Modulation of the stimulus effects of (+)amphetamine by the 5-HT 6 antagonist MS-245

Pharmacology Biochemistry and Behavior

Volumn 78, Issue 2, 2004, Pages 263-268

  Pullagurla, Manik ^a   Bondareva, Tatiana ^a   Young, Richard ^a   Glennon, Richard A ^a  

^a VIRGINIA COMMONWEALTH UNIVERSITY   (United States)

Author keywords

Amphetamine; Cocaine; Dopamine; Drug abuse; Parkinsonism

Indexed keywords

1 BENZENESULFONYL 5 METHOXY N,N DIMETHYLTRYPTAMINE; AMPHETAMINE; COCAINE; SEROTONIN 6 RECEPTOR; SEROTONIN ANTAGONIST; SODIUM CHLORIDE; UNCLASSIFIED DRUG;

ANIMAL BEHAVIOR; ANIMAL EXPERIMENT; ARTICLE; CONTROLLED STUDY; DISCRIMINATION LEARNING; DRUG DOSE; DRUG EFFECT; DRUG RESPONSE; MALE; MODULATION; NONHUMAN; PRIORITY JOURNAL; RAT; STIMULATION;

AMPHETAMINE; ANIMALS; DOSE-RESPONSE RELATIONSHIP, DRUG; MALE; RATS; RATS, SPRAGUE-DAWLEY; RECEPTORS, SEROTONIN; SEROTONIN ANTAGONISTS; TRYPTAMINES;

ANIMALIA;

EID: 3042594449     PISSN: 00913057     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.pbb.2004.03.017     Document Type: Article

References (29)

1. Arnt J. The discriminative stimulus properties of the D-1 agonist SK&F 38393 and the D-2 agonist (-)-NPA are mediated by separate mechanisms. Life Sci. 42:1988;565-574
2. Barrett R.L., Appel J.B. Effects of stimulation and blockade of dopamine receptor subtypes on the discriminative stimulus properties of cocaine. Psychopharmacology. 99:1989;13-16
3. Callahan P.M., Appel J.B., Cunningham K.A. Dopamine D1 and D2 mediation of the discriminative stimulus properties of D-amphetamine and cocaine. Psychopharmacology. 103:1991;50-55
4. 1-like agonists, SKF 81297, SKF 82958 and A-77636, with cocaine: locomotor activity and drug discrimination studies in rodents. Psychopharmacology. 159:2002;145-153
5. Colpaert F.C., Slangen J.L. Drug discrimination: applications in CNS pharmacology. 1982;Elsevier, Amsterdam
6. Costanza R.M., Terry P. The dopamine D4 antagonist L-745, 870: effects in rats discriminating cocaine from saline. Eur. J. Pharmacol. 345:1998;129-132
7. 6 receptor antagonist SB-271046 selectively enhances excitatory neurotransmission in the rat frontal cortex. Neuropharmacology. 25:2001;662-668
8. 6 receptor antagonist. Brain Res. Bull. 59:2002;513-521
9. Elliot E.E., Sibley D.R., Katz J.L. Locomotor and discriminative-stimulus effects of cocaine in dopamine D5 receptor knockout mice. Psychopharmacology. 169:2003;161-168
10. 2C) receptors in rat prefrontal cortex. J. Pharmacol. Exp. Ther. 306:2003;734-743
11. Filip M., Przegalinski E. The role of dopamine receptor subtypes in the discriminative stimulus effects of amphetamine and cocaine in rats. Pol. J. Pharmacol. 49:1997;21-30
12. 6 receptor antagonism potentiates the behavioral and neurochemical effects of amphetamine but not cocaine. Neuropharmacology. 42:2000;170-180
13. 2 receptors in mediating the D-amphetamine discriminative cue. Eur. J. Pharmacol. 202:1991;191-199
14. 7. J. Med. Chem. 46:2003;2795-2812
15. Glennon R.A., Jarbe T.U.C., Frankenheim J. Drug discrimination: application in drug abuse research. NIDA Research Monograph. vol. 116:1991;U.S. Government Printing Office, Washington (DC)
16. Glennon R.A., Young A.M., Martin B.R., DalCason T.A. Methcathinone ("Cat"): an enantiomeric potency comparison. Pharmacol. Biochem. Behav. 50:1995;601-606
17. 6 receptors. J. Med. Chem. 43:2000;1011-1018
18. Goudie A.J. Discriminative stimulus properties of amphetamine, cathinone, and related agents. Glennon R.A., Jarbe T.U.C., Frankenheim J. Drug discrimination: applications to drug abuse research. NIDA Research Monograph. vol. 116:1991;45-60 U.S. Government Printing Office, Washington (DC)
19. Hoyer D., Hannon J.P., Martin G.R. Molecular, pharmacological and functional diversity of 5-HT receptors. Pharmacol. Biochem. Behav. 71:2002;533-554
20. Nielsen E.B., Randrup K., Andersen P.H. Amphetamine discrimination: effects of dopamine receptor agonists. Eur. J. Pharmacol. 160:1989;253-262
21. Rachna S.S., Nader M.A. Modulation of cocaine's discriminative stimulus effects by dopamine D1 agonists in rhesus monkeys. Pharmacol. Biochem. Behav. 68:2001;301-309
22. 6 receptor ligands and their biological functions. Curr. Top. Med. Chem. 2:2002;643-654
23. 6 receptor antagonists for the treatment of CNS diseases. Expert. Opin. Ther. Pat. 12:2002;513-527
24. 1 agonists. Psychopharmacology. 133:1997;282-292
25. Webster R.A. Dopamine (DA). Webster R.A. Neurotransmitters, drugs and brain function. 2001;137-161 Wiley, New York
26. Witkin J.M., Nichols D.E., Terry P., Katz J.L. Behavioral effects of selective dopaminergic compounds in rats discriminating cocaine injections. J. Pharmacol. Exp. Ther. 257:1991;706-713
27. Woolverton W.L. Discriminative stimulus effects of cocaine. Glennon R.A., Jarbe T.U.C., Frankenheim J. Drug discrimination: applications to drug abuse research. NIDA Research Monograph. vol. 116:1991;61-74 U.S. Government Printing Office, Washington (DC)
28. Young R., Glennon R.A. Discriminative stimulus properties of amphetamine and structurally related phenalkylamines. Med. Res. Rev. 6:1986;99-130
29. Young R., Glennon R.A. Cocaine-stimulus generalization to two new designer drugs: methcathinone and 4-methylaminorex. Pharmacol. Biochem. Behav. 45:1993;229-231