SCOPUS 정보 검색 플랫폼

Bioorganic and Medicinal Chemistry Letters

Volumn 15, Issue 11, 2005, Pages 2758-2760

Synthesis and biological studies of yohimbine derivatives on human α2C-adrenergic receptors

(6) Mustafa, Suni M a Bavadekar, Supriya A b Ma, Guoyi b Moore, Bob M a Feller, Dennis R b Miller, Duane D a

a UNIVERSITY OF TENNESSEE HEALTH SCIENCE CENTER (United States)

b UNIVERSITY OF MISSISSIPPI (United States)

Author keywords

[No Author keywords available]

Indexed keywords

ALPHA 2C ADRENERGIC RECEPTOR; YOHIMBINE DERIVATIVE;

ANIMAL CELL; ARTICLE; BINDING AFFINITY; BIOLOGICAL ACTIVITY; CHO CELL; CONTROLLED STUDY; DRUG RECEPTOR BINDING; DRUG SYNTHESIS; NONHUMAN; PHARMACOPHORE;

ANIMALS; CHO CELLS; CRICETINAE; HUMANS; MICE; PROTEIN BINDING; RECEPTORS, ADRENERGIC, ALPHA-2; YOHIMBINE;

CRICETINAE; CRICETULUS GRISEUS;

EID: 19544384921 PISSN: 0960894X EISSN: None Source Type: Journal
DOI: 10.1016/j.bmcl.2005.03.116 Document Type: Article

Times cited : (8)

References (30)

1
- 0018817101
- B.B. Hoffman, and R.J. Lefkowitz Annu. Rev. Pharmacol. Toxicol 20 1980 581
- (1980) Annu. Rev. Pharmacol. Toxicol , vol.20 , pp. 581
- Hoffman, B.B.¹ Lefkowitz, R.J.²

2
- 0025919746
- M.A. Gerhardt, and R.R. Neubig Mol. Pharmacol. 40 1991 707
- (1991) Mol. Pharmacol. , vol.40 , pp. 707
- Gerhardt, M.A.¹ Neubig, R.R.²

3
- 0026741825
- M.G. Eason, H. Kurose, B.D. Holt, J.R. Raymond, and S.B. Liggett J. Biol. Chem. 267 1992 15795
- (1992) J. Biol. Chem. , vol.267 , pp. 15795
- Eason, M.G.¹ Kurose, H.² Holt, B.D.³ Raymond, J.R.⁴ Liggett, S.B.⁵

4
- 0026519531
- D.B. Bylund FASEB J. 6 1992 832
- (1992) FASEB J. , vol.6 , pp. 832
- Bylund, D.B.¹

5
- 0028183015
- D.B. Bylund, D.C. Eikenberg, J.P. Hieble, S.Z. Langer, R.J. Lefkowitz, K.P. Minneman, P.B. Molinoff, R.R. Ruffolo Jr., and U. Trendelenburg Pharmacol. Rev. 46 1994 121
- (1994) Pharmacol. Rev. , vol.46 , pp. 121
- Bylund, D.B.¹ Eikenberg, D.C.² Hieble, J.P.³ Langer, S.Z.⁴ Lefkowitz, R.J.⁵ Minneman, K.P.⁶ Molinoff, P.B.⁷ Ruffolo Jr., R.R.⁸ Trendelenburg, U.⁹

6
- 0029134812
- J.P. Hieble, W.E. Bondinell, and R.R. Ruffolo Jr. J. Med. Chem. 38 1995 3415
- (1995) J. Med. Chem. , vol.38 , pp. 3415
- Hieble, J.P.¹ Bondinell, W.E.² Ruffolo Jr., R.R.³

7
- 0029824446
- J.P. Hieble, and R.R. Ruffolo Jr. Prog. Drug Res. 47 1996 81
- (1996) Prog. Drug Res. , vol.47 , pp. 81
- Hieble, J.P.¹ Ruffolo Jr., R.R.²

8
- 0029022455
- J.P. Hieble, R.R. Ruffolo Jr., A.C. Sulpizio, D.P. Naselsky, T.M. Conway, C. Ellis, A.M. Swift, S. Ganguly, and D.J. Bergsma Pharmacol. Commun. 6 1995 91
- (1995) Pharmacol. Commun. , vol.6 , pp. 91
- Hieble, J.P.¹ Ruffolo Jr., R.R.² Sulpizio, A.C.³ Naselsky, D.P.⁴ Conway, T.M.⁵ Ellis, C.⁶ Swift, A.M.⁷ Ganguly, S.⁸ Bergsma, D.J.⁹

9
- 0029134812
- R.R. Ruffolo Jr., W.E. Bondinell, and J.P. Hieble J. Med. Chem. 38 1995 3415
- (1995) J. Med. Chem. , vol.38 , pp. 3415
- Ruffolo Jr., R.R.¹ Bondinell, W.E.² Hieble, J.P.³

