메뉴 건너뛰기




Volumn 27, Issue 3, 2005, Pages 161-165

Actions of tacrine and galanthamine on histamine-N-methyltransferase

Author keywords

Alzheimer's disease; Galanthamine; Histamine N methyltransferase; Tacrine

Indexed keywords

GALANTAMINE; HISTAMINE; HISTAMINE METHYLTRANSFERASE; HISTAMINE RECEPTOR; TACRINE;

EID: 17644418402     PISSN: 03790355     EISSN: None     Source Type: Journal    
DOI: 10.1358/mf.2005.27.3.890872     Document Type: Article
Times cited : (19)

References (38)
  • 1
    • 0000022008 scopus 로고    scopus 로고
    • Histamine
    • Siegel, G.J., Agranoff, B.W., Albers, R.W., Fisher, S.K., Uhler, M.D. (Eds.). Lippincott-Raven: Philadelphia
    • Hough, L.B. Histamine. In: Basic Neurochemistry. Siegel, G.J., Agranoff, B.W., Albers, R.W., Fisher, S.K., Uhler, M.D. (Eds.). Lippincott-Raven: Philadelphia 1999, 293-313.
    • (1999) Basic Neurochemistry , pp. 293-313
    • Hough, L.B.1
  • 3
    • 0002653043 scopus 로고
    • Histamine N-methyltransferase
    • Boulton, A.A., Baker, G.B., Yu, P.H., Clifton, N.J. (Eds.). Humana Press
    • Verburg, K.M., Henry, D.P. Histamine N-methyltransferase. In: Neuromethods: Neurotransmitter Enzymes. Boulton, A.A., Baker, G.B., Yu, P.H., Clifton, N.J. (Eds.). Humana Press 1986, 147-204.
    • (1986) Neuromethods: Neurotransmitter Enzymes , pp. 147-204
    • Verburg, K.M.1    Henry, D.P.2
  • 4
    • 0034812118 scopus 로고    scopus 로고
    • Two polymorphic forms of human histamine methyltransferase: Structural, thermal, and kinetic comparisons
    • Horton, J.R., Sawada, K., Nishibori, M., Zhang, X., Cheng, X. Two polymorphic forms of human histamine methyltransferase: Structural, thermal, and kinetic comparisons. Structure (Camb.) 2001, 9: 837-49.
    • (2001) Structure (Camb.) , vol.9 , pp. 837-849
    • Horton, J.R.1    Sawada, K.2    Nishibori, M.3    Zhang, X.4    Cheng, X.5
  • 5
    • 0034094292 scopus 로고    scopus 로고
    • Neuronal and vascular localization of histamine N-methyltransferase in the bovine central nervous system
    • Nishibori, M., Tahara, A., Sawada, K., Sakiyama, J., Nakaya, N., Saeki, K. Neuronal and vascular localization of histamine N-methyltransferase in the bovine central nervous system. Eur J Neurosci 2000, 12: 415-24.
    • (2000) Eur J Neurosci , vol.12 , pp. 415-424
    • Nishibori, M.1    Tahara, A.2    Sawada, K.3    Sakiyama, J.4    Nakaya, N.5    Saeki, K.6
  • 6
    • 0036723814 scopus 로고    scopus 로고
    • Membrane-boundhistamine-N-methyltransferase in mouse brain: Possible role in the synoptic inactivation of neuronal histamine
    • Barnes, W.G., Hough, L.B. Membrane-boundhistamine-N-methyltransferase in mouse brain: Possible role in the synoptic inactivation of neuronal histamine. J Neurochem 2002, 82: 1262-71.
    • (2002) J Neurochem , vol.82 , pp. 1262-1271
    • Barnes, W.G.1    Hough, L.B.2
  • 7
    • 0343580446 scopus 로고    scopus 로고
    • Neuronal histamine deficit in Alzheimer's disease
    • Panula, P., Rinne, J., Kuokkanen, K. et al. Neuronal histamine deficit in Alzheimer's disease. Neuroscience 1998, 82: 993-97.
    • (1998) Neuroscience , vol.82 , pp. 993-997
    • Panula, P.1    Rinne, J.2    Kuokkanen, K.3
  • 8
    • 0034706072 scopus 로고    scopus 로고
    • Histamine H(1) receptors in patients with Alzheimer's disease assessed by positron emission tomography
    • Higuchi, M., Yanai, K., Okamura, N. et al. Histamine H(1) receptors in patients with Alzheimer's disease assessed by positron emission tomography. Neuroscience 2000, 99: 721-29.
    • (2000) Neuroscience , vol.99 , pp. 721-729
    • Higuchi, M.1    Yanai, K.2    Okamura, N.3
  • 9
    • 0004945541 scopus 로고    scopus 로고
