SCOPUS 정보 검색 플랫폼

Tetrahedron Letters

Volumn 46, Issue 20, 2005, Pages 3587-3589

A one-pot synthesis of nitrogen-containing heteroaryl α-keto amides from heteroaryl halides

(7) Zhu, Juliang a Wong, Henry a Zhang, Zhongxing a Yin, Zhiwei a Kadow, John F a Meanwell, Nicholas A a Wang, Tao a

a BRISTOL MYERS SQUIBB (United States)

Author keywords

Acyl carbanion equivalent; Condensation oxidation; Heteroaryl keto amide; Cyano acetamide

Indexed keywords

ACETIC ACID DERIVATIVE; AMINOKETONE; ANION; CYANOACETIC ACID; HALIDE; NITROGEN; PERACETIC ACID; PIPERIDINE; UNCLASSIFIED DRUG;

ARTICLE; OXIDATION; SYNTHESIS;

EID: 17844369704 PISSN: 00404039 EISSN: None Source Type: Journal
DOI: 10.1016/j.tetlet.2005.03.100 Document Type: Article

Times cited : (22)

References (43)

1
- 0141680855
- T. Wang, Z. Zhang, O.B. Wallace, M. Deshpande, H. Fang, Z. Yang, L.M. Zadjura, D.L. Tweedie, S. Huang, F. Zhao, S. Ranadive, B.S. Robinson, Y.-F. Gong, K. Ricarrdi, T.P. Spicer, C. Deminie, R. Rose, W.S. Blair, P.-F. Lin, R.J. Colonno, and N.A. Meanwell J. Med. Chem. 46 2003 4236
- (2003) J. Med. Chem. , vol.46 , pp. 4236
- Wang, T.¹ Zhang, Z.² Wallace, O.B.³ Deshpande, M.⁴ Fang, H.⁵ Yang, Z.⁶ Zadjura, L.M.⁷ Tweedie, D.L.⁸ Huang, S.⁹ Zhao, F.¹⁰ Ranadive, S.¹¹ Robinson, B.S.¹² Gong, Y.-F.¹³ Ricarrdi, K.¹⁴ Spicer, T.P.¹⁵ Deminie, C.¹⁶ Rose, R.¹⁷ Blair, W.S.¹⁸ Lin, P.-F.¹⁹ Colonno, R.J.²⁰ Meanwell, N.A.²¹ more..

2
- 85030794607
- WO-199200278, 1992
- (b) Armistead, D. M.; Boger, J. S.; Meyers, H. V.; Saunders, J. O.; Tung, R. D. WO-199200278, 1992
- Armistead, D.M.¹ Boger, J.S.² Meyers, H.V.³ Saunders, J.O.⁴ Tung, R.D.⁵

3
- 85030800547
- WO-2002096420, 2002
- (c) Steiner, J. P.; Snyder, S.; Burnett, A. L. WO-2002096420, 2002
- Steiner, J.P.¹ Snyder, S.² Burnett, A.L.³

4
- 85030795682
- WO-199914998, 1999
- (d) Magal, E. WO-199914998, 1999
- Magal, E.¹

5
- 85030801208
- WO-2002070491, 2002
- (e) Fuji, M. WO-2002070491, 2002
- Fuji, M.¹

6
- 85030804389
- WO-2002085907, 2002
- (f) Failli, A. A.; Dusza, J. P.; Trybulski, E. J.; Memoli, K. A.; Shumsky, J. S. WO-2002085907, 2002
- Failli, A.A.¹ Dusza, J.P.² Trybulski, E.J.³ Memoli, K.A.⁴ Shumsky, J.S.⁵

7
- 0034618184
- A. Slassi, L. Edwards, A. O'Brien, C.Q. Meng, T. Xin, C. Seto, D.K.H. Lee, N. MacLean, D. Hynd, C. Chen, H. Wang, R. Kamboj, and S. Rakhit Bioorg. Med. Chem. Lett. 10 2000 1707
- (2000) Bioorg. Med. Chem. Lett. , vol.10 , pp. 1707
- Slassi, A.¹ Edwards, L.² O'Brien, A.³ Meng, C.Q.⁴ Xin, T.⁵ Seto, C.⁶ Lee, D.K.H.⁷ MacLean, N.⁸ Hynd, D.⁹ Chen, C.¹⁰ Wang, H.¹¹ Kamboj, R.¹² Rakhit, S.¹³

8
- 0034693086
- D.StC. Black, N. Kumar, and D.B. McConnell Tetrahedron 56 2000 8513
- (2000) Tetrahedron , vol.56 , pp. 8513
- Black, D.StC.¹ Kumar, N.² McConnell, D.B.³

9
- 0033532007
- S. Couve-Bonnaire, J.-F. Carpentier, Y. Castanet, and A. Mortreux Tetrahedron Lett. 40 1999 3717
- (1999) Tetrahedron Lett. , vol.40 , pp. 3717
- Couve-Bonnaire, S.¹ Carpentier, J.-F.² Castanet, Y.³ Mortreux, A.⁴

