Studies on the interactions between drugs and estrogen. III. Inhibitory effects of 29 drugs reported to induce gynecomastia on the glucuronidation of estradiol

Biological and Pharmaceutical Bulletin

Volumn 27, Issue 11, 2004, Pages 1844-1849

  Satoh, Takashi ^a   Tomikawa, Yuki ^b,d   Takanashi, Kaori ^b   Itoh, Shinji ^b   Itoh, Shungo ^c   Yoshizawa, Itsuo ^b  

^a Yakuhan Pharmaceutical Co Ltd   (Japan)

^b HOKKAIDO INSTITUTE OF TECHNOLOGY   (Japan)

^c Japan Seamen Relief Association Otaru Hospital   (Japan)

^d Sapporo Chuo Hospital   (Japan)

Author keywords

Drug induced gynecomastia; Estradiol; Interaction; UDP glucuronosyltransferase

Indexed keywords

CHLORMADINONE; DOMPERIDONE; ESTRADIOL; ESTROGEN; IPRIFLAVONE; KETOCONAZOLE; MANIDIPINE; NICARDIPINE; NIFEDIPINE; NISOLDIPINE; NITRENDIPINE; TACROLIMUS; CYTOCHROME P450; DRUG; GLUCURONIDE;

ARTICLE; CHEMICAL INTERACTION; CIRCULATION; CONCENTRATION (PARAMETERS); DRUG OVERDOSE; GYNECOMASTIA; HYDROXYLATION; METABOLISM; MICROSOME; CHEMICALLY INDUCED DISORDER; COMPARATIVE STUDY; DRUG INTERACTION; ENZYMOLOGY; HIGH PERFORMANCE LIQUID CHROMATOGRAPHY; HUMAN; IN VITRO STUDY; LIVER MICROSOME;

CHROMATOGRAPHY, HIGH PRESSURE LIQUID; CYTOCHROME P-450 ENZYME SYSTEM; DRUG INTERACTIONS; ESTRADIOL; GLUCURONIDES; GYNECOMASTIA; HUMANS; HYDROXYLATION; MICROSOMES, LIVER; PHARMACEUTICAL PREPARATIONS;

EID: 22044452396     PISSN: 09186158     EISSN: 13475215     Source Type: Journal    
DOI: 10.1248/bpb.27.1844     Document Type: Article

References (24)

1. Satoh T., Fujita K., Munakata H., Itoh Shi., Nakamura K., Kamataki T., Itoh Shu., Yoshizawa I., Anal. Biochem., 286, 179-186 (2000).
2. Satoh T., Munakata H., Fujita K., Itoh Shi., Itoh Shu., Kamataki T., Yoshizawa I., Biol. Pharm. Bull., 26, 695-700 (2003).
3. Satoh T., Itoh Shi., Seki T., Itoh Shu., Nomura N., Yoshizawa I., J. Steroid Biochem. Molec. Biol., 82, 209-216 (2002).
4. Mackenzie P. I., Owens I. S., Burchell B., Bock K. W., Bairoch A., Bélanger A., Fournel-Gigleux S., Green M., Hum D. W., Iyanagi T., Lancet D., Louisot P., Magdaloe J., Chowdhury J. R., Ritter J. K., Schachter H., Tephly T. R., Tipton K. F., Nebert D. W., Pharmacogenetics, 7, 255-269 (1997).
5. Ritter J. K., Chem.-Biol. Inter., 129, 171-193 (2000).
6. King C. D., Green M. D., Rios G. R., Coffman B. L., Owens I. S., Bishop W. P., Tephly T. R., Arch. Biochem. Biophys., 332, 92-100 (1996).
7. Ebner T., Remmel R. P., Burchell B., Molec. Pharmacol., 43, 649-654 (1993).
8. Jin C., Miners J. O., Lillywhite K. J., Mackenzie P. I., J. Pharmacol. Exp. Ther., 264, 475-479 (1993).
9. Coffman B. L., Rios G. R., King C. D., Tephly T. R., Drug Metab. Dispos., 25, 1-4 (1997).
10. Coffman B. L., King C. D., Rios G. R., Tephly T. R., Drug Metab. Dispos., 26, 73-77 (1998).
11. Kirdani R. Y., Steroids, 6, 845-853 (1965).
12. Czernik P. J., Little J. M., Barone G. W., Raufman J.-P., Radminska-Pandya A., Drug Metab. Dispos., 28, 1210-1216 (2000).
13. Staczyk F. Z., Miyakawa I., Goebelsmann U., Am. J. Obstet. Gynecol., 137, 443-450 (1980).
14. Morikawa A., Goto Y., Suzuki H., Hirohashi T., Sugiyama Y., Pharm. Res., 17, 546-552 (2000).
15. Loe D. W., Almquist K. C., Cole S. P. C., Deeley R. G., J. Biol. Chem., 271, 9683-9689 (1996).
16. Adlercreutz H., Martin F., J. Steroid Biochem., 13, 231-244 (1980).
17. Vree T. B., Timmer C. J., J. Pharm. Pharmacol., 50, 857-864 (1998).
18. Strassburg C. P., Barut A., Obermayer-Straub P., Li Q., Nguyen N., Tukey R. H., Manns M. P., J. Hepatol., 34, 865-872 (2001).
19. Hardman J. G., Limbird L. E., Molinoff P. B., Ruddom R. W. (eds.), "Goodman & Gilman's The Pharmacological Basis of Therapeutics," 9th ed., McGraw-Hill, New York, 1995, pp. 1370-1372.
20. Sampol E., Lacarelle B., Rajaonarison J. F., Catalin J., Durand A., Br. J. Clin. Pharmacol., 40, 83-86 (1995).
21. Grosso D. S., Boyden T. W., Pamenter R. W., Johnson D. G., Stevens D. A., Galgiani J. N., Antimicrob. Agents Chemother., 23, 207-212 (1983).
22. Williams J. A., Ring B. J., Cantrell V. E., Campanale K., Jones D. R., Hall S. D., Wrighton S. A., Drug Metab. Dispos., 30, 1266-1273 (2002).
23. Jakob F., Siggelkow H., Homann D., Köhrle J., Adamski J., Schütze N., J. Steroid Biochem. Molec. Biol., 61, 167-174 (1997).
24. Akaza H., Usami M., Kotake T., Koiso K., Aso Y., Jpn. J. Clin. Oncol., 23, 178-185 (1993).