ANIMAL TISSUE;
ARTICLE;
CONTROLLED STUDY;
DRUG ACTIVITY;
DRUG EFFICACY;
DRUG POTENCY;
DRUG SYNTHESIS;
MALE;
NONHUMAN;
RAT;
VASCULAR RING;
VASODILATATION;
5-(4'-Substituted-2'-nitroanilino)-1,2,3-triazoles as new potential potassium channel activators. I
Biagi G., Calderone V., Giorgi I., Livi O., Scartoni V., Baragatti B., Martinotti E. 5-(4'-Substituted-2'-nitroanilino)-1, 2, 3-triazoles as new potential potassium channel activators. I. Eur. J. Med. Chem. 35:2000;715-720
Triazolyl-benzimidazolones and triazolyl-benzotriazoles: New potential potassium channel activators. II
Baragatti B., Biagi G., Calderone V., Giorgi I., Livi O., Martinotti E., Scartoni V. Triazolyl-benzimidazolones and triazolyl-benzotriazoles: new potential potassium channel activators. II. Eur. J. Med. Chem. 35:2000;949-955
Some structural changes on triazolyl-benzotriazoles and triazolyl-benzimidazolones as potential potassium channel activators. III
Biagi G., Calderone V., Giorgi I., Livi O., Scartoni V., Baragatti B., Martinotti E. Some structural changes on triazolyl-benzotriazoles and triazolyl-benzimidazolones as potential potassium channel activators. III. Farmaco. 56:2001;841-849
The synthesis and structure-activity relationships of 1,3-dyaril 1,2,4-(4H)-triazol-5-ones: A new class of calcium-dependent, large conductance, potassium (maxi-K) channel opener targeted for urge urinary incontinence
Hewawasam P., Erway M., Thalody G., Weiner H., Boissard C.G., Gribkoff V.K., Meanwell N.A., Lodge N., Starrett J.E. Jr. The synthesis and structure-activity relationships of 1, 3-dyaril 1, 2, 4-(4H)-triazol-5-ones: a new class of calcium-dependent, large conductance, potassium (maxi-K) channel opener targeted for urge urinary incontinence. Bioorg. Med. Chem. Lett. 12:2002;1117-1120
Gribkoff V.K., Meanwell N.A., Martin S.W., Hewawasam P., Romine J.L., Starrett J.E. Jr. Diphenylheterocycles as potassium channel modulators. 1998;. International Patent Application, WO 9804135
Recent developments in the biology and medicinal chemistry of potassium channel modulators: Update from a decade of progress
Coghlan M.J., Carroll W.A., Gopalakrishnan M. Recent developments in the biology and medicinal chemistry of potassium channel modulators: update from a decade of progress. J. Med. Chem. 44:2001;1627-1653
Pyrolysis of aryl azides. VII. Interpretation of Hammett correlations of rates of pyrolysis of substituted 2-nitroazidobenzenes
Dyall L.K. Pyrolysis of aryl azides. VII. Interpretation of Hammett correlations of rates of pyrolysis of substituted 2-nitroazidobenzenes. Aust. J. Chem. 39:1986;89-101
Synthesis of new 1,2,3-triazolo[1,2-a] benzotriazole derivatives or substituted 2,3-benzo-1,3a,6,6a-tetraazapentalenes. II
Biagi G., Giorgi I., Livi O., Manera C., Scartoni V., Barili P.L. Synthesis of new 1, 2, 3-triazolo[1, 2-a] benzotriazole derivatives or substituted 2, 3-benzo-1, 3a, 6, 6a-tetraazapentalenes. II. J. Heterocyclic Chem. 34:1997;845-851
Synthesis of N-(2-aminoaryl)-benzamide oximes and their heteroaromatization reactions
Risitano F., Grassi G., Foti F., Caruso F. Synthesis of N-(2-aminoaryl)-benzamide oximes and their heteroaromatization reactions. J. Chem. Res., Synopses. 2:1983;52
Hypervalent iodine-induced nucleophilic substitution of p-substituted phenol ethers. Generation of cation radicals as reactive intermediates
Kita Y., Tohma H., Hatanaka K., Takada T., Fujjita S., Mitoh S., Sakurai H., Oka S. Hypervalent iodine-induced nucleophilic substitution of p-substituted phenol ethers. Generation of cation radicals as reactive intermediates. J. Am. Chem. Soc. 116:1994;3684-3691
Proton magnetic resonance study of the spectra of substituted phenylazides
Treushnikov V.M., Gusarskaya N.L., Oleinik A.V., Ya. Proshko V. Proton magnetic resonance study of the spectra of substituted phenylazides. Zhurnal Fizicheskoi Khimii. 51:1997;380-384
Synthesis and hypoglycemic activity of phenacyltriphenylphosphoranes and phosphonium salts
Blank B., DiTullio N.W., Deviney L., Roberts J.T., Saunders H.L. Synthesis and hypoglycemic activity of phenacyltriphenylphosphoranes and phosphonium salts. J. Med. Chem. 18:1975;952-954
Synthesis and biological activity of novel substituted benzanilides as potassium channel activators
(in press)
G. Biagi, I. Giorgi, O. Livi, A. Nardi, V. Calderone, A. Martelli, E. Martinotti, O.L.R. Salerni, Synthesis and biological activity of novel substituted benzanilides as potassium channel activators. V. Eur. J. Med. Chem. (in press)
Sorrento 18-22 Settembre. XVI Convegno Nazionale della Divisione di Chimica Farmaceutica, abstract
G. Biagi, V. Calderone, I. Giorgi, O. Livi, E. Martinotti, A. Nardi, V. Scartoni, Derivati 1, 2, 3-triazolici a potenziale attività sui canali del potassio, Sorrento 18-22 Settembre 2002. XVI Convegno Nazionale della Divisione di Chimica Farmaceutica, abstract p.120.
Hewawasam P., Ding M., Starrett J.E. Jr. Preparation of N-hydroxybenzyl-1, 3, 4-oxadiazolones and analogs as calcium-activated potassium (BK) channel openers. 1999;. International Patent Application, WO 9938510
Hewawasam P., Chen X., Ding M., Starrett J.E. Jr. Preparation of N-hydroxybenzyl-1, 3, 4-oxadiazolones and analogs as calcium-activated potassium (BK) channel openers. 1999;. International Patent Application, WO 9938854
