메뉴 건너뛰기




Volumn 94, Issue 1-3 SPEC. ISS., 2005, Pages 219-227

The effects of 2-methoxyoestrogen sulphamates on the in vitro and in vivo proliferation of breast cancer cells

Author keywords

Breast cancer; Methoxyoestrogen sulphamate; Oestrogens; Oestrone sulphate; Steroid sulphatase

Indexed keywords

2 METHOXYESTRADIOL 17BETA CYANOMETHYL 3 O SULFAMATE; 2 METHOXYESTRADIOL BIS(SULFAMATE); ESTRADIOL DERIVATIVE; STERYL SULFATASE; UNCLASSIFIED DRUG;

EID: 18144409797     PISSN: 09600760     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.jsbmb.2005.01.022     Document Type: Article
Times cited : (31)

References (31)
  • 1
    • 0018648555 scopus 로고
    • The conversion of androstenedione to oestrone and production of oestrone in women with endometrial cancer
    • M.J. Reed, J.D. Hutton, P.M. Baxendale, V.H.T. James, H.S. Jacobs, and R.P. Fisher The conversion of androstenedione to oestrone and production of oestrone in women with endometrial cancer J. Steroid Biochem. 11 1979 905 911
    • (1979) J. Steroid Biochem. , vol.11 , pp. 905-911
    • Reed, M.J.1    Hutton, J.D.2    Baxendale, P.M.3    James, V.H.T.4    Jacobs, H.S.5    Fisher, R.P.6
  • 2
    • 0023509164 scopus 로고
    • Aromatase activity in normal breast and breast tumour tissue: In vivo and in vitro studies
    • V.H.T. James, J.M. McNeill, L.C. Lai, C.J. Newton, M.W. Ghilchik, and M.J. Reed Aromatase activity in normal breast and breast tumour tissue: in vivo and in vitro studies Steroids 50 1987 269 279
    • (1987) Steroids , vol.50 , pp. 269-279
    • James, V.H.T.1    McNeill, J.M.2    Lai, L.C.3    Newton, C.J.4    Ghilchik, M.W.5    Reed, M.J.6
  • 3
    • 0024419217 scopus 로고
    • In situ oestrone synthesis in normal breast and breast tumour tissue: Effect of treatment with 4-hydroxyandrostenedione
    • M.J. Reed, A.M. Owen, L.C. Lai, N.G. Coldham, M.W. Ghilchik, N.A. Shaikh, and V.H.T. James In situ oestrone synthesis in normal breast and breast tumour tissue: effect of treatment with 4-hydroxyandrostenedione Int. J. Cancer 44 1989 233 237
    • (1989) Int. J. Cancer , vol.44 , pp. 233-237
    • Reed, M.J.1    Owen, A.M.2    Lai, L.C.3    Coldham, N.G.4    Ghilchik, M.W.5    Shaikh, N.A.6    James, V.H.T.7
  • 4
    • 0035716365 scopus 로고    scopus 로고
    • Local endocrine effects of aromatase inhibitors within the breast
    • W.R. Miller, and J.M. Dixon Local endocrine effects of aromatase inhibitors within the breast J. Steroid Biochem. Mol. Biol. 79 2001 93 102
    • (2001) J. Steroid Biochem. Mol. Biol. , vol.79 , pp. 93-102
    • Miller, W.R.1    Dixon, J.M.2
  • 5
    • 0036887724 scopus 로고    scopus 로고
    • Regulation of estrogen synthesis in postmenopausal women
    • A. Purohit, and M.J. Reed Regulation of estrogen synthesis in postmenopausal women Steroids 67 2002 979 983
    • (2002) Steroids , vol.67 , pp. 979-983
    • Purohit, A.1    Reed, M.J.2
  • 6
    • 0029886370 scopus 로고    scopus 로고
    • Active site-directed inhibition of estrone sulfatase by non steroidal Coumarin sulfamates
    • L.W.L. Woo, A. Purohit, M.J. Reed, and B.V.L. Potter Active site-directed inhibition of estrone sulfatase by non steroidal Coumarin sulfamates J. Med. Chem. 39 1996 1349 1351
    • (1996) J. Med. Chem. , vol.39 , pp. 1349-1351
    • Woo, L.W.L.1    Purohit, A.2    Reed, M.J.3    Potter, B.V.L.4
  • 7
    • 0034234951 scopus 로고    scopus 로고
    • In vivo inhibition of estrone sulfatase activity and growth of nitrosomethylurea-induced mammary tumors by 667 COUMATE
    • A. Purohit, L.W.L. Woo, B.V.L. Potter, and M.J. Reed In vivo inhibition of estrone sulfatase activity and growth of nitrosomethylurea-induced mammary tumors by 667 COUMATE Cancer Res. 60 2000 3394 3396
    • (2000) Cancer Res. , vol.60 , pp. 3394-3396