10
- 0022857780
- R.D. Clark, A.D. Michel, and R.L. Whiting Prog. Med. Chem. 23 1986 1
- (1986) Prog. Med. Chem. , vol.23 , pp. 1
- Clark, R.D.¹ Michel, A.D.² Whiting, R.L.³

11
- 0024422263
- P. Yound, J. Berge, H. Chapman, and M.A. Cawthorne Eur. J. Pharmacol. 168 1989 381
- (1989) Eur. J. Pharmacol. , vol.168 , pp. 381
- Yound, P.¹ Berge, J.² Chapman, H.³ Cawthorne, M.A.⁴

12
- 0023887607
- K. Okumura, K. Koike, H. Asai, and I. Takayanagi Gen. Pharmacol. 19 1988 463
- (1988) Gen. Pharmacol. , vol.19 , pp. 463
- Okumura, K.¹ Koike, K.² Asai, H.³ Takayanagi, I.⁴

13
- 0029591282
- L.J. Beeley, J.M. Berge, H. Chapman, J.P. Hieble, J. Kelly, D.P. Naselsky, C.M. Rockell, and P.W. Young Bioorg. Med. Chem. 3 1995 1693
- (1995) Bioorg. Med. Chem. , vol.3 , pp. 1693
- Beeley, L.J.¹ Berge, J.M.² Chapman, H.³ Hieble, J.P.⁴ Kelly, J.⁵ Naselsky, D.P.⁶ Rockell, C.M.⁷ Young, P.W.⁸

14
- 0025019649
- A.D. Michel, D.N. Loury, and R.L. Whiting Br. J. Pharmacol. 99 1990 560
- (1990) Br. J. Pharmacol. , vol.99 , pp. 560
- Michel, A.D.¹ Loury, D.N.² Whiting, R.L.³

15
- 0025718614
- H.S. Blaxall, T.J. Murphy, J.C. Baker, C. Ray, and D.B. Bylund J. Pharmacol. Exp. Ther. 259 1991 323
- (1991) J. Pharmacol. Exp. Ther. , vol.259 , pp. 323
- Blaxall, H.S.¹ Murphy, T.J.² Baker, J.C.³ Ray, C.⁴ Bylund, D.B.⁵

16
- 0027081142
- D.B. Bylund, H.S. Blaxall, L.J. Iverson, M.G. Caron, R.J. Lefkowitz, and J.W. Lomasney Mol. Pharmacol. 42 1992 1
- (1992) Mol. Pharmacol. , vol.42 , pp. 1
- Bylund, D.B.¹ Blaxall, H.S.² Iverson, L.J.³ Caron, M.G.⁴ Lefkowitz, R.J.⁵ Lomasney, J.W.⁶

17
- 19544378217
- U.S. Patent. 6,444,681, 2002;
- Flavahan, N.; Flavahan, S.; Chotani, M.; Mitra, S.; Su, B. U.S. Patent. 6,444,681, 2002; Chem. Abstr. 2002, 137, 103
- (2002) Chem. Abstr. , vol.137 , pp. 103
- Flavahan, N.¹ Flavahan, S.² Chotani, M.³ Mitra, S.⁴ Su, B.⁵

18
- 0021054336
- M.R. Goldberg, and D. Robertson Pharmacol. Rev. 35 1983 143
- (1983) Pharmacol. Rev. , vol.35 , pp. 143
- Goldberg, M.R.¹ Robertson, D.²

19
- 0035811447
- P.S. Portoghese J. Med. Chem. 44 2001 2259
- (2001) J. Med. Chem. , vol.44 , pp. 2259
- Portoghese, P.S.¹

20
- 0034599595
- W. Zheng, L. Lei, S. Lalchandani, G. Sun, D.R. Feller, and D.D. Miller Bioorg. Med. Chem. Lett. 10 2000 627
- (2000) Bioorg. Med. Chem. Lett. , vol.10 , pp. 627
- Zheng, W.¹ Lei, L.² Lalchandani, S.³ Sun, G.⁴ Feller, D.R.⁵ Miller, D.D.⁶

21
- 0036894983
- S.G. Lalchandani, L. Lei, W. Zheng, M.M. Suni, B.M. Moore, S.B. Liggett, D.D. Miller, and D.R. Feller J. Pharmacol. Exp. Ther. 303 2002 979
- (2002) J. Pharmacol. Exp. Ther. , vol.303 , pp. 979
- Lalchandani, S.G.¹ Lei, L.² Zheng, W.³ Suni, M.M.⁴ Moore, B.M.⁵ Liggett, S.B.⁶ Miller, D.D.⁷ Feller, D.R.⁸

