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Bioorganic and Medicinal Chemistry Letters

Volumn 15, Issue 21, 2005, Pages 4681-4684

Inhibition of Src kinase activity by 7-[(2,4-dichloro-5-methoxyphenyl) amino]-2-heteroaryl-thieno[3,2-b]pyridine-6-carbonitriles

(6) Boschelli, Diane H a Wu, Biqi a Barrios Sosa, Ana Carolina a,b Chen, Joan J a Golas, Jennifer M a Boschelli, Frank a

a WYETH RESEARCH (United States)

b Roche Carolina (United States)

Author keywords

Src; Thieno 3,2 b pyridine 6 carbonitrile

Indexed keywords

BOSUTINIB; PROTEIN TYROSINE KINASE INHIBITOR; PYRIDINE DERIVATIVE; THIENO[3,2 B]PYRIDINE DERIVATIVE; UNCLASSIFIED DRUG;

ANIMAL CELL; ANIMAL EXPERIMENT; ARTICLE; CELL ASSAY; ENZYME ACTIVITY; ENZYME INHIBITION; HUMAN; HUMAN CELL; MOUSE; NONHUMAN; PROTEIN FUNCTION; STRUCTURE ACTIVITY RELATION; SUBSTITUTION REACTION;

ANIMALS; ANTINEOPLASTIC AGENTS; CELL LINE; CELL LINE, TUMOR; HUMANS; INHIBITORY CONCENTRATION 50; KINETICS; MICE; MICE, NUDE; NEOPLASMS, EXPERIMENTAL; NITRILES; PHARMACOKINETICS; PROTEIN KINASE INHIBITORS; SRC-FAMILY KINASES; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 25144509569 PISSN: 0960894X EISSN: None Source Type: Journal
DOI: 10.1016/j.bmcl.2005.07.061 Document Type: Article

Times cited : (21)

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