    • Purohit, A.1    Woo, L.W.L.2    Potter, B.V.L.3    Reed, M.J.4
  • 8
    • 0033555597 scopus 로고    scopus 로고
    • Steroid sulfatase expression is an independent predictor of recurrence in human breast cancer
    • T. Utsumi, N. Yoshimura, S. Takeuchi, J. Ando, M. Maruta, K. Maeda, and N. Harada Steroid sulfatase expression is an independent predictor of recurrence in human breast cancer Cancer Res. 59 1999 377 381
    • (1999) Cancer Res. , vol.59 , pp. 377-381
    • Utsumi, T.1    Yoshimura, N.2    Takeuchi, S.3    Ando, J.4    Maruta, M.5    Maeda, K.6    Harada, N.7
  • 9
    • 7044253796 scopus 로고    scopus 로고
    • Intratumoral mRNA expression and genes from the oestradiol metabolic pathway and clinical and histopathological parameters of breast cancer
    • N. Yoshimura, N. Harada, I. Bukholm, R. Karesen, A.-L. Borresen-Dale, and V.N. Kristensen Intratumoral mRNA expression and genes from the oestradiol metabolic pathway and clinical and histopathological parameters of breast cancer Breast Cancer Res. 6 2004 R46 R55
    • (2004) Breast Cancer Res. , vol.6
    • Yoshimura, N.1    Harada, N.2    Bukholm, I.3    Karesen, R.4    Borresen-Dale, A.-L.5    Kristensen, V.N.6
  • 11
    • 0343178292 scopus 로고
    • Covalent binding of endogenous 16α-hydroxyestrone to estradiol receptor in human breast cancer cells: Characterization and intra-nuclear location
    • G.E. Swaneck, and J. Fishman Covalent binding of endogenous 16α-hydroxyestrone to estradiol receptor in human breast cancer cells: characterization and intra-nuclear location Proc. Natl. Acad. Sci. U.S.A. 85 1988 7831 7835
    • (1988) Proc. Natl. Acad. Sci. U.S.A. , vol.85 , pp. 7831-7835
    • Swaneck, G.E.1    Fishman, J.2
  • 12
    • 0000317180 scopus 로고    scopus 로고
    • Is 2-methoxyestradiol an endogenous estrogen metabolite that inhibits mammary carcinogenesis?
    • B.T. Zhu, and A.H. Conney Is 2-methoxyestradiol an endogenous estrogen metabolite that inhibits mammary carcinogenesis? Cancer Res. 58 1998 2269 2277
    • (1998) Cancer Res. , vol.58 , pp. 2269-2277
    • Zhu, B.T.1    Conney, A.H.2
  • 13
    • 0024373582 scopus 로고
    • The cytotoxic effects of estradiol-17β, catecholestradiols and methoxyestradiols on dividing MCF-7 and HeLa cells
    • J. Seegers, M-L. Aveling, C.H. Van Aswegen, M. Cross, F. Koch, and W.S. Joubert The cytotoxic effects of estradiol-17β, catecholestradiols and methoxyestradiols on dividing MCF-7 and HeLa cells J. Steroid Biochem. 32 1989 797 809
    • (1989) J. Steroid Biochem. , vol.32 , pp. 797-809
    • Seegers, J.1    Aveling, M.-L.2    Van Aswegen, C.H.3    Cross, M.4    Koch, F.5    Joubert, W.S.6
  • 14
    • 0028331925 scopus 로고
    • 2-Methoxyestradiol, an endogenous mammalian metabolite, inhibits tubulin polymerization by interacting at the colchicine site
    • R.J. D'Amato, C. Lin, E. Flynn, J. Folkman, and E. Hamel 2-Methoxyestradiol, an endogenous mammalian metabolite, inhibits tubulin polymerization by interacting at the colchicine site Proc. Natl. Acad. Sci. U.S.A. 91 1994 3964 3968
    • (1994) Proc. Natl. Acad. Sci. U.S.A. , vol.91 , pp. 3964-3968
    • D'Amato, R.J.1    Lin, C.2    Flynn, E.3    Folkman, J.4    Hamel, E.5
  • 16
    • 0028220858 scopus 로고    scopus 로고
    • The endogenous oestrogen metabolite 2-methoxyoestradiol inhibits angiogenesis and suppresses tumour growth
    • T. Fotsis, Y. Zhang, M.S. Pepper, H. Adlercreutz, R. Montesano, P.P. Nawroth, and L. Schweigerer The endogenous oestrogen metabolite 2-methoxyoestradiol inhibits angiogenesis and suppresses tumour growth Nature 368 1997 237 239
    • (1997) Nature , vol.368 , pp. 237-239
    • Fotsis, T.1    Zhang, Y.2    Pepper, M.S.3    Adlercreutz, H.4    Montesano, R.5    Nawroth, P.P.6    Schweigerer, L.7
  • 17
    • 0031015504 scopus 로고    scopus 로고
