Peptide inhibitors of G protein-coupled receptor kinases

Biochemical Pharmacology

Volumn 70, Issue 7, 2005, Pages 1001-1008

  Winstel, Rainer ^a   Ihlenfeldt, Hans Georg ^b   Jung, Günther ^b   Krasel, Cornelius ^a,c   Lohse, Martin J ^a  

^a UNIVERSITY OF WÜRZBURG   (Germany)

^b UNIVERSITY OF TÜBINGEN   (Germany)

^c UNIVERSITY OF READING   (United Kingdom)

Author keywords

G protein coupled receptor kinases; Non competitive inhibition; Phosphorylation; Receptor desensitization

Indexed keywords

ACETYLALANYLLYSYLPHENYLALANYLGLUTAMYLARGINYLLEUCYLGLUTAMINYLTHREONYLVALYL THREONYLASPARAGINAMIDATE; ACETYLALANYLLYSYLPHENYLALANYLGLUTAMYLARGINYLLEUCYLGLUTAMINYLTHREONYLVALYL THREONYLASPARAGINYLTYROSYLPHENYLALANINAMIDATE; ACETYLTHREONYLALANYLISOLEUCYLALANYLLYSYLPHENYLALANYLGLUTAMYLARGINYLLEUCYL GLUTAMINYLTHREONYLVALYLTHREONYLASPARAGINYLTYROSYLPHENYLALANYLISOLEUCYLTHREONYL SERINAMIDATE; ADENOSINE TRIPHOSPHATE; ALANYLLYSYLPHENYLALANYLGLUTAMYLARGINYLLEUCYLGLUTAMINYLTHREONYLVALYL THREONYLASPARAGINYLTYROSYLPHENYLALANYLISOLEUCYLTHREONYLSERYLGLUTAMIC ACID; ALANYLLYSYLPHENYLALANYLGLUTAMYLARGINYLLEUCYLGLUTAMINYLTHREONYLVALYL THREONYLASPARAGINYLTYROSYLPHENYLALANYLISOLEUCYLTHREONYLSERYLLYSINE; BETA 2 ADRENERGIC RECEPTOR; CYCLIC AMP DEPENDENT PROTEIN KINASE; G PROTEIN COUPLED RECEPTOR KINASE; G PROTEIN COUPLED RECEPTOR KINASE 2; G PROTEIN COUPLED RECEPTOR KINASE 3; G PROTEIN COUPLED RECEPTOR KINASE 5; GLUTAMYLTHREONYLALANYLISOLEUCYLALANYLLYSYLPHENYLALANYLGLUTAMYLARGINYL LEUCYLGLUTAMINYLTHREONYLVALYLTHREONYLASPARAGINYLTYROSYLPHENYLALANYLISOLEUCYL THREONYLSERYLLYSINE; LYSYLTHREONYLALANYISOLEUCYLALANYLLYSYLPHENYLALANYLGLYCYLARGINYLLEUCYL GLUTAMINYLTHREONYLVALYLTHREONYLASPARAGINYLTYROSYLPHENYLALANYLISOLEUCYLTHREONYL SERYLGLUTAMIC ACID; LYSYLTHREONYLALANYLISOLEUCYLALANYLLYSYLPHENYLALANYLGLUTAMYLARGINYLLEUCYL GLUTAMINYLTHREONYLVALYLTHREONYLASPARAGINE; LYSYLTHREONYLALANYLISOLEUCYLALANYLLYSYLPHENYLALANYLGLUTAMYLARGINYLLEUCYL GLUTAMINYLTHREONYLVALYLTHREONYLASPARAGINYLTYROSYLPHENYLALANYLISOLEUCYLTHREONYL SERYLLYSINE; PHOSPHOTRANSFERASE INHIBITOR; PROTEIN KINASE C; UNCLASSIFIED DRUG;

AMINO TERMINAL SEQUENCE; ARTICLE; CARBOXY TERMINAL SEQUENCE; CONTROLLED STUDY; DRUG POTENCY; DRUG SYNTHESIS; HUMAN; HUMAN CELL; IC 50; PRIORITY JOURNAL;

AMINO ACID SEQUENCE; CYCLIC AMP; ENZYME INHIBITORS; GTP-BINDING PROTEINS; MOLECULAR SEQUENCE DATA; PEPTIDES; PHOSPHORYLATION; RECEPTOR PROTEIN-TYROSINE KINASES;

EID: 24344496159     PISSN: 00062952     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bcp.2005.06.015     Document Type: Article

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