Identification of potent and selective oxytocin antagonists. Part 2: Further investigation of benzofuran derivatives

Bioorganic and Medicinal Chemistry Letters

Volumn 12, Issue 10, 2002, Pages 1405-1411

  Wyatt, Paul G ^a   Allen, Michael J ^a   Chilcott, Josie ^a   Gardner, Christopher J ^a   Livermore, David G ^a   Mordaunt, Jackie E ^a   Nerozzi, Fabrizio ^a   Patel, Mamta ^a   Perren, Marion J ^a   Weingarten, Gordon G ^a   Shabbir, Shalia ^a   Woollard, Patrick M ^a   Zhou, Ping ^a  

^a GLAXOSMITHKLINE   (United Kingdom)

Author keywords

[No Author keywords available]

Indexed keywords

ATOSIBAN; BENZOFURAN DERIVATIVE; HUMAN SERUM ALBUMIN; OXYTOCIN; OXYTOCIN ANTAGONIST; OXYTOCIN RECEPTOR; SERUM ALBUMIN;

ARTICLE; DRUG ACTIVITY; DRUG BIOAVAILABILITY; DRUG IDENTIFICATION; DRUG POTENCY; DRUG SELECTIVITY; DRUG SYNTHESIS; HUMAN; NONHUMAN; PROTEIN BINDING; STRUCTURE ACTIVITY RELATION;

ANIMALS; BENZOFURANS; DRUG DESIGN; FEMALE; HUMANS; KINETICS; MODELS, MOLECULAR; MOLECULAR CONFORMATION; OXYTOCIN; RATS; RECEPTORS, OXYTOCIN; STRUCTURE-ACTIVITY RELATIONSHIP; UTERINE CONTRACTION;

EID: 18344361835     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0960-894X(02)00160-9     Document Type: Article

References (18)