    • Clinical presentation and course of Alzheimer's disease
    • Terry, R.D., Katzman, R., Bick, K.L., Sisodia, S.S. (Eds.). Lippincott Williams & Wilkins: Philadelphia
    • Morris, J.C. Clinical presentation and course of Alzheimer's disease. In: Alzheimer's Disease. Terry, R.D., Katzman, R., Bick, K.L., Sisodia, S.S. (Eds.). Lippincott Williams & Wilkins: Philadelphia 1999, 11-25.
    • (1999) Alzheimer's Disease , pp. 11-25
    • Morris, J.C.1
  • 10
    • 0019972810 scopus 로고
    • The cholinergic hypothesis of geriatric memory dysfunction
    • Bartus, R.T., Dean, R.L., III, Beer, B., Lippa, A.S. The cholinergic hypothesis of geriatric memory dysfunction. Science 1982, 217: 408-14.
    • (1982) Science , vol.217 , pp. 408-414
    • Bartus, R.T.1    Dean III, R.L.2    Beer, B.3    Lippa, A.S.4
  • 11
    • 0034876669 scopus 로고    scopus 로고
    • Maintaining cognitive function in Alzheimer disease: How effective are current treatments?
    • Tariot, P.N. Maintaining cognitive function in Alzheimer disease: How effective are current treatments? Alzheimer Dis Assoc Disord 2001, 15: 526-533.
    • (2001) Alzheimer Dis Assoc Disord , vol.15 , pp. 526-533
    • Tariot, P.N.1
  • 12
    • 0033966913 scopus 로고    scopus 로고
    • Huprine X is a novel high-affinity inhibitor of acetylcholineslerase that is of interest for treatment of Alzheimer's disease
    • Camps, P., Cusack, B., Mallender, W.D. et al. Huprine X is a novel high-affinity inhibitor of acetylcholineslerase that is of interest for treatment of Alzheimer's disease. Mol Pharmacol 2000, 57: 409-17.
    • (2000) Mol Pharmacol , vol.57 , pp. 409-417
    • Camps, P.1    Cusack, B.2    Mallender, W.D.3
  • 13
    • 0025079151 scopus 로고
    • Inhibition of rat brain histamine-N-methyltransferase by 9-amino-1,2,3,4-tetrahydroacridine (THA)
    • Cumming, P., Reiner, P.B., Vincent, S.R. Inhibition of rat brain histamine-N-methyltransferase by 9-amino-1,2,3,4-tetrahydroacridine (THA). Biochem Pharmacol 1990, 40: 1345-50.
    • (1990) Biochem Pharmacol , vol.40 , pp. 1345-1350
    • Cumming, P.1    Reiner, P.B.2    Vincent, S.R.3
  • 14
    • 0025727739 scopus 로고
    • 9-Amino-1,2,3,4-tetrahydroacridine is a potent inhibitor of histamine N-methyltransferase
    • Nishibori, M., Oishi, R., Itoh, Y., Saeki, K. 9-Amino-1,2,3,4- tetrahydroacridine is a potent inhibitor of histamine N-methyltransferase. Jpn J Pharmacol 1991, 55: 539-46.
    • (1991) Jpn J Pharmacol , vol.55 , pp. 539-546
    • Nishibori, M.1    Oishi, R.2    Itoh, Y.3    Saeki, K.4
  • 15
    • 0035251762 scopus 로고    scopus 로고
    • Galantamine, a cholinesterase inhibitor that allosterically modulates nicotinic receptors: Effects on the course of Alzheimer's disease
    • Coyle, J., Kershaw, P. Galantamine, a cholinesterase inhibitor that allosterically modulates nicotinic receptors: Effects on the course of Alzheimer's disease. Biol Psychiatry 2001, 49: 289-99.
    • (2001) Biol Psychiatry , vol.49 , pp. 289-299
    • Coyle, J.1    Kershaw, P.2
  • 16
    • 0035852773 scopus 로고    scopus 로고
    • Galantamine: Effect on nicotinic receptor binding, acetylcholinesterase inhibition, and learning
    • Woodruff-Pak, D.S., Vogel, R.W., III, Wenk, G.L. Galantamine: effect on nicotinic receptor binding, acetylcholinesterase inhibition, and learning. Proc Natl Acad Sci U S A 2001, 98: 2089-209.
    • (2001) Proc Natl Acad Sci U S A , vol.98 , pp. 2089-2209
    • Woodruff-Pak, D.S.1    Vogel III, R.W.2    Wenk, G.L.3
  • 17
    • 0021112663 scopus 로고
    • Rat histamine N-methyltransferase. Quantification, tissue distribution, purification, and immunologic properties
