Design, synthesis, and evaluation of original carriers for targeting vascular endothelial growth factor receptor interactions

Pharmaceutical Research

Volumn 22, Issue 8, 2005, Pages 1411-1421

  Gonçalves, Mario ^a,b   Estieu Gionnet, Karine ^b,c   Berthelot, Thomas ^b   Laïn, Georges ^b   Bayle, Mireille ^b   Canron, Xavier ^b   Betz, Natacha ^a   Bikfalvi, Andreas ^c   Déléris, Gérard ^b  

^a CEA SACLAY   (France)

^b UNIVERSITÉ DE BORDEAUX   (France)

^c INSERM   (France)

Author keywords

Angiogenesis; Chemotherapy; Cyclopeptide modification; Imaging; Receptors targeting; Solid phase peptide synthesis; Vascular endothelial growth factor

Indexed keywords

CYCLOPEPTIDE; DRUG CARRIER; FLUORESCENT DYE; IODINE 125; NANOPARTICLE; VASCULOTROPIN INHIBITOR; VASCULOTROPIN RECEPTOR;

ANGIOGENESIS; ANIMAL CELL; ARTICLE; CHEMICAL MODIFICATION; CHINESE HAMSTER; CONJUGATE; CONTROLLED STUDY; COW; DIAGNOSTIC IMAGING; DRUG ACCUMULATION; DRUG ACTIVITY; DRUG COMPETITION; DRUG DELIVERY SYSTEM; DRUG DESIGN; DRUG DETERMINATION; DRUG EFFECT; DRUG INHIBITION; DRUG RECEPTOR BINDING; DRUG SCREENING; DRUG SELECTIVITY; DRUG SYNTHESIS; DRUG TARGETING; GENETIC LINKAGE; HYDROPHILICITY; NONHUMAN; PRIORITY JOURNAL;

AMINO ACID SEQUENCE; ANGIOGENESIS INHIBITORS; ANIMALS; CHO CELLS; CRICETINAE; DRUG CARRIERS; DRUG DESIGN; ENDOTHELIAL GROWTH FACTORS; INDICATORS AND REAGENTS; MAGNETIC RESONANCE SPECTROSCOPY; MOLECULAR SEQUENCE DATA; PEPTIDES, CYCLIC; PROTEIN BINDING; RECEPTORS, VASCULAR ENDOTHELIAL GROWTH FACTOR; SPECTROMETRY, MASS, MATRIX-ASSISTED LASER DESORPTION-IONIZATION;

EID: 23844556270     PISSN: 07248741     EISSN: None     Source Type: Journal    
DOI: 10.1007/s11095-005-5265-9     Document Type: Article

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