Use of novel, non-imidazole inverse agonist radioligands to define histamine H3 receptor pharmacology

Inflammation Research

Volumn 54, Issue SUPPL. 1, 2005, Pages

  Esbenshade, T A ^a   Yao, B B ^a   Witte, D G ^a   Carr, T L ^a   Sharma, R ^a   Baranowski, J L ^a   Krueger, K M ^a   Miller, T R ^a   Surber, B W ^a   Faghih, R ^a   Hancock, A A ^a  

^a ABBOTT LABORATORIES   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

4 [4 [3 (2,5 DIMETHYLPYRROLIDINYL)PROPOXY]PHENYL]PHENYLMORPHOLIN 4 YLKETONE; A 317920; A 349821; FURAN 2 CARBOXYLIC ACID[2 [4 [3 (4 CYCLOPROPANECARBONYLPHENOXY)PROPYL] PIPERAZIN 1 YL] 1 METHYL 2 OXOETHYL]AMIDE; HISTAMINE H3 RECEPTOR; HISTAMINE H3 RECEPTOR AGONIST; UNCLASSIFIED DRUG;

ANIMAL TISSUE; CONFERENCE PAPER; CONTROLLED STUDY; DRUG POTENCY; DRUG RECEPTOR BINDING; DRUG SYNTHESIS; HUMAN; HUMAN TISSUE; ISOTOPE LABELING; NONHUMAN; RAT; RECEPTOR AFFINITY;

ANIMALS; BIPHENYL COMPOUNDS; CELL LINE; HISTAMINE AGONISTS; HUMANS; IMIDAZOLES; MOLECULAR STRUCTURE; PIPERAZINES; RADIOLIGAND ASSAY; RATS; RECEPTORS, HISTAMINE H3;

EID: 21144439214     PISSN: 10233830     EISSN: None     Source Type: Journal    
DOI: 10.1007/s00011-004-0421-y     Document Type: Conference Paper

References (5)

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