Inhibition of 7,8-diaminopelargonic acid aminotransferase by amiclenomycin and analogues

Biochemical Society Transactions

Volumn 33, Issue 4, 2005, Pages 802-805

  Mann, S ^a   Marquet, A ^a   Ploux, O ^a  

^a SORBONNE UNIVERSITÉ   (France)

Author keywords

7,8 diaminopelargonic acid aminotransferase; Amiclenomycin; Biotin biosynthesis; Drug target; Mycobacterium tuberculosis; Pyridoxal 5 phosphate

Indexed keywords

7,8 DIAMINOPELARGONIC ACID AMINOTRANSFERASE; AMICLENOMYCIN; AMINO ACID; AMINOTRANSFERASE; PYRIDOXAL 5 PHOSPHATE; UNCLASSIFIED DRUG;

CONFERENCE PAPER; DRUG POTENTIATION; ENZYME ACTIVE SITE; ESCHERICHIA COLI; HUMAN; MYCOBACTERIUM TUBERCULOSIS; NONHUMAN; PRIORITY JOURNAL; PROTEIN EXPRESSION; PROTON NUCLEAR MAGNETIC RESONANCE; STEREOISOMERISM; TUBERCULOSIS; ULTRAVIOLET SPECTROSCOPY; X RAY CRYSTALLOGRAPHY;

AMINOBUTYRIC ACIDS; ANTITUBERCULAR AGENTS; BACTERIAL PROTEINS; ENZYME INHIBITORS; KINETICS; MYCOBACTERIUM TUBERCULOSIS; TRANSAMINASES;

ESCHERICHIA COLI; MYCOBACTERIUM TUBERCULOSIS;

EID: 23844435643     PISSN: 03005127     EISSN: None     Source Type: Journal    
DOI: 10.1042/BST0330802     Document Type: Conference Paper

References (20)

1. Okami, Y., Kitahara, T., Hamada, M., Naganawa, H. and Kondo, S. (1974) J. Antibiot. (Tokyo) 27, 656-664
2. Kitahara, T., Hotta, K., Yoshida, M. and Okami, Y. (1975) J. Antibiot. (Tokyo) 28, 215-221
3. Hotta, K., Kitahara, T. and Okami, Y. (1975) J. Antibiot. (Tokyo) 28, 222-228
4. Kern, A., Kabatek, U., Jung, G., Werner, R.G., Poetsh, M. and Zahner, H. (1985) Liebigs Ann. Chem. 5, 877-892
5. Poetsch, M., Zahner, H., Werner, R.G., Kern, A. and Jung, G. (1985) J. Antibiot. (Tokyo) 38, 312-320
6. Mann, S., Carillon, S., Breyne, O. and Marquet, A. (2002) Chem. Eur. J. 8, 439-450
7. Mann, S., Carillon, S., Breyne, O., Duhayon, C., Hamon, L. and Marquet, A. (2002) Eur. J. Org. Chem. 736-744
8. Sandmark, J., Mann, S., Marquet, A. and Schneider, G. (2002) J. Biol. Chem. 277, 43352-43358
9. Mann, S., Lesage, D., Tabet, J.C. and Marquet, A. (2003) Tetrahedron 59, 5209-5214
10. Mann, S., Florentin, D., Lesage, D., Drujon, D., Ploux, O. and Marquet, A. (2003) Helv. Chim. Acta 86, 3836-3850
11. Keer, J., Smeulders, M.J., Gray, K.M. and Williams, H.D. (2000) Microbiology 146, 2209-2217
12. Stoner, G.L. and Eisenberg, M.A. (1975) J. Biol. Chem. 250, 4029-4036
13. Stoner, G.L. and Eisenberg, M.A. (1975) J. Biol. Chem. 250, 4037-4043
14. Eliot, A.C., Sandmark, J., Schneider, G. and Kirsch, J.F. (2002) Biochemistry 41, 12582-12589
15. Kack, H., Gibson, K.J., Gatenby, A.A., Schnieder, G. and Lindqvist, Y. (1998) Acta Crystallogr. D Biol. Crystallogr. 54, 1397-1398
16. Kack, H., Sandark, J., Gibson, K.J., Schneider, G. and Lindqvist, Y. (1999) J. Mol. Biol. 291, 857-876
17. Rando, R.R. (1977) Biochemistry 16, 4605-4610
18. Olson, G.T., Fu, M., Lau, S., Rinehart, K.L. and Silverman, R.B. (1998) J. Am. Chem. Soc. 120, 2256-2267
19. Peisach, D., Chipman, D.M., Van Ophem, P.W., Manning, J.M. and Ringe, D. (1998) J. Am. Chem. Soc. 120, 2268-2274
20. Fenn, T.D., Stamper, G.F., Morollo, A.A. and Ringe, D. (2003) Biochemistry 42, 5775-5783