Novel amide-based inhibitors of inosine 5′-monophosphate dehydrogenase

Bioorganic and Medicinal Chemistry Letters

Volumn 12, Issue 20, 2002, Pages 2879-2882

  Watterson, Scott H ^a   Liu, Chunjian ^a   Dhar, T G Murali ^a   Gu, Henry H ^a   Pitts, William J ^a   Barrish, Joel C ^a   Fleener, Catherine A ^a   Rouleau, Katherine ^a   Sherbina, N Z ^a   Hollenbaugh, Diane L ^a   Iwanowicz, Edwin J ^a  

^a BRISTOL MYERS SQUIBB   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

ENZYME INHIBITOR; INOSINATE DEHYDROGENASE; INOSINATE DEHYDROGENASE INHIBITOR;

ARTICLE; CONTROLLED STUDY; DRUG SYNTHESIS; ENZYME INHIBITION; HUMAN; HUMAN CELL; IN VITRO STUDY; STRUCTURE ACTIVITY RELATION;

AMIDES; ANTIVIRAL AGENTS; CRYSTALLOGRAPHY, X-RAY; ENZYME INHIBITORS; GASTROINTESTINAL DISEASES; IMMUNOSUPPRESSIVE AGENTS; IMP DEHYDROGENASE; INDICATORS AND REAGENTS; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 18644380984     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0960-894X(02)00601-7     Document Type: Article

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