Synthesis and biological activity of a novel squalene epoxidase inhibitor, FR194738

Bioorganic and Medicinal Chemistry Letters

Volumn 14, Issue 3, 2004, Pages 633-637

  Sawada, Masae ^a   Washizuka, Ken Ichi ^a   Okumura, Hiroyuki ^a  

^a ASTELLAS PHARMA INC   (Japan)

Author keywords

[No Author keywords available]

Indexed keywords

CHOLESTEROL; ENZYME INHIBITOR; FR 194738; HYPOCHOLESTEROLEMIC AGENT; SQUALENE MONOOXYGENASE; TRIACYLGLYCEROL;

ANIMAL CELL; ANIMAL EXPERIMENT; ARTICLE; CHOLESTEROL BLOOD LEVEL; CHOLESTEROL SYNTHESIS; CONCENTRATION (PARAMETERS); CONTROLLED STUDY; DRUG ACTIVITY; DRUG POTENCY; DRUG STRUCTURE; DRUG SYNTHESIS; HUMAN; HUMAN CELL; IN VITRO STUDY; MALE; NONHUMAN; RAT; TRIACYLGLYCEROL BLOOD LEVEL;

CANIS FAMILIARIS;

EID: 1642534340     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2003.11.072     Document Type: Article

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