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Bioorganic and Medicinal Chemistry Letters

Volumn 12, Issue 8, 2002, Pages 1199-1202

Anthranilate sulfonamide hydroxamate TACE inhibitors. Part 2: SAR of the acetylenic P1′ group

(14) Levin, J I a Chen, J M a Du, M T a Nelson, F C a Killar, L M a Skala, S a Sung, A a Jin, G a Cowling, R a Barone, D b March, C J b Mohler, K M b Black, R A b Skotnicki, J S a

a PFIZER INC (United States)

b AMGEN INC (United States)

Author keywords

[No Author keywords available]

Indexed keywords

ANTHRANILIC ACID; ENZYME INHIBITOR; HYDROXAMIC ACID; INTERSTITIAL COLLAGENASE; SULFONAMIDE; TUMOR NECROSIS FACTOR ALPHA; TUMOR NECROSIS FACTOR ALPHA CONVERTING ENZYME;

ANIMAL EXPERIMENT; ARTICLE; CHEMICAL STRUCTURE; CONTROLLED STUDY; DRUG ACTIVITY; DRUG POTENCY; DRUG SELECTIVITY; ENZYME ISOLATION; IN VITRO STUDY; IN VIVO STUDY; MOUSE; NONHUMAN; STRUCTURE ACTIVITY RELATION;

ACETYLENE; ADAM PROTEINS; ANTHRANILIC ACIDS; ENZYME INHIBITORS; HYDROXAMIC ACIDS; METALLOENDOPEPTIDASES; STRUCTURE-ACTIVITY RELATIONSHIP; SULFONAMIDES;

EID: 18344375458 PISSN: 0960894X EISSN: None Source Type: Journal
DOI: 10.1016/S0960-894X(02)00136-1 Document Type: Article

Times cited : (71)

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