Synthesis of 3-[1H-imidazol-4-yl] propyl 4-[18F] fluorobenzyl ether ([18F] fluoroproxyfan): A potential radioligand for imaging histamine H3 receptors

Journal of Labelled Compounds and Radiopharmaceuticals

Volumn 43, Issue 9, 2000, Pages 873-882

  Iwata, Ren ^a   Horváth, Géza ^b   Pascali, Claudio ^c   Bogni, A ^c   Yanai, Kazuhiko ^d   Kovács, Zoltán ^e   Ido, Tatsuo ^a  

^a TOHOKU UNIVERSITY   (Japan)

^b UNIVERSITY OF DEBRECEN   (Hungary)

^c NATIONAL CANCER INSTITUTE   (Italy)

^d TOHOKU UNIVERSITY SCHOOL OF MEDICINE   (Japan)

^e INSTITUTE OF NUCLEAR RESEARCH ATOMKI   (Hungary)

Author keywords

Fluorine 18; Fluoroproxyfan; Histamine H3 receptor; PET; Radioligand

Indexed keywords

CHELATION; FLUORINE;

1H-IMIDAZOLE; FLUORINE-18; FLUOROPROXYFAN; HISTAMINE H3 RECEPTOR; HISTAMINES; RADIOCHEMICAL PURITY; RADIOCHEMICAL YIELD; RADIOLIGANDS; RECEPTOR LIGANDS; SILVER TRIFLATE;

ETHERS;

FLUORINE 18; FLUOROPROXYFAN; HISTAMINE H3 RECEPTOR; HISTAMINE H3 RECEPTOR AGONIST; IMIDAZOLE DERIVATIVE; RADIOLIGAND; UNCLASSIFIED DRUG;

ALKYLATION; ARTICLE; DRUG SYNTHESIS; ISOTOPE LABELING; POSITRON EMISSION TOMOGRAPHY;

EID: 17444454357     PISSN: 03624803     EISSN: None     Source Type: Journal    
DOI: 10.1002/1099-1344(200008)43:9<873::AID-JLCR371>3.0.CO;2-A     Document Type: Article

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