(+)-Cyclazosin, a selective α1B-adrenoceptor antagonist: Functional evaluation in rat and rabbit tissues

European Journal of Pharmacology

Volumn 522, Issue 1-3, 2005, Pages 100-107

  Marucci, Gabriella ^a   Angeli, Piero ^a   Buccioni, Michela ^a   Gulini, Ugo ^a   Melchiorre, Carlo ^b   Sagratini, Gianni ^a   Testa, Rodolfo ^c   Giardinà, Dario ^a  

^a UNIVERSITY OF CAMERINO   (Italy)

^b UNIVERSITY OF BOLOGNA   (Italy)

^c Recordati SpA   (Italy)

Author keywords

1 Adrenoceptor antagonist; 1 Adrenoceptor subtype; 1B Adrenoceptor antagonist; 1B Adrenoceptor; (+) Cyclazosin; Rabbit aorta

Indexed keywords

ADRENERGIC RECEPTOR BLOCKING AGENT; ALPHA 1B ADRENERGIC RECEPTOR; CYCLAZOCINE; ADRENERGIC RECEPTOR ALPHA(1A); ADRENERGIC RECEPTOR ALPHA(1B); ADRENERGIC RECEPTOR ALPHA(1D); ALPHA 1 ADRENERGIC RECEPTOR; ALPHA ADRENERGIC RECEPTOR BLOCKING AGENT; ALPHA ADRENERGIC RECEPTOR STIMULATING AGENT; CHLOROETHYLCLONIDINE; CLONIDINE; CYCLAZOSIN; DRUG DERIVATIVE; METHOXAMINE; NORADRENALIN; QUINAZOLINE DERIVATIVE; QUINOXALINE DERIVATIVE;

ANIMAL TISSUE; ARTICLE; BINDING AFFINITY; DRUG EFFECT; NONHUMAN; PRIORITY JOURNAL; RABBIT; RAT; THORACIC AORTA; ANIMAL; BINDING COMPETITION; CHEMICAL STRUCTURE; CHEMISTRY; COMPARATIVE STUDY; DOSE RESPONSE; DRUG ANTAGONISM; DRUG POTENTIATION; IN VITRO STUDY; MALE; MUSCLE CONTRACTION; PHYSIOLOGY; VAS DEFERENS; VASOCONSTRICTION; WISTAR RAT;

ADRENERGIC ALPHA-AGONISTS; ADRENERGIC ALPHA-ANTAGONISTS; ANIMALS; AORTA, THORACIC; BINDING, COMPETITIVE; CLONIDINE; DOSE-RESPONSE RELATIONSHIP, DRUG; MALE; METHOXAMINE; MOLECULAR STRUCTURE; MUSCLE CONTRACTION; NOREPINEPHRINE; QUINAZOLINES; QUINOXALINES; RABBITS; RATS; RATS, WISTAR; RECEPTORS, ADRENERGIC, ALPHA-1; VAS DEFERENS; VASOCONSTRICTION;

EID: 26844450161     PISSN: 00142999     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.ejphar.2005.08.044     Document Type: Article

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