22
- 19544385153
- U.S. Patent 6,638,943 B2, 2003;
- Miller, D. D.; Zheng, W.; Moore, B. M.; Mustafa, S. U.S. Patent 6,638,943 B2, 2003; Chem. Abstr. 2002, 137, 794
- (2002) Chem. Abstr. , vol.137 , pp. 794
- Miller, D.D.¹ Zheng, W.² Moore, B.M.³ Mustafa, S.⁴

23
- 0031008545
- M. Pigini, P. Bousquet, A. Carotti, M. Dontenwill, M. Giannella, R. Moriconi, A. Piergentili, W. Quaglia, S.K. Tayebati, and L. Brasili Bioorg. Med. Chem. 5 1997 833
- (1997) Bioorg. Med. Chem. , vol.5 , pp. 833
- Pigini, M.¹ Bousquet, P.² Carotti, A.³ Dontenwill, M.⁴ Giannella, M.⁵ Moriconi, R.⁶ Piergentili, A.⁷ Quaglia, W.⁸ Tayebati, S.K.⁹ Brasili, L.¹⁰

24
- 0034116519
- M. Pigini, W. Quaglia, F. Gentili, G. Marucci, F. Cantalamessa, S. Franchini, C. Sorbi, and L. Brasili Bioorg. Med. Chem. 8 2000 883
- (2000) Bioorg. Med. Chem. , vol.8 , pp. 883
- Pigini, M.¹ Quaglia, W.² Gentili, F.³ Marucci, G.⁴ Cantalamessa, F.⁵ Franchini, S.⁶ Sorbi, C.⁷ Brasili, L.⁸

25
- 0037011792
- F. Gentili, P. Bousquet, L. Brasili, M. Caretto, A. Carrieri, M. Dontenwill, M. Giannella, G. Marucci, M. Perfumi, A. Piergentili, W. Quaglia, C. Rascente, and M. Pigini J. Med. Chem. 45 2002 32
- (2002) J. Med. Chem. , vol.45 , pp. 32
- Gentili, F.¹ Bousquet, P.² Brasili, L.³ Caretto, M.⁴ Carrieri, A.⁵ Dontenwill, M.⁶ Giannella, M.⁷ Marucci, G.⁸ Perfumi, M.⁹ Piergentili, A.¹⁰ Quaglia, W.¹¹ Rascente, C.¹² Pigini, M.¹³

26
- 0038248835
- F. Gentili, P. Bousquet, L. Brasili, M. Dontenwill, J. Feldman, F. Ghelfi, M. Giannella, A. Piergentili, W. Quaglia, and M. Pigini J. Med. Chem. 46 2003 2169
- (2003) J. Med. Chem. , vol.46 , pp. 2169
- Gentili, F.¹ Bousquet, P.² Brasili, L.³ Dontenwill, M.⁴ Feldman, J.⁵ Ghelfi, F.⁶ Giannella, M.⁷ Piergentili, A.⁸ Quaglia, W.⁹ Pigini, M.¹⁰

27
- 9744260987
- F. Gentili, F. Ghelfi, M. Giannella, A. Piergentili, M. Pigini, W. Quaglia, C. Vesprini, P.A. Crassous, H. Paris, and A. Carrieri J. Med. Chem. 47 2004 6160
- (2004) J. Med. Chem. , vol.47 , pp. 6160
- Gentili, F.¹ Ghelfi, F.² Giannella, M.³ Piergentili, A.⁴ Pigini, M.⁵ Quaglia, W.⁶ Vesprini, C.⁷ Crassous, P.A.⁸ Paris, H.⁹ Carrieri, A.¹⁰

28
- 0035795079
- J.W. Lee, S.I. Jun, and K. Kim Tetrahedron Lett. 42 2001 2709
- (2001) Tetrahedron Lett. , vol.42 , pp. 2709
- Lee, J.W.¹ Jun, S.I.² Kim, K.³

29
- 0015861774
- Y.C. Cheng, and W.H. Prusoff Biochem. Pharacol. 22 1973 3099
- (1973) Biochem. Pharacol. , vol.22 , pp. 3099
- Cheng, Y.C.¹ Prusoff, W.H.²

30
- 17444421249
- Abstract of papers, Philadelphia, PA, Abstract 60
- Mustafa, S. M.; Bavadekar, S. A.; Moore, B. M.; Liggett, S. B.; Feller, D. R.; Miller, D. D. Abstract of papers, 228th National Meeting of the American Chemical Society: Philadelphia, PA, 2004, Abstract 60
- (2004) 228th National Meeting of the American Chemical Society
- Mustafa, S.M.¹ Bavadekar, S.A.² Moore, B.M.³ Liggett, S.B.⁴ Feller, D.R.⁵ Miller, D.D.⁶

* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.