Synthesis of [35S]aryl sulfonyl chlorides from [ 35S]elemental sulfur

Journal of Labelled Compounds and Radiopharmaceuticals

Volumn 48, Issue 4, 2005, Pages 275-283

  Wallace, Michael A ^a,b   Raab, Conrad E ^a   Dean, Dennis C ^a   Melillo, David G ^a  

^a MERCK RESEARCH LABORATORIES   (United States)

^b NONE   (United States)

Author keywords

35S alkyl sulfonyl chlorides; 35S aryl sulfonyl chlorides

Indexed keywords

SULFUR;

ALKYL SULFONYL CHLORIDE; ELEMENTAL SULPHUR; GRIGNARD REAGENT; SULFONYL CHLORIDES; SYNTHETIC METHODOLOGY; [35S]ALKYL SULFONYL CHLORIDE; [35S]ARYL SULFONYL CHLORIDE;

CHLORINE COMPOUNDS;

BENZENESULFONAMIDE DERIVATIVE; METHANESULFONAMIDE DERIVATIVE; RADIOLIGAND; SULFONAMIDE; SULFONYL CHLORIDE S 35; SULFUR 35; SULFUR DERIVATIVE; UNCLASSIFIED DRUG;

ARTICLE; CHEMICAL REACTION; CHEMICAL STRUCTURE; HIGH PERFORMANCE LIQUID CHROMATOGRAPHY; OXIDATION; SYNTHESIS;

EID: 17444412614     PISSN: 03624803     EISSN: None     Source Type: Journal    
DOI: 10.1002/jlcr.920     Document Type: Article

References (9)

1. Dean DC, Nargund R, Pong SS, Chaung L, Griffin P, Melillo D, Ellsworth R, Van Der Ploeg L, Patchett A, Smith R. J Med Chem 1996; 39: 1767-1770; Kale T, Raab C, Yu N, Dean D, Distefano M. J Am Chem Soc 2001; 123: 4373-4381; Kale T, Raab C, Yu N, Aquino A, Dean D, Distefano M. J Label Compd Radiopharm 2003; 46: 29-54.
2. Dean DC, Nargund R, Pong SS, Chaung L, Griffin P, Melillo D, Ellsworth R, Van Der Ploeg L, Patchett A, Smith R. J Med Chem 1996; 39: 1767-1770; Kale T, Raab C, Yu N, Dean D, Distefano M. J Am Chem Soc 2001; 123: 4373-4381; Kale T, Raab C, Yu N, Aquino A, Dean D, Distefano M. J Label Compd Radiopharm 2003; 46: 29-54.
3. Dean DC, Nargund R, Pong SS, Chaung L, Griffin P, Melillo D, Ellsworth R, Van Der Ploeg L, Patchett A, Smith R. J Med Chem 1996; 39: 1767-1770; Kale T, Raab C, Yu N, Dean D, Distefano M. J Am Chem Soc 2001; 123: 4373-4381; Kale T, Raab C, Yu N, Aquino A, Dean D, Distefano M. J Label Compd Radiopharm 2003; 46: 29-54.
4. Pepinsky R, Mumford R, Chen L, Leone D, Amo S, Riper G, Whitty A, Dolinski B, Lobb R, Dean D, Chang L, Raab C, Si Q, Hagmann W, Lingham R. Biochemistry 2002; 41: 7125-7141; Egger L, Cao J, McCallum C, Kidambi U, Riper G, McCauley E, Mumford R, Lanza T, Lin L, de Laszlo S, Young D, Yang G, Dean D, Raab C, Wallace M, Jones A, Hagmann W, Schmidt J, Pepinsky R, Scott D, Lee WC, Cornebise M, Detmers P. J Pharmacol Exp Ther 2003; 306: 903-913.
5. Pepinsky R, Mumford R, Chen L, Leone D, Amo S, Riper G, Whitty A, Dolinski B, Lobb R, Dean D, Chang L, Raab C, Si Q, Hagmann W, Lingham R. Biochemistry 2002; 41: 7125-7141; Egger L, Cao J, McCallum C, Kidambi U, Riper G, McCauley E, Mumford R, Lanza T, Lin L, de Laszlo S, Young D, Yang G, Dean D, Raab C, Wallace M, Jones A, Hagmann W, Schmidt J, Pepinsky R, Scott D, Lee WC, Cornebise M, Detmers P. J Pharmacol Exp Ther 2003; 306: 903-913.
6. van Leusen AM, Hundscheid FJ, Tandon VK, Rouwette P. Tetrahedron 1987; 43: 5073-5088; Tercio J, Ferreria B, Catani V, Comasseto JV. Synthesis 1987; 2: 149-153.
7. van Leusen AM, Hundscheid FJ, Tandon VK, Rouwette P. Tetrahedron 1987; 43: 5073-5088; Tercio J, Ferreria B, Catani V, Comasseto JV. Synthesis 1987; 2: 149-153.
8. Park YJ, Shin HH, Kim YH. Chem Lett 1992; 8: 1483-1486.
9. Mallon JM, Bebb RL. Chem Rev 1969; 69: 693-755.