Synthesis and antiplasmodial activity in vitro of new ferrocenechloroquine analogues

Dalton Transactions

Volumn , Issue 15, 2003, Pages 3046-3051

  Beagley, Paul ^a   Blackie, Margaret A L ^a   Chibale, Kelly ^a   Clarkson, Cailean ^a   Meijboom, Reinout ^a   Moss, John R ^a   Smith, Peter J ^a   Su, Hong ^a  

^a UNIVERSITY OF CAPE TOWN   (South Africa)

Author keywords

[No Author keywords available]

Indexed keywords

ETHANE; SYNTHESIS (CHEMICAL); X RAY CRYSTALLOGRAPHY;

ANTIPLASMODIAL ACTIVITY; CHLOROQUINOLIN; DIAMINE; DIMETHYLAMINOMETHYLFERROCEN;

ORGANIC COMPOUNDS;

EID: 3042776362     PISSN: 14779226     EISSN: None     Source Type: Journal    
DOI: 10.1039/b303335j     Document Type: Article

References (26)

1. P. A. Winstanley, Parasitol. Today, 2000,16, 146.
2. Weekly Epidemioloeical Record, W.H.O., 1997, vol. 72 (No I, II, III), p. 1.
3. T. J. Egan, Expert Opin. Ther. Pat., 2001, 11, 185 and references therein.
4. (a) R. A. Sánchez-Delgado, M. Navarro, H. Pérez and J. A. Urbina, J. Med. Chem., 1996, 39, 1095;
5. (b) M. Navarro, H. Pérez and R. A. Sánchez-Delgado, J. Med. Chem., 1997, 40, 1937;
6. (c) N. Wasi and H. B. Singh, Synth. React. Inorg. Met.-Org. Chem., 1988, 18, 473;
7. (d) N. Wasi and H. B. Singh, Synth. React. Inorg. Met-Org. Chem., 1987, 17, 129;
8. (e) N. Wasi, H. B. Singh, A. Gajanana and A. N. Raichowdhary, Inorg. Chim. Acta, 1987, 135, 133.
9. C. Biot, G. Glorian, L. A. Maciewski, J. S. Brocard, O. Domarle, G. Blampain, P. Millet, A. J. Georges, H. Abessolo, D. Dive and J. Lebibi, J. Med. Chem., 1997, 40, 3715.
10. M. A. L. Blackie, P. Beagley, J. R. Moss, H. Kendrick, S. L. Croft and K. Chibale, submitted for publication.
11. K. Chibale, J. R. Moss, M. Blackie, D. van Schalkwyk and P. J. Smith, Tetrahedron Lett., 2000, 41, 6231.
12. P. Beagley, M. A. L. Blackie, K. Chibale, C. Clarkson, J. R. Moss and P. J. Smith, J. Chem. Soc.. Dalton Trans., 2002, 4426.
13. (a) S. Picart-Goetgheluck, O. Delacroix, L. Maciejewski and J. Brocard, Synthesis, 2000, 10, 1421;
14. (b) K. Schlögl and M. Walser, Tetrahedron Lett., 1968, 9, 5885.
15. M. E. Wright, Organometallics, 1990, 9, 853.
16. R. Meijboom, A. T. Hutton and J. R. Moss, Organometallics, 2003, 22, 1811.
17. M. Schlosser, in Organometallics in Synthesis, a manual, ed. M. Schlosser, Wiley, Chichester, 1994, ch 1.2, pp. 9-11.
18. D. De, L. D. Byer and D. J. Krogstad, Heterocyclic Chem., 1997, 34, 315.
19. I. R. Butler, in Inorganic Experiments, ed. J. D. Woollins, VCH, Weinheim, 1994, ch. 3, pp. 61-66.
20. G. S. Silverman, in Handbook of Grignard Reagents, ed. G. S. Silverman and P. E. Rakita, Marcel Dekker, Inc., New York, 1996, ch. 6, pp. 89-92.
21. A. L. Wayda and J. L. Dye, J. Chem. Educ., 1985, 62, 356.
22. W. Trager and J. B. Jensen, Science, 1976, 193, 673.
23. COLLECT, Data Collection Software, Nonius B.V., Delft, The Netherlands, 2000.
24. Z. Otwinoski and W. Minor, Methods Enzymol., 1997, 276, 307.
25. G. M. Sheldrick, SHELX97, Program for solving crystal structures, University of Göttingen, Göttingen, Germany, 1997.
26. L. J. Barbour, X-Seed graphical interface for the SHELX program, University of MissouriColumbia, USA, 1999.