10
- 0041374164
- Z. Yang, Z. Zhang, N.A. Meanwell, J.F. Kadow, and T. Wang Org. Lett. 4 2002 1103
- (2002) Org. Lett. , vol.4 , pp. 1103
- Yang, Z.¹ Zhang, Z.² Meanwell, N.A.³ Kadow, J.F.⁴ Wang, T.⁵

11
- 0030061605
- I.T. Forbes, H.K.A. Morgan, and M. Thompson Synth. Commun. 26 1996 745
- (1996) Synth. Commun. , vol.26 , pp. 745
- Forbes, I.T.¹ Morgan, H.K.A.² Thompson, M.³

12
- 0028170373
- S. El-Kousy Pharmazie 49 1994 480
- (1994) Pharmazie , vol.49 , pp. 480
- El-Kousy, S.¹

13
- 37049069626
- G. L'abbe, L. Bastin, W. Dehaen, S. Toppet, P. Delbeke, D. Vlieghe, and L. Van Meervelt J. Chem. Soc., Perkin Trans. 1 1994 2545
- (1994) J. Chem. Soc., Perkin Trans. 1 , pp. 2545
- L'Abbe, G.¹ Bastin, L.² Dehaen, W.³ Toppet, S.⁴ Delbeke, P.⁵ Vlieghe, D.⁶ Van Meervelt, L.⁷

14
- 84993624370
- L.H. Klemm, D.R. Muchiri, M. Anderson, W. Salbador, and J. Ford J. Heterocycl. Chem. 31 1994 261
- (1994) J. Heterocycl. Chem. , vol.31 , pp. 261
- Klemm, L.H.¹ Muchiri, D.R.² Anderson, M.³ Salbador, W.⁴ Ford, J.⁵

15
- 0002837667
- Z. El-Gendy Indian J. Chem., Sect. B 33 1994 326
- (1994) Indian J. Chem., Sect. B , vol.33 , pp. 326
- El-Gendy, Z.¹

16
- 0026316851
- N. Hamamichi Tetrahedron Lett. 32 1991 7415
- (1991) Tetrahedron Lett. , vol.32 , pp. 7415
- Hamamichi, N.¹

17
- 0025981614
- S. Ohba, S. Konno, and H. Yamanaka Chem. Pharm. Bull. 39 1991 486
- (1991) Chem. Pharm. Bull. , vol.39 , pp. 486
- Ohba, S.¹ Konno, S.² Yamanaka, H.³

18
- 0001641882
- A.L. Borror, and A.F. Haeberer J. Org. Chem. 30 1965 243
- (1965) J. Org. Chem. , vol.30 , pp. 243
- Borror, A.L.¹ Haeberer, A.F.²

19
- 0142026581
- J. You, and J.G. Verkade J. Org. Chem. 68 2003 8003
- (2003) J. Org. Chem. , vol.68 , pp. 8003
- You, J.¹ Verkade, J.G.²

20
- 0042912889
- C. Gao, X. Tao, Y. Qian, and J. Huang Synlett. 2003 1716
- (2003) Synlett. , pp. 1716
- Gao, C.¹ Tao, X.² Qian, Y.³ Huang, J.⁴

21
- 0028113602
- H. Suzuki, H. Abe, and S.V. Thiruvikraman J. Org. Chem. 59 1994 6116
- (1994) J. Org. Chem. , vol.59 , pp. 6116
- Suzuki, H.¹ Abe, H.² Thiruvikraman, S.V.³

22
- 0027731073
- K. Okuro, M. Furuune, M. Miura, and M. Nomura J. Org. Chem. 58 1993 7606
- (1993) J. Org. Chem. , vol.58 , pp. 7606
- Okuro, K.¹ Furuune, M.² Miura, M.³ Nomura, M.⁴

23
- 58149155215
- T. Sakamoto, E. Katoh, Y. Kondo, and H. Yamanaka Chem. Pharm. Bull. 36 1988 1664
- (1988) Chem. Pharm. Bull. , vol.36 , pp. 1664
- Sakamoto, T.¹ Katoh, E.² Kondo, Y.³ Yamanaka, H.⁴

24
- 85078346696
- M. Uno, K. Seto, W. Ueda, M. Masuda, and S. Takahashi Synthesis 1985 506
- (1985) Synthesis , pp. 506
- Uno, M.¹ Seto, K.² Ueda, W.³ Masuda, M.⁴ Takahashi, S.⁵

25
- 85083051824
- A. Osuka, T. Kobayashi, and H. Suzuki Synthesis 1983 67
- (1983) Synthesis , pp. 67
- Osuka, A.¹ Kobayashi, T.² Suzuki, H.³

