftsson T, Leeves N, Bjornsdottir N, Duffy L, Masson M (1999) Effect of cyclodextrins and polymers on triclosan availability and substantivity in toothpastes in vivo, J Pharm Sci 88: 1254-1258.
8. Lu J, Hill MA, Hood M, Greeson DF, Horton JR, Orndorff PE, Herndon AS, Tonelli AE (2001) Formation of antibiotic, biodegradable polymers by processing with Irgasan DP 300R (triclosan) and its inclusion compound with β-cyclodextrin, J Fiber Pol Sci 82: 300-309.
9. Narsai K, De Villiers MM, Du Plessis J (1997) The effect of a change in ionic character on the rheological properties of stearate type o/w creams containing α-hydroxy acids. Pharmazie 52: 486-487.
10. Nissan HP, Ochs D (1998) Triclosan: an antimicrobial active ingredient with anti-inflammatory activity. Cosmet Toil 113: 61-64.
11. Ramachandra RSP, Surolia A, Surolia, N (2003) Triclosan: A shot in the arm for antimalarial chemotherapy. Mol Cell Biochem 253: 55-63.
12. Rege PR, Vilivalam VD, Collins CC (1998) Development in release testing of topical dosage forms: use of the Enhancer Cell with automated sampling. J Pharm Biomed Anal 17: 1226-1233.
13. Savage CA (1971) A new bacteriostat for skin care products. Drug Cosmet Ind 109: 36-38, 163.
14. Surolia N, Surolia A (2001) Triclosan offers protection against blood stages of malaria by inhibiting enoyl-ACP reductase of Plasmodium falciparum. Nature Med 7: 636.
15. Taylor TJ, Seitz EP, Fox P, Fischler GE, Fuis JL, Weidner PL (2004) Physicochemical factors affecting the rapid bactericidal efficacy of the phenolic antibacterial triclosan. Int J Cosmet Sci 26: 111-116.
16. The United States Pharmacopeia (2000) 24th Revision. United States Pharmacopeial Convention, Rockville, MD.
17. Toricht E, Eros I (1977) Study of salves with highly dispersed silicon dioxide. Part 2: colloidal physical and rheological stability of gels with Aerosil and Syloid. Pharmazie 32: 169-171.
18. Villalain J, Mateo C, Reyes AFJ, Shapiro S, Micol V (2001) Membranotropic effects of the antibacterial agent triclosan. Arch Biochem Biophys 390: 128-136.
19. Waaler SM, Roella G, Skjoerland KK, Oegaard B (1993) Effects of oral rinsing with triclosan and sodium lauryl sulphate on dental plaque formation: a pilot study. Scan J Den Res 101: 192-195.