Discovery of selective aldo-keto reductase ligands - An on-bead assay strategy

Bioorganic and Medicinal Chemistry Letters

Volumn 15, Issue 11, 2005, Pages 2938-2942

  Dixon, Seth ^a   Robins, Lori ^a   Elling, Robert A ^a   Liu, Ruiwu ^b   Lam, Kit S ^b   Wilson, David K ^a   Kurth, Mark J ^a  

^a UNIVERSITY OF CALIFORNIA   (United States)

^b UNIVERSITY OF CALIFORNIA   (United States)

Author keywords

ALR1; ALR2; On bead assay; Protein binding; Protein fluorescent labeling; Selective binding

Indexed keywords

ALDEHYDE REDUCTASE; LIGAND; OXIDOREDUCTASE;

ARTICLE; ENZYME ACTIVITY; ENZYME STRUCTURE; FLUORESCENCE MICROSCOPY; LIGAND BINDING; ULTRAVIOLET SPECTROSCOPY;

ALCOHOL OXIDOREDUCTASES; ALDEHYDE REDUCTASE; LIGANDS; MICROSCOPY, FLUORESCENCE; MODELS, MOLECULAR;

EID: 19544371932     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2005.03.010     Document Type: Article

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