    • Bowsher, R.R., Verburg, K.M., Henry, D.P. Rat histamine N-methyltransferase. Quantification, tissue distribution, purification, and immunologic properties. J Biol Chem 1983, 258: 12215-2220.
    • (1983) J Biol Chem , vol.258 , pp. 12215-12220
    • Bowsher, R.R.1    Verburg, K.M.2    Henry, D.P.3
  • 18
    • 0029875216 scopus 로고    scopus 로고
    • Human histamine N-methyltransferase gene: Structural characterization and chromosomal location
    • Aksoy, S., Raftogianis, R., Weinshilboum, R. Human histamine N-methyltransferase gene: Structural characterization and chromosomal location. Biochem Biophys Res Commun 1996, 219: 548-54.
    • (1996) Biochem Biophys Res Commun , vol.219 , pp. 548-554
    • Aksoy, S.1    Raftogianis, R.2    Weinshilboum, R.3
  • 19
    • 0031969375 scopus 로고    scopus 로고
    • Human histamine N-methyltransferase pharmacogenetics: Common genetic polymorphisms that alter activity
    • Preuss, C.V., Wood, T.C., Szumlanski, C.L. et al. Human histamine N-methyltransferase pharmacogenetics: Common genetic polymorphisms that alter activity. Mol Pharmacol 1998, 53: 708-17.
    • (1998) Mol Pharmacol , vol.53 , pp. 708-717
    • Preuss, C.V.1    Wood, T.C.2    Szumlanski, C.L.3
  • 20
    • 0020625427 scopus 로고
    • A new radioenzymatic assay for histamine using purified histamine N-methyltransferase
    • Verburg, K.M., Bowsher, R.R., Henry, D.P. A new radioenzymatic assay for histamine using purified histamine N-methyltransferase. Life Sci 1983, 32: 2855-67.
    • (1983) Life Sci , vol.32 , pp. 2855-2867
    • Verburg, K.M.1    Bowsher, R.R.2    Henry, D.P.3
  • 21
    • 0001880598 scopus 로고    scopus 로고
    • Cholinergic systems in Alzheimer's disease
    • Terry, R.D., Katzman, R., Bick, K.L., Sisodia, S.S. (Eds.). Lippincott Williams & Wilkins: Philadelphia
    • Geula, C., Mesulam, M. Cholinergic systems in Alzheimer's disease. In: Alzheimers Disease. Terry, R.D., Katzman, R., Bick, K.L., Sisodia, S.S. (Eds.). Lippincott Williams & Wilkins: Philadelphia 1999, 11-25.
    • (1999) Alzheimers Disease , pp. 11-25
    • Geula, C.1    Mesulam, M.2
  • 22
    • 0027454927 scopus 로고
    • A detailed autoradiographic mapping of histamine H3 receptors in rat brain areas
    • Pollard, H., Moreau, J., Arrang, J.M., Schwartz, J.C. A detailed autoradiographic mapping of histamine H3 receptors in rat brain areas. Neuroscience 1993, 52: 169-89.
    • (1993) Neuroscience , vol.52 , pp. 169-189
    • Pollard, H.1    Moreau, J.2    Arrang, J.M.3    Schwartz, J.C.4
  • 23
    • 0029583271 scopus 로고
    • Effects of thioperamide on the cholinergic system and the step-through passive avoidance test in mice
    • Miyazaki, S., Imaizumi, M., Onodera, K. Effects of thioperamide on the cholinergic system and the step-through passive avoidance test in mice. Methods Find Exp Clin Pharmacol 1995, 17: 653-58.
    • (1995) Methods Find Exp Clin Pharmacol , vol.17 , pp. 653-658
    • Miyazaki, S.1    Imaizumi, M.2    Onodera, K.3
  • 24
    • 0030849712 scopus 로고    scopus 로고
    • Effects of clobenpropit (VUF-9153), a histamine H3-receptor antagonist, on learning and memory, and on cholinergic and monoaminergic systems in mice
    • Miyazaki, S., Onodera, K., Imaizumi, M., Timmerman, H. Effects of clobenpropit (VUF-9153), a histamine H3-receptor antagonist, on learning and memory, and on cholinergic and monoaminergic systems in mice. Life Sci 1997, 61: 355-61.
    • (1997) Life Sci , vol.61 , pp. 355-361
    • Miyazaki, S.1    Onodera, K.2    Imaizumi, M.3    Timmerman, H.4
  • 25
    • 0036076825 scopus 로고    scopus 로고
    • Behavioral characterization of mice lacking histamine H(3) receptors
    • Toyota, H., Dugovic, C., Koehl, M. et al. Behavioral characterization of mice lacking histamine H(3) receptors. Mol Pharmacol 2002, 62: 389-97.