26
- 1242307320
- Z. Yin, Z. Zhang, J.F. Kadow, N.A. Meanwell, and T. Wang J. Org. Chem. 69 2004 1364
- (2004) J. Org. Chem. , vol.69 , pp. 1364
- Yin, Z.¹ Zhang, Z.² Kadow, J.F.³ Meanwell, N.A.⁴ Wang, T.⁵

27
- 1242307319
- Z. Zhang, Z. Yin, J.F. Kadow, N.A. Meanwell, and T. Wang J. Org. Chem. 69 2004 1360
- (2004) J. Org. Chem. , vol.69 , pp. 1360
- Zhang, Z.¹ Yin, Z.² Kadow, J.F.³ Meanwell, N.A.⁴ Wang, T.⁵

28
- 0035966599
- H. Hamada, T. Tanaka, T. Furuya, H. Takahata, and H. Nemoto Tetrahedron Lett. 42 2001 909
- (2001) Tetrahedron Lett. , vol.42 , pp. 909
- Hamada, H.¹ Tanaka, T.² Furuya, T.³ Takahata, H.⁴ Nemoto, H.⁵

29
- 0019193201
- K.A. Parker, and J. Kallmerten J. Org. Chem. 45 1980 2614
- (1980) J. Org. Chem. , vol.45 , pp. 2614
- Parker, K.A.¹ Kallmerten, J.²

30
- 0002007261
- Y. Masuyama, Y. Ueno, and M. Okawara Chem. Lett. 1977 1439
- (1977) Chem. Lett. , pp. 1439
- Masuyama, Y.¹ Ueno, Y.² Okawara, M.³

31
- 0141784398
- S.J. Selikson, and D.S. Watt Tetrahedron Lett. 15 1974 3029
- (1974) Tetrahedron Lett. , vol.15 , pp. 3029
- Selikson, S.J.¹ Watt, D.S.²

32
- 33847802830
- S.J. Selikson, and D.S. Watt J. Org. Chem. 40 1975 267
- (1975) J. Org. Chem. , vol.40 , pp. 267
- Selikson, S.J.¹ Watt, D.S.²

33
- 0346925658
- R.R. Wroble, and D.S. Watt J. Org. Chem. 41 1976 2939
- (1976) J. Org. Chem. , vol.41 , pp. 2939
- Wroble, R.R.¹ Watt, D.S.²

34
- 0021338245
- M. Kuchar, B. Brunova, V. Rejholec, M. Jelinkova, J. Holubek, and O. Nemecek Collect. Czech. Chem. Commun. 49 1984 122
- (1984) Collect. Czech. Chem. Commun. , vol.49 , pp. 122
- Kuchar, M.¹ Brunova, B.² Rejholec, V.³ Jelinkova, M.⁴ Holubek, J.⁵ Nemecek, O.⁶

35
- 0028068289
- R.B. Grossman, and S.V. Ley Tetrahedron 50 1994 11553
- (1994) Tetrahedron , vol.50 , pp. 11553
- Grossman, R.B.¹ Ley, S.V.²

36
- 33947294845
- N. Rabjohn, and C.A. Harbert J. Org. Chem. 35 1970 3240
- (1970) J. Org. Chem. , vol.35 , pp. 3240
- Rabjohn, N.¹ Harbert, C.A.²

37
- 0026040506
- S. Adam Tetrahedron 47 1991 7609
- (1991) Tetrahedron , vol.47 , pp. 7609
- Adam, S.¹

38
- 0001557636
- A. Ouladyakhlef, S. Boukhris, A. Souizi, and A. Robert Bull. Soc. Chim. France 134 1997 111
- (1997) Bull. Soc. Chim. France , vol.134 , pp. 111
- Ouladyakhlef, A.¹ Boukhris, S.² Souizi, A.³ Robert, A.⁴

39
- 0030041808
- I. Chehidi, M.M. Chaabouni, and A. Baklouti Synth. Commun. 26 1996 237
- (1996) Synth. Commun. , vol.26 , pp. 237
- Chehidi, I.¹ Chaabouni, M.M.² Baklouti, A.³

40
- 0002137256
- A. Majcen-le Marechal, J. Pavc, A. Robert, and P. le Grel J. Chem. Soc., Perkin Trans. 1 1994 2045
- (1994) J. Chem. Soc., Perkin Trans. 1 , pp. 2045
- Majcen-Le Marechal, A.¹ Pavc, J.² Robert, A.³ Le Grel, P.⁴

41
- 0001210887
- J.H. Babler, C.J. Marcuccilli, and J.E. Oblong Synth. Commun. 20 1990 1831
- (1990) Synth. Commun. , vol.20 , pp. 1831
- Babler, J.H.¹ Marcuccilli, C.J.² Oblong, J.E.³

42
- 85030797586
- note
- The reaction and the subsequent work-up should be undertaken with care in a well ventilated hood due to the possibility of HCN liberation

43
- 85030794958
- note
- 4: 281.1250. Found 281.1254

* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.