Evidence against adenosine analogues being agonists at the growth hormone secretagogue receptor

Biochemical Pharmacology

Volumn 70, Issue 4, 2005, Pages 598-605

  Johansson, Stina ^a   Fredholm, Bertil B ^a   Hjort, Charlotta ^b   Morein, Torbjörn ^b   Kull, Björn ^b   Hu, Ping Sheng ^b  

^a KAROLINSKA INSTITUTE   (Sweden)

^b BIOVITRUM AB   (Sweden)

Author keywords

Adenosine A2B receptor; CHO cells; Ghrelin; GHSR1a; HEK 293 cells

Indexed keywords

2 CHLORADENOSINE; 8 CYCLOPENTYL 1,3 DIPROPYLXANTHINE; ADENOSINE; ADENOSINE 5' (N ETHYLCARBOXAMIDE); ADENOSINE A2B RECEPTOR; ADENOSINE DERIVATIVE; GHRELIN; GROWTH HORMONE SECRETAGOGUE RECEPTOR 1A AGONIST; HORMONE RECEPTOR STIMULATING AGENT; IBUTAMOREN; SUBSTANCE P [1 DEXTRO ARGININE 5 DEXTRO PHENYLALANINE 7,9 DEXTRO TRYPTOPHAN 11 LEUCINE]; UNCLASSIFIED DRUG;

ANIMAL CELL; ARTICLE; BINDING AFFINITY; CALCIUM CELL LEVEL; CELL MEMBRANE; CONTROLLED STUDY; DRUG EFFECT; DRUG POTENTIATION; DRUG RECEPTOR BINDING; GENETIC TRANSFECTION; HUMAN; HUMAN CELL; NONHUMAN; PHARMACODYNAMICS; PRIORITY JOURNAL;

ADENOSINE; ANIMALS; CALCIUM; CELL LINE; CHO CELLS; CRICETINAE; CYCLIC AMP; GLUTATHIONE; HUMANS; PEPTIDE HORMONES; RADIOLIGAND ASSAY; RECEPTORS, G-PROTEIN-COUPLED; SIGNAL TRANSDUCTION;

EID: 22144488132     PISSN: 00062952     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bcp.2005.05.023     Document Type: Article

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