    • (2002) Mol Pharmacol , vol.62 , pp. 389-397
    • Toyota, H.1    Dugovic, C.2    Koehl, M.3
  • 27
    • 0031858013 scopus 로고    scopus 로고
    • Therapeutic potential of histamine H3 receptor agonists and antagonists
    • Leurs, R., Blandina, P., Tedford, C., Timmerman, H. Therapeutic potential of histamine H3 receptor agonists and antagonists. Trends Pharmacol Sci 1998, 19: 177-83.
    • (1998) Trends Pharmacol Sci , vol.19 , pp. 177-183
    • Leurs, R.1    Blandina, P.2    Tedford, C.3    Timmerman, H.4
  • 29
    • 0030574248 scopus 로고    scopus 로고
    • Inhibition of histamine versus acetylcholine metabolism as a mechanism of tacrine activity
    • Morisset, S., Traiffort, E., Schwartz, J.C. inhibition of histamine versus acetylcholine metabolism as a mechanism of tacrine activity. Eur J Pharmacol 1996, 315: R1-R2.
    • (1996) Eur J Pharmacol , vol.315
    • Morisset, S.1    Traiffort, E.2    Schwartz, J.C.3
  • 30
    • 0024818025 scopus 로고
    • Correlation of brain levels of 9-amino-1,2,3,4-tetrahydroacridine (THA) with neurochemical and behavioral changes
    • Nielsen, J.A., Mena, E.E., Williams, I.H., Nocerini, M.R., Liston, D. Correlation of brain levels of 9-amino-1,2,3,4-tetrahydroacridine (THA) with neurochemical and behavioral changes. Eur J Pharmacol 1989, 173: 53-64.
    • (1989) Eur J Pharmacol , vol.173 , pp. 53-64
    • Nielsen, J.A.1    Mena, E.E.2    Williams, I.H.3    Nocerini, M.R.4    Liston, D.5
  • 32
    • 0030061024 scopus 로고    scopus 로고
    • Steady-state pharmacokinetics of tacrine in long-term treatment of Alzheimer's patients
    • Johansson, M., Hellstrom-Lindahl, E., Nordberg, A. Steady-state pharmacokinetics of tacrine in long-term treatment of Alzheimer's patients. Dementia 1996, 7(2): 111-17.
    • (1996) Dementia , vol.7 , Issue.2 , pp. 111-117
    • Johansson, M.1    Hellstrom-Lindahl, E.2    Nordberg, A.3
  • 33
    • 0023848903 scopus 로고
    • Structural features of potent inhibitors of rat kidney histamine N-methyltransferase
    • Harle, D.O., Baldo, B.A. Structural features of potent inhibitors of rat kidney histamine N-methyltransferase. Biochem Pharmacol 1988, 37: 385-8.
    • (1988) Biochem Pharmacol , vol.37 , pp. 385-388
    • Harle, D.O.1    Baldo, B.A.2
  • 34
    • 0037447913 scopus 로고    scopus 로고
    • Imidazole derivatives as a novel class of hybrid compounds with inhibitory histamine N-methyltransferase potencies and histamine hH(3) receptor affinities
    • Grassmann, S., Apelt, J., Sippl, W. et al. Imidazole derivatives as a novel class of hybrid compounds with inhibitory histamine N-methyltransferase potencies and histamine hH(3) receptor affinities. Bioorg Med Chem 2003, 11: 2163-74.
    • (2003) Bioorg Med Chem , vol.11 , pp. 2163-2174
    • Grassmann, S.1    Apelt, J.2    Sippl, W.3
  • 35
    • 0035991580 scopus 로고    scopus 로고
    • Understanding and managing behavioral symptoms in Alzheimer's disease and related dementias: Focus on rivastigmine
    • Robert, P. Understanding and managing behavioral symptoms in Alzheimer's disease and related dementias: Focus on rivastigmine. Curr Med Res Opin 2002, 18: 156-71.
    • (2002) Curr Med Res Opin , vol.18 , pp. 156-171
    • Robert, P.1
  • 37
    • 0031019973 scopus 로고    scopus 로고
    • A risk-benefit assessment oftacrine in the treatment of Alzheimer's disease
    • Samuels, S.C., Davis, K.L. A risk-benefit assessment oftacrine in the treatment of Alzheimer's disease. Drug Saf 1997, 16: 66-77.
    • (1997) Drug Saf , vol.16 , pp. 66-77
    • Samuels, S.C.1    Davis, K.L.2


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.