QSAR analysis of thiazole benzenesulfonamide substituted 3-pyridylethanolamines as β3-adrenergic receptor agonist

Bioorganic and Medicinal Chemistry Letters

Volumn 15, Issue 12, 2005, Pages 3167-3173

  Hanumantharao, P ^a   Sambasivarao, S V ^a   Soni, Love K ^a   Gupta, A K ^a   Kaskhedikar, S G ^a  

^a CADD Laboratory   (India)

Author keywords

3 adrenergic receptor agonist; Anti hyperlipidemic agents; QSAR (quantitative structure activity relationship); Substituted benzene sulfonamide 3 pyridylethanolamines

Indexed keywords

BENZENESULFONAMIDE DERIVATIVE; BETA 3 ADRENERGIC RECEPTOR STIMULATING AGENT; ETHANOLAMINE DERIVATIVE;

ANIMAL CELL; ARTICLE; CORRELATION COEFFICIENT; ELECTRIC POTENTIAL; LIPOPHILICITY; NONHUMAN; PHYSICAL CHEMISTRY; QUANTITATIVE STRUCTURE ACTIVITY RELATION; STATISTICAL SIGNIFICANCE; SUBSTITUTION REACTION;

ADRENERGIC BETA-AGONISTS; ETHANOLAMINES; HUMANS; MODELS, MOLECULAR; MOLECULAR STRUCTURE; QUANTITATIVE STRUCTURE-ACTIVITY RELATIONSHIP; RECEPTORS, ADRENERGIC, BETA-3; SULFONAMIDES; THIAZOLES;

EID: 19944375454     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2005.03.119     Document Type: Article

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