GPCR screening via ERK 1/2: A novel platform for screening G protein-coupled receptors

Journal of Biomolecular Screening

Volumn 10, Issue 7, 2005, Pages 730-737

  Osmond, Ronald I W ^a   Sheehan, Antony ^a   Borowicz, Romana ^a   Barnett, Emma ^a   Harvey, Georgina ^a   Turner, Cheryl ^a   Brown, Andrea ^a   Crouch, Michael F ^a   Dyer, Anthony R ^a  

^a TGR BioSciences   (Australia)

Author keywords

Cell based assay; ERK 1 2; GPCR; HTS; MAPK

Indexed keywords

ATROPINE; CARBACHOL; CHOLECYSTOKININ OCTAPEPTIDE; CYCLIC AMP; G PROTEIN COUPLED RECEPTOR; G PROTEIN COUPLED RECEPTOR AGONIST; G PROTEIN COUPLED RECEPTOR ANTAGONIST; GUANINE NUCLEOTIDE BINDING PROTEIN Q; INOSITOL TRISPHOSPHATE; ITRIGLUMIDE; MITOGEN ACTIVATED PROTEIN KINASE 1; MITOGEN ACTIVATED PROTEIN KINASE 3; RECEPTOR AGONIST; RECEPTOR BLOCKING AGENT; UNCLASSIFIED DRUG;

ANIMAL CELL; ARTICLE; ASSAY; CALCIUM CELL LEVEL; CALCIUM MOBILIZATION; CELL CULTURE; CELL STRAIN 3T3; CELL STRAIN COS7; CULTURE MEDIUM; ENZYME ACTIVATION; ENZYME PHOSPHORYLATION; HIGH THROUGHPUT SCREENING; IC 50; NONHUMAN; PARAMETER; PRIORITY JOURNAL;

ANIMALS; CARBACHOL; CELL LINE; CERCOPITHECUS AETHIOPS; COS CELLS; HUMANS; MITOGEN-ACTIVATED PROTEIN KINASE 1; MITOGEN-ACTIVATED PROTEIN KINASE 3; NEUROTENSIN; RECEPTORS, G-PROTEIN-COUPLED; TRANSFECTION;

ANIMALIA;

EID: 26944466076     PISSN: 10870571     EISSN: 1552454X     Source Type: Journal    
DOI: 10.1177/1087057105277968     Document Type: Article

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