    • Inhibition of angiogenesis and breast cancer in mice by the microtuble inhibitors 2-methoxyestradiol and taxol
    • N. Klauber, S. Parangi, E. Flynn, E. Hamel, and R.J. D'Amato Inhibition of angiogenesis and breast cancer in mice by the microtuble inhibitors 2-methoxyestradiol and taxol Cancer Res. 57 1997 81 86
    • (1997) Cancer Res. , vol.57 , pp. 81-86
    • Klauber, N.1    Parangi, S.2    Flynn, E.3    Hamel, E.4    D'Amato, R.J.5
  • 19
    • 0034820420 scopus 로고    scopus 로고
    • 2-Methoxymethylestradiol: A new 2-methoxyestrogen analog that exhibits antiproliferative activity and alters tubulin dynamics
    • R.W. Bruggemeier, A.S. Bhat, C.J. Lovely, H.D. Coughenour, F. Yusuf, and W.G. Burak 2-Methoxymethylestradiol: a new 2-methoxyestrogen analog that exhibits antiproliferative activity and alters tubulin dynamics J. Steroid Biochem. Mol. Biol. 78 2001 145 156
    • (2001) J. Steroid Biochem. Mol. Biol. , vol.78 , pp. 145-156
    • Bruggemeier, R.W.1    Bhat, A.S.2    Lovely, C.J.3    Coughenour, H.D.4    Yusuf, F.5    Burak, W.G.6
  • 22
    • 0033956376 scopus 로고    scopus 로고
    • The effect of 2-methoxyestrone sulfamate on the growth of breast cancer cells and induced mammary tumors
    • A. Purohit, H.A.M. Hejaz, L. Walden, B.V.L. Potter, and M.J. Reed The effect of 2-methoxyestrone sulfamate on the growth of breast cancer cells and induced mammary tumors Int. J. Cancer 85 2000 584 589
    • (2000) Int. J. Cancer , vol.85 , pp. 584-589
    • Purohit, A.1    Hejaz, H.A.M.2    Walden, L.3    Potter, B.V.L.4    Reed, M.J.5
  • 23
    • 0034307330 scopus 로고    scopus 로고
    • Differential effects of estrone and estrone-3-O-sulfamate derivatives on mitotic arrest, apoptosis and microtuble assembly in human breast cancer cells
    • L. MacCarthy-Morrogh, P.A. Townsend, A. Purohit, H.A.M. Hejaz, B.V.L. Potter, M.J. reed, and G. Packham Differential effects of estrone and estrone-3-O-sulfamate derivatives on mitotic arrest, apoptosis and microtuble assembly in human breast cancer cells Cancer Res. 60 2000 5441 5450
    • (2000) Cancer Res. , vol.60 , pp. 5441-5450
    • MacCarthy-Morrogh, L.1    Townsend, P.A.2    Purohit, A.3    Hejaz, H.A.M.4    Potter, B.V.L.5    Reed, M.J.6    Packham, G.7
  • 25
    • 0027397024 scopus 로고
    • Inhibition of estrone sulfatase activity by estrone-3- methylthiophosphonate: A potential therapeutic agent in breast cancer
    • L.J. Duncan, A. Purohit, N.M. Howarth, B.V.L. Potter, and M.J. Reed Inhibition of estrone sulfatase activity by estrone-3-methylthiophosphonate: a potential therapeutic agent in breast cancer Cancer Res. 53 1993 298 303
    • (1993) Cancer Res. , vol.53 , pp. 298-303
    • Duncan, L.J.1    Purohit, A.2    Howarth, N.M.3    Potter, B.V.L.4    Reed, M.J.5
  • 26
    • 0029114308 scopus 로고
    • Inactivation of steroid sulfatase by an active site-directed inhibitor, estrone-3-O-sulfamate
    • A. Purohit, G.J. Williams, N.M. Howarth, B.V.L. Potter, and M.J. Reed Inactivation of steroid sulfatase by an active site-directed inhibitor, estrone-3-O-sulfamate Biochemistry 34 1995 11508 11514
    • (1995) Biochemistry , vol.34 , pp. 11508-11514
    • Purohit, A.1    Williams, G.J.2    Howarth, N.M.3    Potter, B.V.L.4    Reed, M.J.5
  • 31
    • 0028879855 scopus 로고
    • In vivo inhibition of oestrone sulphatase and dehydroepiandrosterone sulphatase by oestrone-3-O-sulphamate
    • A. Purohit, G.J. Williams, C.J. Roberts, B.V.L. Potter, and M.J. Reed In vivo inhibition of oestrone sulphatase and dehydroepiandrosterone sulphatase by oestrone-3-O-sulphamate Int. J. Cancer 63 1995 106 111
    • (1995) Int. J. Cancer , vol.63 , pp. 106-111
    • Purohit, A.1    Williams, G.J.2    Roberts, C.J.3    Potter, B.V.L.4    Reed, M.J.5


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.