Determination of the stereoselectivity of chiral drug transport across Caco-2 cell monolayers

Chirality

Volumn 18, Issue 1, 2006, Pages 64-69

  He, Ying ^a   Zeng, Su ^a  

^a ZHEJIANG UNIVERSITY   (China)

Author keywords

Carrier mediated mechanism; Enantioselectivity; Esmolol; Permeability; Transport

Indexed keywords

2,3,4,6 TETRA O ACETYL BETA DEXTRO GLUCOPYRANOSYL ISOTHIOCYANATE; DRUG; ESMOLOL; GLUCOSE DERIVATIVE; PROPRANOLOL; UNCLASSIFIED DRUG;

ACTIVE TRANSPORT; ARTICLE; CELL STRAIN CACO 2; CHIRALITY; DERIVATIZATION; DIFFUSION; DRUG ABSORPTION; DRUG DETERMINATION; DRUG ELIMINATION; DRUG STRUCTURE; DRUG TRANSPORT; ENANTIOMER; HUMAN; HUMAN CELL; INTESTINE EPITHELIUM; MODEL; MONOLAYER CULTURE; PASSIVE TRANSPORT; PERMEABILITY; PRIORITY JOURNAL; REVERSED PHASE HIGH PERFORMANCE LIQUID CHROMATOGRAPHY; STEREOCHEMISTRY; TRANSCYTOSIS;

ADRENERGIC BETA-ANTAGONISTS; BIOLOGICAL TRANSPORT, ACTIVE; CACO-2 CELLS; CELL MEMBRANE PERMEABILITY; HUMANS; PHARMACEUTICAL PREPARATIONS; PROPANOLAMINES; STEREOISOMERISM;

EID: 29744465624     PISSN: 08990042     EISSN: None     Source Type: Journal    
DOI: 10.1002/chir.20218     Document Type: Article

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