Synthesis and chemiluminescent high throughput screening for inhibition of acetylcholinesterase activity by imidazo[2,1-b]thiazole derivatives

European Journal of Medicinal Chemistry

Volumn 40, Issue 12, 2005, Pages 1331-1334

  Andreani, Aldo ^a   Granaiola, Massimiliano ^a   Guardigli, Massimo ^a   Leoni, Alberto ^a   Locatelli, Alessandra ^a   Morigi, Rita ^a   Rambaldi, Mirella ^a   Roda, Aldo ^a  

^a UNIVERSITY OF BOLOGNA   (Italy)

Author keywords

Alzheimer's disease; Antiacetylcholinesterase activity; Bisammonium salts; Chemiluminescence; Glaucoma; Imidazo 2,1 b thiazole; Miastenia gravis; Neuromuscular transmission

Indexed keywords

ACETYLCHOLINESTERASE; CHOLINESTERASE INHIBITOR; IMIDAZO[2,1 B]THIAZOLE DERIVATIVE;

ARTICLE; CHEMOLUMINESCENCE; DRUG ACTIVITY; DRUG SCREENING; DRUG SOLUBILITY; DRUG STRUCTURE; DRUG SYNTHESIS; ENZYME INHIBITION; HIGH THROUGHPUT SCREENING;

ACETYLCHOLINESTERASE; CHEMILUMINESCENT MEASUREMENTS; DRUG EVALUATION, PRECLINICAL; IMIDAZOLES; MOLECULAR STRUCTURE; SENSITIVITY AND SPECIFICITY; STRUCTURE-ACTIVITY RELATIONSHIP; THIAZOLES;

EID: 27744439922     PISSN: 02235234     EISSN: 17683254     Source Type: Journal    
DOI: 10.1016/j.ejmech.2005.05.010     Document Type: Article

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