Design of potent inhibitors for Schistosoma japonica glutathione S-transferase

Bioorganic and Medicinal Chemistry

Volumn 14, Issue 2, 2006, Pages 304-318

  Jao, Shu Chuan ^a   Chen, Jessica ^b   Yang, Kelvin ^a   Li, Wen Shan ^a  

^a INSTITUTE OF CHEMISTRY   (Taiwan)

^b NATIONAL CENTRAL UNIVERSITY   (Taiwan)

Author keywords

Drug design; Epiandrosterone; Inhibitors; Molecular modeling; Schistosoma japonica glutathione S transferase

Indexed keywords

(17 CHLORO 3BETA HYDROXYANDROSTA 5,16 DIENE)SUCCINYL GLUTATHIONE; ENZYME INHIBITOR; EPIANDROSTERONE SUCCINYL GLUTATHIONE; GLUTATHIONE DERIVATIVE; GLUTATHIONE TRANSFERASE; MONOMER; PRASTERONE SUCCINYL GLUTATHIONE; SCHISTOSOMA JAPONICA GLUTATHIONE TRANSFERASE; UNCLASSIFIED DRUG;

ARTICLE; COMPARATIVE STUDY; ISOTHERMAL TITRATION CALORIMETRY; NONHUMAN; SCHISTOSOMA JAPONICUM; STOICHIOMETRY;

ANIMALS; BASE SEQUENCE; CLONING, MOLECULAR; DNA PRIMERS; ENZYME INHIBITORS; GLUTATHIONE TRANSFERASE; MAGNETIC RESONANCE SPECTROSCOPY; MOLECULAR STRUCTURE; SCHISTOSOMA; SPECTROMETRY, MASS, FAST ATOM BOMBARDMENT;

SCHISTOSOMA JAPONICUM;

EID: 28844458423     PISSN: 09680896     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmc.2005.07.077     Document Type: Article

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