Synthesis, anorexigenic activity and QSAR of substituted aryloxypropanolamines

Medicinal Chemistry Research

Volumn 13, Issue 8-9, 2004, Pages 631-642

  Srivastava, Shipra ^a   Bhandari, Kalpana ^a   Shankar, Girija ^a   Singh, H K ^a   Saxena, Anil K ^a  

^a CENTRAL DRUG RESEARCH INSTITUTE   (India)

Author keywords

[No Author keywords available]

Indexed keywords

1 (2'' METHOXYARYLOXY) 3 [N METHYL N (3' ARYL 3' (4''' ALPHA,ALPHA,ALPHA TRIFLUOROMETHYLARYLOXY)PROPYL)AMINO]PROPAN 2 OL; 1 (2'' METHYLARYLOXY) 3 [N METHYL N (3' ARYL 3' (4''' ALPHA,ALPHA,ALPHA TRIFLUOROMETHYLARYLOXY)PROPYL)AMINO]PROPAN 2 OL; 1 (2'' NAPHTHYLOXY) 3 [N METHYL N (3' ARYL 3' (4''' ALPHA,ALPHA,ALPHA TRIFLUOROMETHYLARYLOXY)PROPYL)AMINO]PROPAN 2 OL; 1 (3'' ALPHA,ALPHA,ALPHA TRIFLUOROMETHYLARYLOXY) 3 [N METHYL N (3' ARYL 3' (4''' ALPHA,ALPHA,ALPHA TRIFLUOROMETHYLARYLOXY)PROPYL)AMINO]PROPAN 2 OL; 1 (4'' ACETAMIDOARYLOXY) 3 [N METHYL N (3' ARYL 3' (4''' ALPHA,ALPHA,ALPHA TRIFLUOROMETHYLARYLOXY)PROPYL)AMINO]PROPAN 2 OL; 1 (4'' ACETYLARYLOXY) 3 [N METHYL N (3' ARYL 3' (4''' ALPHA,ALPHA,ALPHA TRIFLUOROMETHYLARYLOXY)PROPYL)AMINO]PROPAN 2 OL; 1 (4'' ALPHA,ALPHA,ALPHA TRIFLUOROMETHYLARYLOXY) 3 [N METHYL N (3' ARYL 3' (4''' ALPHA,ALPHA,ALPHA TRIFLUOROMETHYLARYLOXY)PROPYL)AMINO]PROPAN 2 OL; 1 (4'' BROMOARYLOXY) 3 [N METHYL N (3' ARYL 3' (4''' ALPHA,ALPHA,ALPHA TRIFLUOROMETHYLARYLOXY)PROPYL)AMINO]PROPAN 2 OL; 1 (4'' CHLOROARYLOXY) 3 [N METHYL N (3' ARYL 3' (4''' ALPHA,ALPHA,ALPHA TRIFLUOROMETHYLARYLOXY)PROPYL)AMINO]PROPAN 2 OL; 1 (4'' CYANOARYLOXY) 3 [N METHYL N (3' ARYL 3' (4''' ALPHA,ALPHA,ALPHA TRIFLUOROMETHYLARYLOXY)PROPYL)AMINO]PROPAN 2 OL; 1 (4'' FORMYLARYLOXY) 3 [N METHYL N (3' ARYL 3' (4''' ALPHA,ALPHA,ALPHA TRIFLUOROMETHYLARYLOXY)PROPYL)AMINO]PROPAN 2 OL; 1 (4'' METHOXYARYLOXY) 3 [N METHYL N (3' ARYL 3' (4''' ALPHA,ALPHA,ALPHA TRIFLUOROMETHYLARYLOXY)PROPYL)AMINO]PROPAN 2 OL; 1 (4'' N ETHYLAMINOARYLOXY) 3 [N METHYL N (3' ARYL 3' (4''' ALPHA,ALPHA,ALPHA TRIFLUOROMETHYLARYLOXY)PROPYL)AMINO]PROPAN 2 OL; 1 (4'' PROPIONYLARYLOXY) 3 [N METHYL N (3' ARYL 3' (4''' ALPHA,ALPHA,ALPHA TRIFLUOROMETHYLARYLOXY)PROPYL)AMINO]PROPAN 2 OL; 1 ARYLOXY 3 [N METHYL N (3' ARYL 3' (4''' ALPHA,ALPHA,ALPHA TRIFLUOROMETHYLARYLOXY)PROPYL)AMINO]PROPAN 2 OL; ANOREXIGENIC AGENT; ARYLOXYPROPANOLAMINE; UNCLASSIFIED DRUG;

CONFERENCE PAPER; DEBENZYLATION; DRUG ACTIVITY; DRUG EFFECT; DRUG SCREENING; DRUG STRUCTURE; DRUG SYNTHESIS; HYDROPHOBICITY; MANNICH REACTION; PHYSICAL CHEMISTRY; QUANTITATIVE STRUCTURE ACTIVITY RELATION; SUBSTITUTION REACTION;

EID: 22644445635     PISSN: 10542523     EISSN: None     Source Type: Journal    
DOI: 10.1007/s00044-004-0107-6     Document Type: Conference Paper

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